The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
26393374 |
34 |
Improving the Selectivity of Engineered Protease Inhibitors: Optimizing the P2 Prime Residue Using a Versatile Cyclic Peptide Library. |
Queensland University of Technology |
24211642 |
49 |
Identification by in silico and in vitro screenings of small organic molecules acting as reversible inhibitors of kallikreins. |
Universit£ |
23849879 |
23 |
1,2,4-Triazole derivatives as transient inactivators of kallikreins involved in skin diseases. |
Universit£ |
30691925 |
34 |
Kallikrein 5 inhibitors identified through structure based drug design in search for a treatment for Netherton Syndrome. |
Glaxosmithkline R&D |
31521475 |
205 |
Design and development of a series of borocycles as selective, covalent kallikrein 5 inhibitors. |
Glaxosmithkline |
31005442 |
64 |
Structure guided drug design to develop kallikrein 5 inhibitors to treat Netherton syndrome. |
Glaxosmithkline R&D |
30888159 |
18 |
Amino Acid Scanning at P5' within the Bowman-Birk Inhibitory Loop Reveals Specificity Trends for Diverse Serine Proteases. |
The University of Queensland |
30613336 |
32 |
Potent, Selective, and Cell-Penetrating Inhibitors of Kallikrein-Related Peptidase 4 Based on the Cyclic Peptide MCoTI-II. |
The University of Queensland |
30212625 |
107 |
Depsipeptides Featuring a Neutral P1 Are Potent Inhibitors of Kallikrein-Related Peptidase 6 with On-Target Cellular Activity. |
German Cancer Research Center (Dkfz) |
29517911 |
87 |
Stable and Long-Lasting, Novel Bicyclic Peptide Plasma Kallikrein Inhibitors for the Treatment of Diabetic Macular Edema. |
Bicycle Therapeutics |