Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Voltage-dependent L-type calcium channel subunit alpha-1C (RAT) | BDBM50462274 (CHEMBL4246869) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Siena Curated by ChEMBL | Assay Description Inhibition of CaV1.2 channel in rat tail artery myocytes assessed as reduction in Ba2+ current at -50 mV holding potential by whole-cell patch-clamp ... | Eur J Med Chem 150: 698-718 (2018) Article DOI: 10.1016/j.ejmech.2018.03.024 BindingDB Entry DOI: 10.7270/Q2PC3518 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phosphoethanolamine N-methyltransferase (Plasmodium falciparum) | BDBM50462274 (CHEMBL4246869) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.43E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Siena Curated by ChEMBL | Assay Description Inhibition of plasmodium falciparum phosphoethanolamine N-methyltransferase expressed in Escherichia coli using phosphoethanolamine as substrate and ... | Eur J Med Chem 150: 698-718 (2018) Article DOI: 10.1016/j.ejmech.2018.03.024 BindingDB Entry DOI: 10.7270/Q2PC3518 | |||||||||||
More data for this Ligand-Target Pair |