null
SMILES: Cc1ccc(C[C@H](NC(=O)c2ccccc2)C(=O)Nc2cccc3c(cccc23)S(=O)(=O)NC(C)(C)C)cc1
InChI Key: InChIKey=XJZDZBZJPVLTAP-MHZLTWQESA-N
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Ubiquitin carboxyl-terminal hydrolase 30 (Homo sapiens (Human)) | BDBM490023![]() ((S)-N-(1-((5-(N-(tert- butyl)sulfamoyl)naphthalen-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ubiquitin carboxyl-terminal hydrolase 30 (Homo sapiens (Human)) | BDBM490023![]() ((S)-N-(1-((5-(N-(tert- butyl)sulfamoyl)naphthalen-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | US Patent | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Mitobridge, Inc. US Patent | Assay Description The in vitro assay for USP30 evaluates the ability of a test compound to inhibit the activity of the enzyme to cleave ubiquitin from a substrate. Ubi... | US Patent US10968172 (2021) | |||||||||||
More data for this Ligand-Target Pair |