BDBM100703 US8507676, 51-R::US8507676, 51-S
SMILES: CC(c1cnc2ccc(nn12)C(\C)=N\OCCO)c1c(F)cc2n(C)ncc2c1F
InChI Key: InChIKey=FSGDBTOPVQONBI-RPPGKUMJSA-N
Data: 2 IC50
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Hepatocyte growth factor receptor (Homo sapiens (Human)) | BDBM100703![]() (US8507676, 51-R | US8507676, 51-S) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 460 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-... | US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hepatocyte growth factor receptor (Homo sapiens (Human)) | BDBM100703![]() (US8507676, 51-R | US8507676, 51-S) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 2.80 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis AG US Patent | Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-... | US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9 | |||||||||||
More data for this Ligand-Target Pair |