null
SMILES: COc1ccccc1CNc1ncnc2cc(N)ncc12
InChI Key: InChIKey=UIKUPKYKBYMHFU-UHFFFAOYSA-N
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM3341 (4-N-[(2-methoxyphenyl)methyl]pyrido[4,3-d]pyrimidi...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Auckland | Assay Description IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe... | J Med Chem 38: 3780-8 (1995) Article DOI: 10.1021/jm00019a007 BindingDB Entry DOI: 10.7270/Q2Z899M8 | |||||||||||
More data for this Ligand-Target Pair |