null
SMILES: C[C@@H](COc1ccc(F)c(c1)C(O)=O)Oc1ccc(C(=O)CC(C)(C)C)c(O)c1C
InChI Key:
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Metabotropic glutamate receptor 2 (Rattus norvegicus) | BDBM50576825 (CHEMBL4862778) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 257 | n/a | n/a | n/a | n/a |
TBA | Assay Description Positive allosteric modulator activity at rat mGlu2 receptor transfected in GIRK channel overexpressing cells assessed as potentiation of glutamate-i... | Citation and Details Article DOI: 10.1016/j.bmcl.2021.128342 BindingDB Entry DOI: 10.7270/Q22F7S71 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 3 (Rattus norvegicus (Rat)) | BDBM50576825 (CHEMBL4862778) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.12E+3 | n/a | n/a | n/a | n/a |
TBA | Assay Description Positive allosteric modulator activity at rat mGlu3 receptor transfected in GIRK channel overexpressing cells assessed as potentiation of glutamate-i... | Citation and Details Article DOI: 10.1016/j.bmcl.2021.128342 BindingDB Entry DOI: 10.7270/Q22F7S71 | |||||||||||
More data for this Ligand-Target Pair |