null
SMILES: CC1(CC1)NS(=O)(=O)c1ccc2CCN(C(=O)CN3CCNC3=O)c2c1
InChI Key: InChIKey=QYQULHAWPZDXII-UHFFFAOYSA-N
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Poly(ADP-ribose) glycohydrolase (Homo sapiens (Human)) | BDBM421430 (N-(1-Methylcyclopropyl)-1-[2-(2-oxoimidazolidin-1-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 5.23E+3 | n/a | n/a | n/a | n/a |
Cancer Research Technology Limited US Patent | Assay Description PARG In vitro assays were conducted in a total volume of 15 ul in a standard 384 well format. 5 ul of Human Full Length PARG (Produced internally by ... | US Patent US10995073 (2021) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Poly(ADP-ribose) glycohydrolase (Homo sapiens (Human)) | BDBM421430 (N-(1-Methylcyclopropyl)-1-[2-(2-oxoimidazolidin-1-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 5.23E+3 | n/a | n/a | n/a | n/a |
Cancer Research Technology Limited US Patent | Assay Description PARG In vitro assays were conducted in a total volume of 15 ul in a standard 384 well format. 5 ul of Human Full Length PARG (Produced internally by ... | US Patent US10508086 (2019) BindingDB Entry DOI: 10.7270/Q26112QF | |||||||||||
More data for this Ligand-Target Pair |