null
SMILES: Cc1ccc(o1)C(=O)Nc1cc(ccc1N1CCN(Cc2ccco2)CC1)C(F)(F)F
InChI Key: InChIKey=XRHFXIQYYDGMMC-UHFFFAOYSA-N
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
SRSF protein kinase 1 (Homo sapiens (Human)) | BDBM448548 (5-methyl-N-(2-(4-((furan-2-yl)methyl)piperazin-1-y...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | 17.6 | n/a | n/a | n/a | n/a | n/a | n/a |
Exonate Limited US Patent | Assay Description Screening of a series of molecules identified compounds (Compounds 5, 8, 16 to 18 and 43 of Table 3) that had improved potency against SRPK1 against ... | US Patent US10696661 (2020) | |||||||||||
More data for this Ligand-Target Pair |