null
SMILES: Fc1ccc(NC(=O)N[C@H]2[C@@H](CNC2=O)c2c(F)cc(cc2F)C#N)cc1
InChI Key:
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
fMet-Leu-Phe receptor (Homo sapiens (Human)) | BDBM50559825 (CHEMBL4758129) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 4.00E+4 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at human FPR1 expressed in HEK 293 cells co-expressing Galpha15 measured every 1.5 sec for 80 sec by Fluo-4 NW staining based scanni... | Citation and Details Article DOI: 10.1021/acs.jmedchem.9b02101 BindingDB Entry DOI: 10.7270/Q2V98CSC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
N-formyl peptide receptor 2 (Homo sapiens (Human)) | BDBM50559825 (CHEMBL4758129) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 9.70 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at human FPR2 expressed in HEK 293 cells co-expressing Galpha15 measured every 1.5 sec for 80 sec by Fluo-4 NW staining based scanni... | Citation and Details Article DOI: 10.1021/acs.jmedchem.9b02101 BindingDB Entry DOI: 10.7270/Q2V98CSC | |||||||||||
More data for this Ligand-Target Pair |