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null

SMILES: COc1cc(ccc1-c1cn(C\C=C\C)c(=O)c2[nH]ccc12)C(C)(C)O

InChI Key:

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 47 hits for monomerid = 50615275
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Bromodomain-containing protein 9 (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	UniChem	n/a	n/a	48	n/a	n/a	n/a	n/a	n/a	n/a
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Platelet-derived growth factor receptor alpha/beta (Mus musculus (mouse))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	MMDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet	UniChem	n/a	n/a	4.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
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Bromodomain-containing protein 4 (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	UniChem	n/a	n/a	>2.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
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Chromatin remodeling regulator CECR2 (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	UniChem	n/a	n/a	>2.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
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Transcription initiation factor TFIID subunit 1 (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	UniChem	n/a	n/a	>2.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
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Bromodomain-containing protein 9 (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	n/a	190	n/a	n/a	n/a	n/a
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Stromelysin-3 (Mus musculus)	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	UniChem	n/a	n/a	1.02E+4	n/a	n/a	n/a	n/a	n/a	n/a
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ATPase family AAA domain-containing protein 2 (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
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ATPase family AAA domain-containing protein 2B (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
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Bromodomain adjacent to zinc finger domain protein 2A (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
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Bromodomain adjacent to zinc finger domain protein 2B (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
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Bromodomain-containing protein 1 (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
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Bromodomain-containing protein 2 (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	2.70E+3	n/a	n/a	n/a	n/a	n/a
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Bromodomain-containing protein 2 (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	2.80E+3	n/a	n/a	n/a	n/a	n/a
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Bromodomain-containing protein 2 (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	3.30E+3	n/a	n/a	n/a	n/a	n/a
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Bromodomain-containing protein 3 (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	3.20E+3	n/a	n/a	n/a	n/a	n/a
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Bromodomain-containing protein 3 (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	5.50E+3	n/a	n/a	n/a	n/a	n/a
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Bromodomain-containing protein 3 (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	4.00E+3	n/a	n/a	n/a	n/a	n/a
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Bromodomain-containing protein 4 (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	1.60E+3	n/a	n/a	n/a	n/a	n/a
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Bromodomain-containing protein 4 (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	1.70E+3	n/a	n/a	n/a	n/a	n/a
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Bromodomain-containing protein 4 (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	3.70E+3	n/a	n/a	n/a	n/a	n/a
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Bromodomain-containing protein 4 (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	580	n/a	n/a	n/a	n/a	n/a
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Bromodomain-containing protein 7 (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	340	n/a	n/a	n/a	n/a	n/a
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Bromodomain-containing protein 8 (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
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Bromodomain-containing protein 8 (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
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Bromodomain-containing protein 9 (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	25	n/a	n/a	n/a	n/a	n/a
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Bromodomain testis-specific protein (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	830	n/a	n/a	n/a	n/a	n/a
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Bromodomain testis-specific protein (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	1.20E+3	n/a	n/a	n/a	n/a	n/a
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Bromodomain testis-specific protein (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	2.60E+3	n/a	n/a	n/a	n/a	n/a
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Peregrin (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
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Bromodomain and PHD finger-containing protein 3 (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
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Chromatin remodeling regulator CECR2 (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
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CREB-binding protein (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	3.50E+3	n/a	n/a	n/a	n/a	n/a
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Histone acetyltransferase p300 (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	4.50E+3	n/a	n/a	n/a	n/a	n/a
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Nucleosome-remodeling factor subunit BPTF (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
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Histone acetyltransferase KAT2A (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	410	n/a	n/a	n/a	n/a	n/a
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Protein polybromo-1 (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	7.60E+3	n/a	n/a	n/a	n/a	n/a
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Protein polybromo-1 (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
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Histone acetyltransferase KAT2B (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
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Probable global transcription activator SNF2L2 (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
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Transcription activator BRG1 (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
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Transcription initiation factor TFIID subunit 1 (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
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Transcription initiation factor TFIID subunit 1-like (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
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Transcription intermediary factor 1-alpha (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
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E3 ubiquitin-protein ligase TRIM33 (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
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Bromodomain and WD repeat-containing protein 1 (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	UniChem	n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
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Bromodomain-containing protein 4 (Homo sapiens (Human))	BDBM50615275 (CHEMBL5282240) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	UniChem	n/a	n/a	5.10E+3	n/a	n/a	n/a	n/a	n/a	n/a
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