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null

SMILES: COCc1ccccc1-c1ccc(o1)C(=O)NC[C@@H](N)C(O)=O

InChI Key:

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50583024
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Glutamate receptor ionotropic, NMDA 1/2A (Rattus norvegicus (Rat)-RAT)	BDBM50583024 (CHEMBL5087170) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	3.10E+3	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at rat GluN1/GluN2A NMDA receptor expressed in Xenopus oocytes measured after 4 days in presence of L-glutamte by two-electrode volt...				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c01810 BindingDB Entry DOI: 10.7270/Q21R6VFZ
TBA					More data for this Ligand-Target Pair
Glutamate receptor ionotropic, NMDA 1/2D (RAT-Rattus norvegicus (Rat))	BDBM50583024 (CHEMBL5087170) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	3.20E+3	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at rat GluN1/GluN2D NMDA receptor expressed in Xenopus oocytes measured after 4 days in presence of L-glutamte by two-electrode volt...				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c01810 BindingDB Entry DOI: 10.7270/Q21R6VFZ
TBA					More data for this Ligand-Target Pair
Glutamate receptor ionotropic, NMDA 1/2C (RAT-Rattus norvegicus (Rat))	BDBM50583024 (CHEMBL5087170) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	1.60E+3	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at rat GluN1/GluN2C NMDA receptor expressed in Xenopus oocytes measured after 4 days in presence of L-glutamte by two-electrode volt...				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c01810 BindingDB Entry DOI: 10.7270/Q21R6VFZ
TBA					More data for this Ligand-Target Pair