Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50019646 (2-(alpha-(2,6-Dichlorophenoxy)ethyl)2-imidazoline ...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid UniChem Patents Similars | Article PubMed | 4.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Agonist activity at human adrenoceptor aplha 2A expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri... | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50419889 (CHEMBL155866) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 12 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Agonist activity at human adrenoceptor aplha 2A expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri... | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50419885 (CHEMBL157206) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 17 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Agonist activity at human adrenoceptor aplha 2A expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri... | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50419874 (CHEMBL1956192) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 23 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Agonist activity at human adrenoceptor aplha 2A expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri... | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50419886 (CHEMBL156336) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 24 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Agonist activity at human adrenoceptor aplha 2A expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri... | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50419890 (CHEMBL1956191) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 29 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Agonist activity at human adrenoceptor aplha 2A expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri... | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50419884 (CHEMBL157955) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 32 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RS-79948-197 from human adrenoceptor aplha 2A expressed in CHO cells | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50419878 (CHEMBL1956195) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 36 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Agonist activity at human adrenoceptor aplha 2A expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri... | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50419881 (CHEMBL1956199) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 58 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Agonist activity at human adrenoceptor aplha 2A expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri... | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2B adrenergic receptor (Homo sapiens (Human)) | BDBM50019646 (2-(alpha-(2,6-Dichlorophenoxy)ethyl)2-imidazoline ...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid UniChem Patents Similars | Article PubMed | 68 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RS-79948-197 from human adrenoceptor aplha 2B expressed in CHO cells | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2C adrenergic receptor (Homo sapiens (Human)) | BDBM50019646 (2-(alpha-(2,6-Dichlorophenoxy)ethyl)2-imidazoline ...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid UniChem Patents Similars | Article PubMed | 69 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RS-79948-197 from human adrenoceptor aplha 2C expressed in CHO cells | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50419877 (CHEMBL1956194) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 72 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Agonist activity at human adrenoceptor aplha 2A expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri... | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50419876 (CHEMBL266613) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 72 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Agonist activity at human adrenoceptor aplha 2A expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri... | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50419887 (CHEMBL14208) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 83 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Agonist activity at human adrenoceptor aplha 2A expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri... | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50419880 (CHEMBL1956197) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 83 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Agonist activity at human adrenoceptor aplha 2A expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri... | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50419879 (CHEMBL1956196) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 98 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Agonist activity at human adrenoceptor aplha 2A expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri... | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2C adrenergic receptor (Homo sapiens (Human)) | BDBM50419885 (CHEMBL157206) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 129 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RS-79948-197 from human adrenoceptor aplha 2C expressed in CHO cells | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2B adrenergic receptor (Homo sapiens (Human)) | BDBM50419889 (CHEMBL155866) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 182 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RS-79948-197 from human adrenoceptor aplha 2B expressed in CHO cells | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50419875 (CHEMBL1956193) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 182 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Agonist activity at human adrenoceptor aplha 2A expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri... | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2C adrenergic receptor (Homo sapiens (Human)) | BDBM50419889 (CHEMBL155866) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 251 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RS-79948-197 from human adrenoceptor aplha 2C expressed in CHO cells | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2B adrenergic receptor (Homo sapiens (Human)) | BDBM50419884 (CHEMBL157955) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 269 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RS-79948-197 from human adrenoceptor aplha 2B expressed in CHO cells | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2B adrenergic receptor (Homo sapiens (Human)) | BDBM50419885 (CHEMBL157206) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 275 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RS-79948-197 from human adrenoceptor aplha 2B expressed in CHO cells | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2C adrenergic receptor (Homo sapiens (Human)) | BDBM50419884 (CHEMBL157955) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 275 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RS-79948-197 from human adrenoceptor aplha 2C expressed in CHO cells | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2C adrenergic receptor (Homo sapiens (Human)) | BDBM50419878 (CHEMBL1956195) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 275 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RS-79948-197 from human adrenoceptor aplha 2C expressed in CHO cells | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2C adrenergic receptor (Homo sapiens (Human)) | BDBM50419874 (CHEMBL1956192) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 282 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RS-79948-197 from human adrenoceptor aplha 2C expressed in CHO cells | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2B adrenergic receptor (Homo sapiens (Human)) | BDBM50419886 (CHEMBL156336) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 282 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RS-79948-197 from human adrenoceptor aplha 2B expressed in CHO cells | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2C adrenergic receptor (Homo sapiens (Human)) | BDBM50419886 (CHEMBL156336) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 288 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RS-79948-197 from human adrenoceptor aplha 2C expressed in CHO cells | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2B adrenergic receptor (Homo sapiens (Human)) | BDBM50419890 (CHEMBL1956191) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 331 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RS-79948-197 from human adrenoceptor aplha 2B expressed in CHO cells | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2B adrenergic receptor (Homo sapiens (Human)) | BDBM50419874 (CHEMBL1956192) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 355 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RS-79948-197 from human adrenoceptor aplha 2B expressed in CHO cells | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2C adrenergic receptor (Homo sapiens (Human)) | BDBM50419887 (CHEMBL14208) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 398 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RS-79948-197 from human adrenoceptor aplha 2C expressed in CHO cells | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2B adrenergic receptor (Homo sapiens (Human)) | BDBM50419878 (CHEMBL1956195) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 407 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RS-79948-197 from human adrenoceptor aplha 2B expressed in CHO cells | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2C adrenergic receptor (Homo sapiens (Human)) | BDBM50419876 (CHEMBL266613) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 457 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RS-79948-197 from human adrenoceptor aplha 2C expressed in CHO cells | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50419873 (CHEMBL1956203) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 490 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Agonist activity at human adrenoceptor aplha 2A expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri... | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2C adrenergic receptor (Homo sapiens (Human)) | BDBM50419890 (CHEMBL1956191) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 490 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RS-79948-197 from human adrenoceptor aplha 2C expressed in CHO cells | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2C adrenergic receptor (Homo sapiens (Human)) | BDBM50419877 (CHEMBL1956194) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 603 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RS-79948-197 from human adrenoceptor aplha 2C expressed in CHO cells | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2C adrenergic receptor (Homo sapiens (Human)) | BDBM50419873 (CHEMBL1956203) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 631 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RS-79948-197 from human adrenoceptor aplha 2C expressed in CHO cells | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2C adrenergic receptor (Homo sapiens (Human)) | BDBM50419880 (CHEMBL1956197) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 676 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RS-79948-197 from human adrenoceptor aplha 2C expressed in CHO cells | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2C adrenergic receptor (Homo sapiens (Human)) | BDBM50419879 (CHEMBL1956196) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 759 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RS-79948-197 from human adrenoceptor aplha 2C expressed in CHO cells | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2C adrenergic receptor (Homo sapiens (Human)) | BDBM50419881 (CHEMBL1956199) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 832 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RS-79948-197 from human adrenoceptor aplha 2C expressed in CHO cells | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2B adrenergic receptor (Homo sapiens (Human)) | BDBM50419881 (CHEMBL1956199) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 871 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RS-79948-197 from human adrenoceptor aplha 2B expressed in CHO cells | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2B adrenergic receptor (Homo sapiens (Human)) | BDBM50419877 (CHEMBL1956194) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 871 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RS-79948-197 from human adrenoceptor aplha 2B expressed in CHO cells | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2B adrenergic receptor (Homo sapiens (Human)) | BDBM50419876 (CHEMBL266613) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 933 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RS-79948-197 from human adrenoceptor aplha 2B expressed in CHO cells | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2C adrenergic receptor (Homo sapiens (Human)) | BDBM50419875 (CHEMBL1956193) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 977 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RS-79948-197 from human adrenoceptor aplha 2C expressed in CHO cells | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50419888 (CHEMBL1956202) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.02E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RS-79948-197 from human adrenoceptor aplha 2A expressed in CHO cells | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2B adrenergic receptor (Homo sapiens (Human)) | BDBM50419880 (CHEMBL1956197) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.05E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RS-79948-197 from human adrenoceptor aplha 2B expressed in CHO cells | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50419883 (CHEMBL1956201) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.05E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RS-79948-197 from human adrenoceptor aplha 2A expressed in CHO cells | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2B adrenergic receptor (Homo sapiens (Human)) | BDBM50419879 (CHEMBL1956196) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.32E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RS-79948-197 from human adrenoceptor aplha 2B expressed in CHO cells | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2B adrenergic receptor (Homo sapiens (Human)) | BDBM50419887 (CHEMBL14208) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.59E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RS-79948-197 from human adrenoceptor aplha 2B expressed in CHO cells | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2B adrenergic receptor (Homo sapiens (Human)) | BDBM50419875 (CHEMBL1956193) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.62E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RS-79948-197 from human adrenoceptor aplha 2B expressed in CHO cells | Bioorg Med Chem 20: 2082-90 (2012) Article DOI: 10.1016/j.bmc.2012.01.035 BindingDB Entry DOI: 10.7270/Q2TD9ZKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor (RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50482773 (CHEMBL1253513) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 1.92E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RX821002 from alpha2 adrenergic receptor in rat brain membrane | Bioorg Med Chem 18: 7085-91 (2010) Article DOI: 10.1016/j.bmc.2010.08.005 BindingDB Entry DOI: 10.7270/Q2KP850W | |||||||||||
More data for this Ligand-Target Pair |
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