Found 4 hits for monomerid = 50202530 Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
cAMP-specific 3',5'-cyclic phosphodiesterase 4D
(Homo sapiens (Human)) | BDBM50202530
(9-cyclopentyl-5,6-dihydro-7-ethyl-3-(3-pyridyl)-9H...)Show InChI InChI=1S/C19H22N6/c1-2-16-15-9-11-24-18(13-6-5-10-20-12-13)21-22-19(24)17(15)25(23-16)14-7-3-4-8-14/h5-6,10,12,14H,2-4,7-9,11H2,1H3 | PDB
KEGG
UniProtKB/SwissProt UniProtKB/TrEMBL
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| n/a | n/a | 70 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development
Curated by ChEMBL
| Assay Description Inhibition of human recombinant PDE4D |
J Med Chem 50: 344-9 (2007)
Article DOI: 10.1021/jm060904g BindingDB Entry DOI: 10.7270/Q2K0753Z |
More data for this Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4B
(Homo sapiens (Human)) | BDBM50202530
(9-cyclopentyl-5,6-dihydro-7-ethyl-3-(3-pyridyl)-9H...)Show InChI InChI=1S/C19H22N6/c1-2-16-15-9-11-24-18(13-6-5-10-20-12-13)21-22-19(24)17(15)25(23-16)14-7-3-4-8-14/h5-6,10,12,14H,2-4,7-9,11H2,1H3 | PDB
UniProtKB/SwissProt UniProtKB/TrEMBL
antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| n/a | n/a | 210 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development
Curated by ChEMBL
| Assay Description Inhibition of human recombinant PDE4B |
J Med Chem 50: 344-9 (2007)
Article DOI: 10.1021/jm060904g BindingDB Entry DOI: 10.7270/Q2K0753Z |
More data for this Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4C isoform 1
(Homo sapiens (Human)) | BDBM50202530
(9-cyclopentyl-5,6-dihydro-7-ethyl-3-(3-pyridyl)-9H...)Show InChI InChI=1S/C19H22N6/c1-2-16-15-9-11-24-18(13-6-5-10-20-12-13)21-22-19(24)17(15)25(23-16)14-7-3-4-8-14/h5-6,10,12,14H,2-4,7-9,11H2,1H3 | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| n/a | n/a | 700 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development
Curated by ChEMBL
| Assay Description Inhibition of human recombinant PDE4C |
J Med Chem 50: 344-9 (2007)
Article DOI: 10.1021/jm060904g BindingDB Entry DOI: 10.7270/Q2K0753Z |
More data for this Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4A
(Homo sapiens (Human)) | BDBM50202530
(9-cyclopentyl-5,6-dihydro-7-ethyl-3-(3-pyridyl)-9H...)Show InChI InChI=1S/C19H22N6/c1-2-16-15-9-11-24-18(13-6-5-10-20-12-13)21-22-19(24)17(15)25(23-16)14-7-3-4-8-14/h5-6,10,12,14H,2-4,7-9,11H2,1H3 | PDB MMDB
KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| n/a | n/a | 250 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development
Curated by ChEMBL
| Assay Description Inhibition of human recombinant PDE4A |
J Med Chem 50: 344-9 (2007)
Article DOI: 10.1021/jm060904g BindingDB Entry DOI: 10.7270/Q2K0753Z |
More data for this Ligand-Target Pair | |