The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
27774126 |
95 |
Exploring |
University of California San Francisco |
23562062 |
4 |
Arylsulfonamide pyrimidines as VLA-4 antagonists. |
Elan Pharmaceuticals |
17387018 |
74 |
Discovery of +(2-{4-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethoxy]phenyl}-cyclopropyl)acetic acid as potent and selective alphavbeta3 inhibitor: design, synthesis, and optimization. |
Pfizer |
16298127 |
80 |
Convergent, parallel synthesis of a series of beta-substituted 1,2,4-oxadiazole butanoic acids as potent and selective alpha(v)beta3 receptor antagonists. |
Pfizer |
15006384 |
179 |
Synthesis of cinnamic acids and related isosteres as potent and selective alpha v beta 3 receptor antagonists. |
Pfizer |
14698164 |
39 |
Synthesis and biological evaluation of nonpeptide integrin antagonists containing spirocyclic scaffolds. |
Pharmaceutical Research Institute |
31999923 |
16 |
Insights into Protein-Ligand Interactions in Integrin Complexes: Advances in Structure Determinations. |
Pliant Therapeutics |
10406646 |
15 |
Orally bioavailable nonpeptide vitronectin receptor antagonists with efficacy in an osteoporosis model. |
Smithkline Beecham Pharmaceuticals |
31381331 |
70 |
Profile of a Highly Selective Quaternized Pyrrolidine Betaine ? |
Glaxosmithkline Medicines Research Centre |
24568695 |
76 |
Strategies to inhibit tumor associated integrin receptors: rationale for dual and multi-antagonists. |
University of Bradford |
30215258 |
228 |
Discovery of ( S)-3-(3-(3,5-Dimethyl-1 H-pyrazol-1-yl)phenyl)-4-(( R)-3-(2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl)pyrrolidin-1-yl)butanoic Acid, a Nonpeptidic ? |
University of Strathclyde |