Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Reverse transcriptase protein (Human immunodeficiency virus 1) | BDBM50479470![]() (CHEMBL489586 | MK-4965) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet ![]() | MCE PC cid PC sid PDB UniChem | Article PubMed | 0.390 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Labs. Curated by ChEMBL | Assay Description Inhibition of Human immunodeficiency virus reverse transcriptase K103N mutant by SPA assay | Bioorg Med Chem Lett 21: 7344-50 (2011) Article DOI: 10.1016/j.bmcl.2011.10.027 BindingDB Entry DOI: 10.7270/Q25Q4ZZ2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Reverse transcriptase protein (Human immunodeficiency virus 1) | BDBM50484496![]() (CHEMBL1928648) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 0.480 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Labs. Curated by ChEMBL | Assay Description Inhibition of Human immunodeficiency virus reverse transcriptase K103N mutant by SPA assay | Bioorg Med Chem Lett 21: 7344-50 (2011) Article DOI: 10.1016/j.bmcl.2011.10.027 BindingDB Entry DOI: 10.7270/Q25Q4ZZ2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Reverse transcriptase protein (Human immunodeficiency virus 1) | BDBM50484495![]() (CHEMBL1928645) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 1.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Labs. Curated by ChEMBL | Assay Description Inhibition of Human immunodeficiency virus reverse transcriptase K103N mutant by SPA assay | Bioorg Med Chem Lett 21: 7344-50 (2011) Article DOI: 10.1016/j.bmcl.2011.10.027 BindingDB Entry DOI: 10.7270/Q25Q4ZZ2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Reverse transcriptase protein (Human immunodeficiency virus 1) | BDBM50484493![]() (CHEMBL1928646) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 1.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Labs. Curated by ChEMBL | Assay Description Inhibition of Human immunodeficiency virus reverse transcriptase K103N mutant by SPA assay | Bioorg Med Chem Lett 21: 7344-50 (2011) Article DOI: 10.1016/j.bmcl.2011.10.027 BindingDB Entry DOI: 10.7270/Q25Q4ZZ2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Reverse transcriptase protein (Human immunodeficiency virus 1) | BDBM50484494![]() (CHEMBL1928647) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 2.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Labs. Curated by ChEMBL | Assay Description Inhibition of Human immunodeficiency virus reverse transcriptase K103N mutant by SPA assay | Bioorg Med Chem Lett 21: 7344-50 (2011) Article DOI: 10.1016/j.bmcl.2011.10.027 BindingDB Entry DOI: 10.7270/Q25Q4ZZ2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Reverse transcriptase protein (Human immunodeficiency virus 1) | BDBM50484492![]() (CHEMBL1928643) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 3.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Labs. Curated by ChEMBL | Assay Description Inhibition of Human immunodeficiency virus reverse transcriptase K103N mutant by SPA assay | Bioorg Med Chem Lett 21: 7344-50 (2011) Article DOI: 10.1016/j.bmcl.2011.10.027 BindingDB Entry DOI: 10.7270/Q25Q4ZZ2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Reverse transcriptase protein (Human immunodeficiency virus 1) | BDBM50484497![]() (CHEMBL1928644) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 58 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Labs. Curated by ChEMBL | Assay Description Inhibition of Human immunodeficiency virus reverse transcriptase K103N mutant by SPA assay | Bioorg Med Chem Lett 21: 7344-50 (2011) Article DOI: 10.1016/j.bmcl.2011.10.027 BindingDB Entry DOI: 10.7270/Q25Q4ZZ2 | |||||||||||
More data for this Ligand-Target Pair |