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SMILES: COCCNCc1ccc(nc1)-n1[nH]cc(-c2cccnc2)c1=O

InChI Key: InChIKey=FSTZVIZVILWMNI-UHFFFAOYSA-N

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 109266   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kcal/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Transmembrane prolyl 4-hydroxylase


(Homo sapiens (Human))		BDBM109266
PNG
(US8609698, 5)
Show SMILES COCCNCc1ccc(nc1)-n1[nH]cc(-c2cccnc2)c1=O
Show InChI InChI=1S/C17H19N5O2/c1-24-8-7-19-9-13-4-5-16(20-10-13)22-17(23)15(12-21-22)14-3-2-6-18-11-14/h2-6,10-12,19,21H,7-9H2,1H3
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Similars
US Patent
n/an/a 6.30E+3n/an/an/an/an/an/a



Bayer Intellectual Property GmbH

US Patent


Assay Description
Inhibition of the Activity of HIF Prolyl Hydroxylase is carried out as described [Oehme F., Jonghaus W., Narouz-Ott L., Huetter J., Flamme I., Anal. ...

US Patent US8609698 (2013)


BindingDB Entry DOI: 10.7270/Q2G44NZ8
More data for this
Ligand-Target Pair