Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Elastase (Pseudomonas aeruginosa) | BDBM50498101![]() (CHEMBL3403862) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.81E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Technical University of Denmark Curated by ChEMBL | Assay Description Antagonist activity at lasB in Pseudomonas aeruginosa harboring lasB-gfp gene assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing by green ... | Bioorg Med Chem 23: 1638-50 (2015) Article DOI: 10.1016/j.bmc.2015.01.038 BindingDB Entry DOI: 10.7270/Q2F192P6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Elastase (Pseudomonas aeruginosa) | BDBM50498105![]() (CHEMBL3403858) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.25E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Technical University of Denmark Curated by ChEMBL | Assay Description Antagonist activity at lasB in Pseudomonas aeruginosa harboring lasB-gfp gene assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing by green ... | Bioorg Med Chem 23: 1638-50 (2015) Article DOI: 10.1016/j.bmc.2015.01.038 BindingDB Entry DOI: 10.7270/Q2F192P6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Elastase (Pseudomonas aeruginosa) | BDBM50498098![]() (CHEMBL3403859) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.99E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Technical University of Denmark Curated by ChEMBL | Assay Description Antagonist activity at lasB in Pseudomonas aeruginosa harboring lasB-gfp gene assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing by green ... | Bioorg Med Chem 23: 1638-50 (2015) Article DOI: 10.1016/j.bmc.2015.01.038 BindingDB Entry DOI: 10.7270/Q2F192P6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Elastase (Pseudomonas aeruginosa) | BDBM50498104![]() (CHEMBL3403865) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.82E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Technical University of Denmark Curated by ChEMBL | Assay Description Antagonist activity at lasB in Pseudomonas aeruginosa harboring lasB-gfp gene assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing by green ... | Bioorg Med Chem 23: 1638-50 (2015) Article DOI: 10.1016/j.bmc.2015.01.038 BindingDB Entry DOI: 10.7270/Q2F192P6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Elastase (Pseudomonas aeruginosa) | BDBM50498097![]() (CHEMBL3403860) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.10E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Technical University of Denmark Curated by ChEMBL | Assay Description Antagonist activity at lasB in Pseudomonas aeruginosa harboring lasB-gfp gene assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing by green ... | Bioorg Med Chem 23: 1638-50 (2015) Article DOI: 10.1016/j.bmc.2015.01.038 BindingDB Entry DOI: 10.7270/Q2F192P6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Elastase (Pseudomonas aeruginosa) | BDBM50498102![]() (CHEMBL3403856) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.78E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Technical University of Denmark Curated by ChEMBL | Assay Description Antagonist activity at lasB in Pseudomonas aeruginosa harboring lasB-gfp gene assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing by green ... | Bioorg Med Chem 23: 1638-50 (2015) Article DOI: 10.1016/j.bmc.2015.01.038 BindingDB Entry DOI: 10.7270/Q2F192P6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Elastase (Pseudomonas aeruginosa) | BDBM50498100![]() (CHEMBL3403864) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.92E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Technical University of Denmark Curated by ChEMBL | Assay Description Antagonist activity at lasB in Pseudomonas aeruginosa harboring lasB-gfp gene assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing by green ... | Bioorg Med Chem 23: 1638-50 (2015) Article DOI: 10.1016/j.bmc.2015.01.038 BindingDB Entry DOI: 10.7270/Q2F192P6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Elastase (Pseudomonas aeruginosa) | BDBM50498103![]() (CHEMBL3403861) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 8.89E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Technical University of Denmark Curated by ChEMBL | Assay Description Antagonist activity at lasB in Pseudomonas aeruginosa harboring lasB-gfp gene assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing by green ... | Bioorg Med Chem 23: 1638-50 (2015) Article DOI: 10.1016/j.bmc.2015.01.038 BindingDB Entry DOI: 10.7270/Q2F192P6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Elastase (Pseudomonas aeruginosa) | BDBM50498099![]() (CHEMBL3403868) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.10E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Technical University of Denmark Curated by ChEMBL | Assay Description Antagonist activity at lasB in Pseudomonas aeruginosa harboring lasB-gfp gene assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing by green ... | Bioorg Med Chem 23: 1638-50 (2015) Article DOI: 10.1016/j.bmc.2015.01.038 BindingDB Entry DOI: 10.7270/Q2F192P6 | |||||||||||
More data for this Ligand-Target Pair |