BDBM466546 US10799518, Compound 14::rel-(2R,3 S)-3-[(4- brornophenyl)carbarnoyl]spiro [bicyclo[2.2.1]heptane-7,1'- cyclopropane]-2-carboxylic acid
SMILES: OC(=O)C1C2CCC(C1C(=O)Nc1ccc(Br)cc1)C21CC1
InChI Key: InChIKey=CVTBABUFIBCHCY-UHFFFAOYSA-N
Data: 1 EC50
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
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N-formyl peptide receptor 2 (Homo sapiens (Human)) | BDBM466546![]() (US10799518, Compound 14 | rel-(2R,3 S)-3-[(4- bror...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 4 | n/a | n/a | n/a | n/a |
ALLERGAN, INC. US Patent | Assay Description HEK-Gα16 cells stably expressing the human FPR2 receptor was utilized. Cells were plated into 384-well poly-D-lysine coated plates at a density ... | US Patent US10799518 (2020) | |||||||||||
More data for this Ligand-Target Pair |