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25 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
28435528 24 Discovery of Highly Selective Inhibitors of the Immunoproteasome Low Molecular Mass Polypeptide 2 (LMP2) Subunit.EBI Kezar Life Sciences
25006746 85 Structure-based design of฿1i or฿5i specific inhibitors of human immunoproteasomes.EBI Leiden Institute of Chemistry and Netherlands Proteomics Centre
24524217 65 Structurally novel highly potent proteasome inhibitors created by the structure-based hybridization of nonpeptidic belactosin derivatives and peptide boronates.EBI Hokkaido University
32189500 56 LMP2 Inhibitors as a Potential Treatment for Alzheimer's Disease.EBI University of Kentucky
27563406 128 Discovery of Fluoromethylketone-Based Peptidomimetics as Covalent ATG4B (Autophagin-1) Inhibitors.EBI Roche Pharma Research and Early Development
30639896 42 Covalent docking modelling-based discovery of tripeptidyl epoxyketone proteasome inhibitors composed of aliphatic-heterocycles.EBI Hangzhou Institute of Innovative Medicine
30611983 48 Exploration of novel macrocyclic dipeptide N-benzyl amides as proteasome inhibitors.EBI Zhejiang University
30380863 196 Required Immunoproteasome Subunit Inhibition Profile for Anti-Inflammatory Efficacy and Clinical Candidate KZR-616 ((2 S,3 R)- N-(( S)-3-(Cyclopent-1-en-1-yl)-1-(( R)-2-methyloxiran-2-yl)-1-oxopropan-2-yl)-3-hydroxy-3-(4-methoxyphenyl)-2-(( S)-2-(2-morpholinoacetamido)propanamido)propenamide).EBI Kezar Life Sciences
31521028 67 Immunoproteasome-selective inhibitors: An overview of recent developments as potential drugs for hematologic malignancies and autoimmune diseases.EBI Hangzhou Xixi Hospital
30964987 13 Development of Novel Epoxyketone-Based Proteasome Inhibitors as a Strategy To Overcome Cancer Resistance to Carfilzomib and Bortezomib.EBI University of Kentucky
30587447 3 Analysis of chain length, substitution patterns, and unsaturation of AM-404 derivatives as 20S proteasome stimulators.EBI Purdue University
30657666 263 Structure-Based Design of Inhibitors Selective for Human Proteasome ?2c or ?2i Subunits.EBI Leiden Institute of Chemistry and Netherlands Proteomics Centre
31801019 5 Novel Cell-Penetrating Peptide Conjugated Proteasome Inhibitors: Anticancer and Antifungal Investigations.EBI University of Auckland
30455150 10 Tetradehydrohalicyclamine B, a new proteasome inhibitor from the marine sponge Acanthostrongylophora ingens.EBI Kumamoto University
17249727 8 Cinnabaramides A-G: analogues of lactacystin and salinosporamide from a terrestrial streptomycete.EBI Intermed Discovery Gmbh (Imd)
15780623 39 Structure-based design of derivatives of tyropeptin A as the potent and selective inhibitors of mammalian 20S proteasome.EBI Numazu Bio-Medical Research Institute
7608891 7 Potent inhibitors of proteasome.EBI Cephalon
11992770 19 Structure-based optimisation of 2-aminobenzylstatine derivatives: potent and selective inhibitors of the chymotrypsin-like activity of the human 20S proteasome.EBI Novartis Pharma
29339252 124 Structure-based design of human immuno- and constitutive proteasomes inhibitors.EBI Universit£
29652143 22 Reviewing Hit Discovery Literature for Difficult Targets: Glutathione Transferase Omega-1 as an Example.EBI Monash University