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15 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
27774126 95 ExploringEBI University of California San Francisco
23562062 4 Arylsulfonamide pyrimidines as VLA-4 antagonists.EBI Elan Pharmaceuticals
17387018 74 Discovery of +(2-{4-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethoxy]phenyl}-cyclopropyl)acetic acid as potent and selective alphavbeta3 inhibitor: design, synthesis, and optimization.EBI Pfizer
16298127 80 Convergent, parallel synthesis of a series of beta-substituted 1,2,4-oxadiazole butanoic acids as potent and selective alpha(v)beta3 receptor antagonists.EBI Pfizer
15006384 179 Synthesis of cinnamic acids and related isosteres as potent and selective alpha v beta 3 receptor antagonists.EBI Pfizer
14698164 39 Synthesis and biological evaluation of nonpeptide integrin antagonists containing spirocyclic scaffolds.EBI Pharmaceutical Research Institute
31999923 16 Insights into Protein-Ligand Interactions in Integrin Complexes: Advances in Structure Determinations.EBI Pliant Therapeutics
10406646 15 Orally bioavailable nonpeptide vitronectin receptor antagonists with efficacy in an osteoporosis model.EBI Smithkline Beecham Pharmaceuticals
31381331 70 Profile of a Highly Selective Quaternized Pyrrolidine Betaine ?EBI Glaxosmithkline Medicines Research Centre
24568695 76 Strategies to inhibit tumor associated integrin receptors: rationale for dual and multi-antagonists.EBI University of Bradford
30215258 228 Discovery of ( S)-3-(3-(3,5-Dimethyl-1 H-pyrazol-1-yl)phenyl)-4-(( R)-3-(2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl)pyrrolidin-1-yl)butanoic Acid, a Nonpeptidic ?EBI University of Strathclyde