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SMILES: CC(C)CC(Nc1nc2ccccc2nc1C)c1ccc(cc1)C(=O)NCCC(O)=O

InChI Key: InChIKey=UUBRGIQNDRIPIE-UHFFFAOYSA-N

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 142027   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kcal/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Pro-glucagon


(Homo sapiens (Human))		BDBM142027
PNG
(US8927577, 8)
Show SMILES CC(C)CC(Nc1nc2ccccc2nc1C)c1ccc(cc1)C(=O)NCCC(O)=O
Show InChI InChI=1S/C24H28N4O3/c1-15(2)14-21(28-23-16(3)26-19-6-4-5-7-20(19)27-23)17-8-10-18(11-9-17)24(31)25-13-12-22(29)30/h4-11,15,21H,12-14H2,1-3H3,(H,25,31)(H,27,28)(H,29,30)
Reactome pathway
KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
 979n/an/an/an/an/an/a7.4n/a



Pfizer Inc.

US Patent


Assay Description
The Glucagon SPA assay is used to determine the ability of test compounds to block the binding of glucagon-cex to the glucagon receptor. Test compoun...

US Patent US8927577 (2015)


BindingDB Entry DOI: 10.7270/Q29S1PRV
More data for this
Ligand-Target Pair