Found 9 hits for monomerid = 50032973 Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
Gamma-aminobutyric acid type B receptor subunit 1
(Rattus norvegicus (Rat)) | BDBM50032973
(((Z)-3-Amino-propenyl)-methyl-phosphinic acid | 3-...)Show InChI InChI=1S/C4H10NO2P/c1-8(6,7)4-2-3-5/h3,5H,2,4H2,1H3,(H,6,7) | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| 650 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Sydney
Curated by PDSP Ki Database
| |
Eur J Pharmacol 329: 223-9 (1997)
BindingDB Entry DOI: 10.7270/Q2H41PZV |
More data for this Ligand-Target Pair | |
GABA A receptor alpha-3/beta-2/gamma-2
(Homo sapiens (Human)) | BDBM50032973
(((Z)-3-Amino-propenyl)-methyl-phosphinic acid | 3-...)Show InChI InChI=1S/C4H10NO2P/c1-8(6,7)4-2-3-5/h3,5H,2,4H2,1H3,(H,6,7) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| 5.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Sydney
Curated by PDSP Ki Database
| |
Eur J Pharmacol 329: 223-9 (1997)
BindingDB Entry DOI: 10.7270/Q2H41PZV |
More data for this Ligand-Target Pair | |
Gamma-aminobutyric acid receptor subunit alpha-1
(Rattus norvegicus (Rat)) | BDBM50032973
(((Z)-3-Amino-propenyl)-methyl-phosphinic acid | 3-...)Show InChI InChI=1S/C4H10NO2P/c1-8(6,7)4-2-3-5/h3,5H,2,4H2,1H3,(H,6,7) | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Sydney
Curated by PDSP Ki Database
| |
Eur J Pharmacol 329: 223-9 (1997)
BindingDB Entry DOI: 10.7270/Q2H41PZV |
More data for this Ligand-Target Pair | |
Gamma-aminobutyric acid type B receptor subunit 1
(Rattus norvegicus (Rat)) | BDBM50032973
(((Z)-3-Amino-propenyl)-methyl-phosphinic acid | 3-...)Show InChI InChI=1S/C4H10NO2P/c1-8(6,7)4-2-3-5/h3,5H,2,4H2,1H3,(H,6,7) | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Sydney
Curated by PDSP Ki Database
| |
Eur J Pharmacol 329: 223-9 (1997)
BindingDB Entry DOI: 10.7270/Q2H41PZV |
More data for this Ligand-Target Pair | |
GABA A receptor alpha-3/beta-2/gamma-2
(Homo sapiens (Human)) | BDBM50032973
(((Z)-3-Amino-propenyl)-methyl-phosphinic acid | 3-...)Show InChI InChI=1S/C4H10NO2P/c1-8(6,7)4-2-3-5/h3,5H,2,4H2,1H3,(H,6,7) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Sydney
Curated by PDSP Ki Database
| |
Eur J Pharmacol 329: 223-9 (1997)
BindingDB Entry DOI: 10.7270/Q2H41PZV |
More data for this Ligand-Target Pair | |
Gamma-aminobutyric acid receptor subunit alpha-1
(Rattus norvegicus (Rat)) | BDBM50032973
(((Z)-3-Amino-propenyl)-methyl-phosphinic acid | 3-...)Show InChI InChI=1S/C4H10NO2P/c1-8(6,7)4-2-3-5/h3,5H,2,4H2,1H3,(H,6,7) | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Sydney
Curated by PDSP Ki Database
| |
Eur J Pharmacol 329: 223-9 (1997)
BindingDB Entry DOI: 10.7270/Q2H41PZV |
More data for this Ligand-Target Pair | |
GABA-C receptor
(Homo sapiens (Human)) | BDBM50032973
(((Z)-3-Amino-propenyl)-methyl-phosphinic acid | 3-...)Show InChI InChI=1S/C4H10NO2P/c1-8(6,7)4-2-3-5/h3,5H,2,4H2,1H3,(H,6,7) | Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 5.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Sydney
Curated by ChEMBL
| Assay Description Antagonist activity at human GABAc Rho1 receptor expressed in Xenopus oocytes assessed as whole cell current production by two electrode voltage clam... |
J Med Chem 51: 3825-40 (2008)
Article DOI: 10.1021/jm7015842 BindingDB Entry DOI: 10.7270/Q27M07RR |
More data for this Ligand-Target Pair | |
GABA-B receptor 1/2
(Rattus norvegicus (Rat)) | BDBM50032973
(((Z)-3-Amino-propenyl)-methyl-phosphinic acid | 3-...)Show InChI InChI=1S/C4H10NO2P/c1-8(6,7)4-2-3-5/h3,5H,2,4H2,1H3,(H,6,7) | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| n/a | n/a | 665 | n/a | n/a | n/a | n/a | n/a | n/a |
CIBA-GEIGY AG
Curated by ChEMBL
| Assay Description Inhibition of [3H]-CGP-27,492 binding to Gamma-aminobutyric acid type B receptor of rat cortex |
J Med Chem 38: 3297-312 (1995)
BindingDB Entry DOI: 10.7270/Q2N58KDP |
More data for this Ligand-Target Pair | |
GABA-B receptor 1/2
(Rattus norvegicus (Rat)) | BDBM50032973
(((Z)-3-Amino-propenyl)-methyl-phosphinic acid | 3-...)Show InChI InChI=1S/C4H10NO2P/c1-8(6,7)4-2-3-5/h3,5H,2,4H2,1H3,(H,6,7) | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| n/a | n/a | 1.66E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
CIBA-GEIGY AG
Curated by ChEMBL
| Assay Description Inhibition of [3H]-CGP-27,492 binding to Gamma-aminobutyric acid type B receptor of rat cortex |
J Med Chem 38: 3297-312 (1995)
BindingDB Entry DOI: 10.7270/Q2N58KDP |
More data for this Ligand-Target Pair | |