BDBM50133913 CHEMBL343517::Dimethyl-[3-(10-methyl-benzo[c]phenothiazin-7-yl)-propyl]-amine
SMILES: CN(C)CCCN1c2ccc(C)cc2Sc2c1ccc1ccccc21
InChI Key: InChIKey=ZWVAIFKVPKWGLE-UHFFFAOYSA-N
Data: 1 KI
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
D(3) dopamine receptor (Homo sapiens (Human)) | BDBM50133913 (CHEMBL343517 | Dimethyl-[3-(10-methyl-benzo[c]phen...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 1.42E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Michigan Curated by ChEMBL | Assay Description Ability to compete with [3H]YM-09151-2 binding to the human dopamine receptor D3 transfected in CHO cells | J Med Chem 46: 4377-92 (2003) Article DOI: 10.1021/jm030085p BindingDB Entry DOI: 10.7270/Q21V5FPS | |||||||||||
More data for this Ligand-Target Pair |