BDBM119464 US8680120, 25-12
SMILES: COc1ccc2n(Cc3csc(n3)C(O)=O)c(cc2c1)-c1ccccc1
InChI Key: InChIKey=UGVGPIXOUUXAAC-UHFFFAOYSA-N
Data: 1 IC50
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Prostanoid EP1 receptor (Rattus norvegicus (Rat)) | BDBM119464 (US8680120, 25-12) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 55 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Co., Ltd. US Patent | Assay Description The rat EP1 receptor-expressing cells were washed with the assay buffer. 100 μL of a fluorescent calcium indicator (Calcium kit II, Fluo 4 (Doji... | US Patent US8680120 (2014) BindingDB Entry DOI: 10.7270/Q2183554 | |||||||||||
More data for this Ligand-Target Pair |