BDBM350530 N-(4-bromophenyl)-2-(4-ethyl-2,5- dioxo-4-phenylimidazolidin-1- yl)acetamide::US10208071, Table 3.6::US10799518, Structure TABLE 3.6
SMILES: CCC1(NC(=O)N(CC(=O)Nc2ccc(Br)cc2)C1=O)c1ccccc1
InChI Key: InChIKey=KHDSTUZMHJIGKK-UHFFFAOYSA-N
Data: 2 EC50
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
N-formyl peptide receptor 2 (Homo sapiens (Human)) | BDBM350530 (N-(4-bromophenyl)-2-(4-ethyl-2,5- dioxo-4-phenylim...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 523 | n/a | n/a | n/a | n/a |
ALLERGAN, INC. US Patent | Assay Description HEK-Gα16 cells stably expressing the human FPR2 receptor was utilized. Cells were plated into 384-well poly-D-lysine coated plates at a density ... | US Patent US10799518 (2020) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
N-formyl peptide receptor 2 (Homo sapiens (Human)) | BDBM350530 (N-(4-bromophenyl)-2-(4-ethyl-2,5- dioxo-4-phenylim...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 5.23E+5 | n/a | n/a | n/a | n/a |
ALLERGAN, INC. US Patent | Assay Description HEK-Gα16 cells stably expressing the human FPR2 receptor was utilized. Cells were plated into 384-well poly-D-lysine coated plates at a density ... | US Patent US10208071 (2019) BindingDB Entry DOI: 10.7270/Q2TH8PT9 | |||||||||||
More data for this Ligand-Target Pair |