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12 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
15771450 42 Synthesis of new benzoxazinone derivatives as neuropeptide Y5 antagonists for the treatment of obesity.EBI Laboratorios Dr. Esteve
21924902 43 5-(2'-Pyridyl)-2-aminothiazoles: alkyl amino sulfonamides and sulfamides as potent NPY(5) antagonists.EBI Lundbeck Research Usa
21782428 61 Discovery of Lu AA33810: a highly selective and potent NPY5 antagonist with in vivo efficacy in a model of mood disorder.EBI Lundbeck Research Usa
19720539 32 Discovery of trans-N-[1-(2-fluorophenyl)-3-pyrazolyl]-3-oxospiro[6-azaisobenzofuran-1(3H),1'-cyclohexane]-4'-carboxamide, a potent and orally active neuropeptide Y Y5 receptor antagonist.EBI Tsukuba Research Institute
19464889 43 Aryl urea derivatives of spiropiperidines as NPY Y5 receptor antagonists.EBI Tsukuba Research Institute
15109631 86 Discovery and SAR of potent, orally available and brain-penetrable 5,6-dihydro-4H-3-thia-1-aza-benzo[e]azulen- and 4,5-dihydro-6-oxa-3-thia-1-aza-benzo[e]azulen derivatives as neuropeptide Y Y5 receptor antagonists.EBI Novartis Pharma
12593645 2 In vitro and in vivo characterization of 3-[2-[6-(2-tert-butoxyethoxy)pyridin-3-yl]-1H-imidazol-4-yl]benzonitrile hydrochloride salt, a potent and selective NPY5 receptor antagonist.EBI Pfizer
12139462 34 Discovery and optimization of a series of carbazole ureas as NPY5 antagonists for the treatment of obesity.EBI Astrazeneca
12067557 24 Discovery of potent and selective small molecule NPY Y5 receptor antagonists.EBI Lundbeck Research Usa
10866375 50 Design, synthesis and SAR of a series of 2-substituted 4-amino-quinazoline neuropeptide Y Y5 receptor antagonists.EBI Novartis Pharma
9925722 18 Pharmacological treatment of obesity: therapeutic strategies.EBI The R. W. Johnson Pharmaceutical Research Institute