null
SMILES: CCCC(C)N1CCC(CC1)N(Cc1ccccc1)C(=O)Nc1cccc(OC(F)(F)F)c1
InChI Key:
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM518708 (US11116757, No. A12) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 82.7 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair |