The following articles (labelled with PubMed ID or TBD) are for your review
| PMID | Data | Article Title | Organization |
|---|
| 28254377 |
3 |
Impact of androstane A- and D-ring inversion on 17ß-hydroxysteroid dehydrogenase type 3 inhibitory activity, androgenic effect and metabolic stability. |
Chu De Qu£Bec-Research Center |
| 24960438 |
24 |
Ligand-based pharmacophore modeling and virtual screening for the discovery of novel 17ß-hydroxysteroid dehydrogenase 2 inhibitors. |
University of Innsbruck |
| 22691057 |
32 |
Discovery of a potent, selective, and orally bioavailable acidic 11ß-hydroxysteroid dehydrogenase type 1 (11ß-HSD1) inhibitor: discovery of 2-[(3S)-1-[5-(cyclohexylcarbamoyl)-6-propylsulfanylpyridin-2-yl]-3-piperidyl]acetic acid (AZD4017). |
Astrazeneca |
| 22512907 |
49 |
Discovery of potent and orally bioavailable 17ß-hydroxysteroid dehydrogenase type 3 inhibitors. |
Sumitomo Chemical |
| 16078844 |
18 |
Androsterone 3alpha-ether-3beta-substituted and androsterone 3beta-substituted derivatives as inhibitors of type 3 17beta-hydroxysteroid dehydrogenase: chemical synthesis and structure-activity relationship. |
Chuq-Pavillon Chul and Universit£ |
| 11806715 |
13 |
Synthesis and optimization of a new family of type 3 17 beta-hydroxysteroid dehydrogenase inhibitors by parallel liquid-phase chemistry. |
Centre Hospitalier Universitaire De Qu£Bec and Universit£ |
| 11086723 |
12 |
Androsterone 3beta-substituted derivatives as inhibitors of type 3 17beta-hydroxysteroid dehydrogenase. |
Laval University |
| 22137341 |
10 |
Identification of oxazolidinediones and thiazolidinediones as potent 17ß-hydroxysteroid dehydrogenase type 3 inhibitors. |
Sumitomo Chemical |
| 21741247 |
2 |
Development of 3-substituted-androsterone derivatives as potent inhibitors of 17ß-hydroxysteroid dehydrogenase type 3. |
Chuq (Chul)-Research Center |
| 20346654 |
16 |
Curcumin derivatives inhibit testicular 17beta-hydroxysteroid dehydrogenase 3. |
School of Pharmacy |
| 19954971 |
40 |
Coumarins as novel 17beta-hydroxysteroid dehydrogenase type 3 inhibitors for potential treatment of prostate cancer. |
Sumitomo Chemical |
| 16797984 |
12 |
Synthesis, biochemical evaluation and rationalisation of the inhibitory activity of a series of 4-hydroxyphenyl ketones as potential inhibitors of 17beta-hydroxysteroid dehydrogenase type 3 (17beta-HSD3). |
Kingston University |
| 16386902 |
87 |
Identification of a novel series of tetrahydrodibenzazocines as inhibitors of 17beta-hydroxysteroid dehydrogenase type 3. |
Bristol-Myers Squibb Pharmaceutical Research Institute |
| 31268309 |
17 |
A- and D-Ring Structural Modifications of an Androsterone Derivative Inhibiting 17?-Hydroxysteroid Dehydrogenase Type 3: Chemical Synthesis and Structure-Activity Relationships. |
Chu De Queb£C-Research Center |
| 27025340 |
3 |
Synthesis of a dansyl-labeled inhibitor of 17?-hydroxysteroid dehydrogenase type 3 for optical imaging. |
Chu De Qu£Bec-Research Center |
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