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SMILES: CC(C)n1c2cc(cnc2n(-c2cccc(OC(F)(F)C(F)F)c2)c1=O)C(=O)NC1(C)CS(=O)(=O)C1

InChI Key:

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 530662   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kcal/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Diacylglycerol O-acyltransferase 2


(Homo sapiens (Human))		BDBM530662
PNG
(WO2022076495, EXAMPLE 93)
Show SMILES CC(C)n1c2cc(cnc2n(-c2cccc(OC(F)(F)C(F)F)c2)c1=O)C(=O)NC1(C)CS(=O)(=O)C1
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KEGG

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antibodypedia
GoogleScholar
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PC cid
PC sid
UniChem
WIPO WO2022076495
n/an/a 24n/an/an/an/an/an/a


TBA

Assay Description
DGAT2 activity was determined by measuring the amount of enzymatic product 13Ci8-triolein (13C-l,2,3-Tri(cis-9-octadecenoyl)glycerol) using the membr...

Citation and Details

BindingDB Entry DOI: 10.7270/Q2ZP4981
More data for this
Ligand-Target Pair