The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
27774128 |
38 |
Discovery of ONO-7300243 from a Novel Class of Lysophosphatidic Acid Receptor 1 Antagonists: From Hit to Lead. |
Ono Pharmaceutical |
25746814 |
80 |
Discovery of novel S1P2 antagonists. Part 1: discovery of 1,3-bis(aryloxy)benzene derivatives. |
Ono Pharmaceutical |
25100502 |
15 |
Design and synthesis of sulfamoyl benzoic acid analogues with subnanomolar agonist activity specific to the LPA2 receptor. |
The University of Tennessee Health Science Center |
23395664 |
66 |
Phosphorothioate analogs of sn-2 radyl lysophosphatidic acid (LPA): metabolically stabilized LPA receptor agonists. |
The University of Utah |
22801643 |
6 |
Selective non-lipid modulator of LPA5 activity in human platelets. |
Sanofi-Aventis Deutschland |
18178086 |
26 |
Discovery of potent LPA2 (EDG4) antagonists as potential anticancer agents. |
Amgen |
17379528 |
30 |
Synthesis and SAR studies of a novel class of S1P1 receptor antagonists. |
Sankyo |
19800804 |
19 |
Structure-based drug design identifies novel LPA3 antagonists. |
The University of Memphis |
18467108 |
26 |
Identification of non-lipid LPA3 antagonists by virtual screening. |
The University of Memphis |
16913720 |
15 |
Phosphonothioate and fluoromethylene phosphonate analogues of cyclic phosphatidic acid: Novel antagonists of lysophosphatidic acid receptors. |
The University of Utah |
16290140 |
54 |
Identification of Darmstoff analogs as selective agonists and antagonists of lysophosphatidic acid receptors. |
University of Tennessee Health Science Center |
16263282 |
43 |
Synthesis and pharmacological evaluation of second-generation phosphatidic acid derivatives as lysophosphatidic acid receptor ligands. |
University of Tennessee Health Science Center |
16033271 |
81 |
Synthesis, structure-activity relationships, and biological evaluation of fatty alcohol phosphates as lysophosphatidic acid receptor ligands, activators of PPARgamma, and inhibitors of autotaxin. |
University of Tennessee Health Science Center |
15177461 |
140 |
Selecting against S1P3 enhances the acute cardiovascular tolerability of 3-(N-benzyl)aminopropylphosphonic acid S1P receptor agonists. |
Merck Research Laboratories |
15177455 |
27 |
Synthesis and biological evaluation of phosphonic and thiophosphoric acid derivatives of lysophosphatidic acid. |
Oxford University |