BDBM119482 US8680120, 25-42
SMILES: COc1cc2cc(-c3cccnc3)n(Cc3cccc(n3)C(O)=O)c2cc1Cl
InChI Key: InChIKey=MZBDRQVEULUYPF-UHFFFAOYSA-N
Data: 1 IC50
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Prostaglandin E2 receptor EP1 subtype (Rattus norvegicus (Rat)) | BDBM119482 (US8680120, 25-42) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 28 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Co., Ltd. US Patent | Assay Description The rat EP1 receptor-expressing cells were washed with the assay buffer. 100 μL of a fluorescent calcium indicator (Calcium kit II, Fluo 4 (Doji... | US Patent US8680120 (2014) BindingDB Entry DOI: 10.7270/Q2183554 | |||||||||||
More data for this Ligand-Target Pair |