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Compile Data Set for Download or QSAR

Found 38 hits with Last Name = 'nicolaes' and Initial = 'gaf'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
N-formyl peptide receptor 2


(Homo sapiens (Human))
BDBM50582808
PNG
(CHEMBL5085435)
Show SMILES Brc1ccc(NC(=O)NC2CCN(CC3CCN(Cc4ccccc4)CC3)C2=O)cc1
PDB

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n/an/an/an/a 250n/an/an/an/a


TBA

Assay Description
Agonist activity at FPRL1 (unknown origin) expressed in CHO-K1 cells assessed as increase in calcium mobilization incubated for 2.5 hrs by cellular b...


Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113805
BindingDB Entry DOI: 10.7270/Q2QF8XRP
More data for this
Ligand-Target Pair
N-formyl peptide receptor 2


(Homo sapiens (Human))
BDBM50582817
PNG
(CHEMBL5076914)
Show SMILES Brc1ccc(NC(=O)NC2CCN(C2=O)c2ccccc2)cc1
PDB

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n/an/an/an/a 7.36E+3n/an/an/an/a


TBA

Assay Description
Agonist activity at human FPR2 expressed in HEK293-A cells assessed as ERK phosphorylation level incubated for 5 mins by ELISA assay


Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113805
BindingDB Entry DOI: 10.7270/Q2QF8XRP
More data for this
Ligand-Target Pair
N-formyl peptide receptor 2


(Homo sapiens (Human))
BDBM50582810
PNG
(CHEMBL5085818)
Show SMILES Brc1ccc(NC(=O)NC2CCN(C3CCN(Cc4ccccc4)C3)C2=O)cc1
PDB

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n/an/an/an/a 2.70E+3n/an/an/an/a


TBA

Assay Description
Agonist activity at FPRL1 (unknown origin) expressed in CHO-K1 cells assessed as increase in calcium mobilization incubated for 2.5 hrs by cellular b...


Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113805
BindingDB Entry DOI: 10.7270/Q2QF8XRP
More data for this
Ligand-Target Pair
N-formyl peptide receptor 2


(Homo sapiens (Human))
BDBM50582810
PNG
(CHEMBL5085818)
Show SMILES Brc1ccc(NC(=O)NC2CCN(C3CCN(Cc4ccccc4)C3)C2=O)cc1
PDB

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n/an/an/an/a 2.70E+3n/an/an/an/a


TBA

Assay Description
Agonist activity at FPRL1 (unknown origin) expressed in CHO-K1 cells assessed as increase in calcium mobilization incubated for 2.5 hrs by cellular b...


Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113805
BindingDB Entry DOI: 10.7270/Q2QF8XRP
More data for this
Ligand-Target Pair
N-formyl peptide receptor 2


(Homo sapiens (Human))
BDBM50582811
PNG
(CHEMBL5087410)
Show SMILES CC(C)(C)OC(=O)N1CCC[C@@H](C1)N1CCC(NC(=O)Nc2ccc(Br)cc2)C1=O |r|
PDB

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n/an/an/an/a 130n/an/an/an/a


TBA

Assay Description
Agonist activity at FPRL1 (unknown origin) expressed in CHO-K1 cells assessed as increase in calcium mobilization incubated for 2.5 hrs by cellular b...


Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113805
BindingDB Entry DOI: 10.7270/Q2QF8XRP
More data for this
Ligand-Target Pair
N-formyl peptide receptor 2


(Homo sapiens (Human))
BDBM50582811
PNG
(CHEMBL5087410)
Show SMILES CC(C)(C)OC(=O)N1CCC[C@@H](C1)N1CCC(NC(=O)Nc2ccc(Br)cc2)C1=O |r|
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n/an/an/an/a 130n/an/an/an/a


TBA

Assay Description
Agonist activity at FPRL1 (unknown origin) expressed in CHO-K1 cells assessed as increase in calcium mobilization incubated for 2.5 hrs by cellular b...


Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113805
BindingDB Entry DOI: 10.7270/Q2QF8XRP
More data for this
Ligand-Target Pair
N-formyl peptide receptor 2


(Homo sapiens (Human))
BDBM50582812
PNG
(CHEMBL5076199)
Show SMILES Cc1nn(c(C)c1N1CCC(NC(=O)Nc2ccc(Br)cc2)C1=O)-c1ccccc1
PDB

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n/an/an/an/a 280n/an/an/an/a


TBA

Assay Description
Agonist activity at FPRL1 (unknown origin) expressed in CHO-K1 cells assessed as increase in calcium mobilization incubated for 2.5 hrs by cellular b...


Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113805
BindingDB Entry DOI: 10.7270/Q2QF8XRP
More data for this
Ligand-Target Pair
N-formyl peptide receptor 2


(Homo sapiens (Human))
BDBM50582813
PNG
(CHEMBL5093348)
Show SMILES Brc1ccc(NC(=O)NC2CCN(C3CCN(CC3)c3ncccn3)C2=O)cc1
PDB

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n/an/an/an/a 8n/an/an/an/a


TBA

Assay Description
Agonist activity at FPRL1 (unknown origin) expressed in CHO-K1 cells assessed as increase in calcium mobilization incubated for 2.5 hrs by cellular b...


Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113805
BindingDB Entry DOI: 10.7270/Q2QF8XRP
More data for this
Ligand-Target Pair
N-formyl peptide receptor 2


(Homo sapiens (Human))
BDBM50582814
PNG
(CHEMBL5088283)
Show SMILES Fc1ccccc1N1CCC(NC(=O)Nc2ccc(cc2)C#N)C1=O
PDB

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n/an/an/an/a 1.50E+4n/an/an/an/a


TBA

Assay Description
Agonist activity at FPRL1 (unknown origin) expressed in CHO-K1 cells assessed as increase in calcium mobilization incubated for 2.5 hrs by cellular b...


Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113805
BindingDB Entry DOI: 10.7270/Q2QF8XRP
More data for this
Ligand-Target Pair
N-formyl peptide receptor 2


(Homo sapiens (Human))
BDBM50582815
PNG
(CHEMBL5078594)
Show SMILES Cc1nn(C)cc1N1CCC(NC(=O)Nc2ccc(Br)cc2)C1=O
PDB

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n/an/an/an/a 142n/an/an/an/a


TBA

Assay Description
Agonist activity at FPRL1 (unknown origin) expressed in CHO-K1 cells assessed as increase in calcium mobilization incubated for 2.5 hrs by cellular b...


Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113805
BindingDB Entry DOI: 10.7270/Q2QF8XRP
More data for this
Ligand-Target Pair
N-formyl peptide receptor 2


(Homo sapiens (Human))
BDBM50582816
PNG
(CHEMBL5084099)
Show SMILES CC(C)n1cc(cn1)N1CCC(NC(=O)Nc2ccc(Br)cc2)C1=O
PDB

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n/an/an/an/a 884n/an/an/an/a


TBA

Assay Description
Agonist activity at FPRL1 (unknown origin) expressed in CHO-K1 cells assessed as increase in calcium mobilization incubated for 2.5 hrs by cellular b...


Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113805
BindingDB Entry DOI: 10.7270/Q2QF8XRP
More data for this
Ligand-Target Pair
N-formyl peptide receptor 2


(Homo sapiens (Human))
BDBM50582817
PNG
(CHEMBL5076914)
Show SMILES Brc1ccc(NC(=O)NC2CCN(C2=O)c2ccccc2)cc1
PDB

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n/an/an/an/a 430n/an/an/an/a


TBA

Assay Description
Agonist activity at FPRL1 (unknown origin) expressed in CHO-K1 cells assessed as increase in calcium mobilization incubated for 2.5 hrs by cellular b...


Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113805
BindingDB Entry DOI: 10.7270/Q2QF8XRP
More data for this
Ligand-Target Pair
N-formyl peptide receptor 2


(Homo sapiens (Human))
BDBM50582818
PNG
(CHEMBL5085666)
Show SMILES Fc1ccc(cc1)N1CCC(NC(=O)Nc2ccc(Br)cc2)C1=O
PDB

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n/an/an/an/a 1.97E+3n/an/an/an/a


TBA

Assay Description
Agonist activity at FPRL1 (unknown origin) expressed in CHO-K1 cells assessed as increase in calcium mobilization incubated for 2.5 hrs by cellular b...


Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113805
BindingDB Entry DOI: 10.7270/Q2QF8XRP
More data for this
Ligand-Target Pair
N-formyl peptide receptor 2


(Homo sapiens (Human))
BDBM50582819
PNG
(CHEMBL5087710)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N1CCC(NC(=O)Nc2ccc(Br)cc2)C1=O
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n/an/an/an/a 730n/an/an/an/a


TBA

Assay Description
Agonist activity at FPRL1 (unknown origin) expressed in CHO-K1 cells assessed as increase in calcium mobilization incubated for 2.5 hrs by cellular b...


Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113805
BindingDB Entry DOI: 10.7270/Q2QF8XRP
More data for this
Ligand-Target Pair
N-formyl peptide receptor 2


(Homo sapiens (Human))
BDBM50582820
PNG
(CHEMBL5090603)
Show SMILES CC(C)(C)OC(=O)N1CCC(CN2CCC(NC(=O)Nc3ccc(Br)cc3)C2=O)CC1
PDB

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n/an/an/an/a 400n/an/an/an/a


TBA

Assay Description
Agonist activity at FPRL1 (unknown origin) expressed in CHO-K1 cells assessed as increase in calcium mobilization incubated for 2.5 hrs by cellular b...


Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113805
BindingDB Entry DOI: 10.7270/Q2QF8XRP
More data for this
Ligand-Target Pair
N-formyl peptide receptor 2


(Homo sapiens (Human))
BDBM50582821
PNG
(CHEMBL5084374)
Show SMILES Brc1ccc(NC(=O)NC2CCN(CC3CCNCC3)C2=O)cc1
PDB

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n/an/an/an/a 270n/an/an/an/a


TBA

Assay Description
Agonist activity at FPRL1 (unknown origin) expressed in CHO-K1 cells assessed as increase in calcium mobilization incubated for 2.5 hrs by cellular b...


Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113805
BindingDB Entry DOI: 10.7270/Q2QF8XRP
More data for this
Ligand-Target Pair
N-formyl peptide receptor 2


(Homo sapiens (Human))
BDBM50582822
PNG
(CHEMBL5075000)
Show SMILES Brc1ccc(NC(=O)NC2CCN(C3CCNCC3)C2=O)cc1
PDB

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n/an/an/an/a 230n/an/an/an/a


TBA

Assay Description
Agonist activity at FPRL1 (unknown origin) expressed in CHO-K1 cells assessed as increase in calcium mobilization incubated for 2.5 hrs by cellular b...


Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113805
BindingDB Entry DOI: 10.7270/Q2QF8XRP
More data for this
Ligand-Target Pair
N-formyl peptide receptor 2


(Homo sapiens (Human))
BDBM50582823
PNG
(CHEMBL5080179)
Show SMILES CC(C)(C)OC(=O)N1CC(C1)N1CCC(NC(=O)Nc2ccc(Br)cc2)C1=O
PDB

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n/an/an/an/a 410n/an/an/an/a


TBA

Assay Description
Agonist activity at FPRL1 (unknown origin) expressed in CHO-K1 cells assessed as increase in calcium mobilization incubated for 2.5 hrs by cellular b...


Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113805
BindingDB Entry DOI: 10.7270/Q2QF8XRP
More data for this
Ligand-Target Pair
N-formyl peptide receptor 2


(Homo sapiens (Human))
BDBM50582823
PNG
(CHEMBL5080179)
Show SMILES CC(C)(C)OC(=O)N1CC(C1)N1CCC(NC(=O)Nc2ccc(Br)cc2)C1=O
PDB

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n/an/an/an/a 2.35E+3n/an/an/an/a


TBA

Assay Description
Agonist activity at FPRL1 (unknown origin) expressed in CHO-K1 cells assessed as stimulation of beta-arrestin recruitment incubated for 150 mins by b...


Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113805
BindingDB Entry DOI: 10.7270/Q2QF8XRP
More data for this
Ligand-Target Pair
N-formyl peptide receptor 2


(Homo sapiens (Human))
BDBM50582808
PNG
(CHEMBL5085435)
Show SMILES Brc1ccc(NC(=O)NC2CCN(CC3CCN(Cc4ccccc4)CC3)C2=O)cc1
PDB

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n/an/an/an/a 2.25E+3n/an/an/an/a


TBA

Assay Description
Agonist activity at FPRL1 (unknown origin) expressed in CHO-K1 cells assessed as stimulation of beta-arrestin recruitment incubated for 150 mins by b...


Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113805
BindingDB Entry DOI: 10.7270/Q2QF8XRP
More data for this
Ligand-Target Pair
N-formyl peptide receptor 2


(Homo sapiens (Human))
BDBM50582809
PNG
(CHEMBL5070452)
Show SMILES Brc1ccc(NC(=O)NC2CCN(C3CCN(Cc4ccccc4)CC3)C2=O)cc1
PDB

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n/an/an/an/a 2.87E+3n/an/an/an/a


TBA

Assay Description
Agonist activity at FPRL1 (unknown origin) expressed in CHO-K1 cells assessed as stimulation of beta-arrestin recruitment incubated for 150 mins by b...


Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113805
BindingDB Entry DOI: 10.7270/Q2QF8XRP
More data for this
Ligand-Target Pair
N-formyl peptide receptor 2


(Homo sapiens (Human))
BDBM50582810
PNG
(CHEMBL5085818)
Show SMILES Brc1ccc(NC(=O)NC2CCN(C3CCN(Cc4ccccc4)C3)C2=O)cc1
PDB

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n/an/an/an/a 1.37E+3n/an/an/an/a


TBA

Assay Description
Agonist activity at FPRL1 (unknown origin) expressed in CHO-K1 cells assessed as stimulation of beta-arrestin recruitment incubated for 150 mins by b...


Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113805
BindingDB Entry DOI: 10.7270/Q2QF8XRP
More data for this
Ligand-Target Pair
N-formyl peptide receptor 2


(Homo sapiens (Human))
BDBM50582810
PNG
(CHEMBL5085818)
Show SMILES Brc1ccc(NC(=O)NC2CCN(C3CCN(Cc4ccccc4)C3)C2=O)cc1
PDB

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n/an/an/an/a 1.37E+3n/an/an/an/a


TBA

Assay Description
Agonist activity at FPRL1 (unknown origin) expressed in CHO-K1 cells assessed as stimulation of beta-arrestin recruitment incubated for 150 mins by b...


Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113805
BindingDB Entry DOI: 10.7270/Q2QF8XRP
More data for this
Ligand-Target Pair
N-formyl peptide receptor 2


(Homo sapiens (Human))
BDBM50582811
PNG
(CHEMBL5087410)
Show SMILES CC(C)(C)OC(=O)N1CCC[C@@H](C1)N1CCC(NC(=O)Nc2ccc(Br)cc2)C1=O |r|
PDB

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n/an/an/an/a 1.38E+3n/an/an/an/a


TBA

Assay Description
Agonist activity at FPRL1 (unknown origin) expressed in CHO-K1 cells assessed as stimulation of beta-arrestin recruitment incubated for 150 mins by b...


Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113805
BindingDB Entry DOI: 10.7270/Q2QF8XRP
More data for this
Ligand-Target Pair
N-formyl peptide receptor 2


(Homo sapiens (Human))
BDBM50582811
PNG
(CHEMBL5087410)
Show SMILES CC(C)(C)OC(=O)N1CCC[C@@H](C1)N1CCC(NC(=O)Nc2ccc(Br)cc2)C1=O |r|
PDB

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n/an/an/an/a 1.38E+3n/an/an/an/a


TBA

Assay Description
Agonist activity at FPRL1 (unknown origin) expressed in CHO-K1 cells assessed as stimulation of beta-arrestin recruitment incubated for 150 mins by b...


Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113805
BindingDB Entry DOI: 10.7270/Q2QF8XRP
More data for this
Ligand-Target Pair
N-formyl peptide receptor 2


(Homo sapiens (Human))
BDBM50582812
PNG
(CHEMBL5076199)
Show SMILES Cc1nn(c(C)c1N1CCC(NC(=O)Nc2ccc(Br)cc2)C1=O)-c1ccccc1
PDB

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n/an/an/an/a 400n/an/an/an/a


TBA

Assay Description
Agonist activity at FPRL1 (unknown origin) expressed in CHO-K1 cells assessed as stimulation of beta-arrestin recruitment incubated for 150 mins by b...


Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113805
BindingDB Entry DOI: 10.7270/Q2QF8XRP
More data for this
Ligand-Target Pair
N-formyl peptide receptor 2


(Homo sapiens (Human))
BDBM50582813
PNG
(CHEMBL5093348)
Show SMILES Brc1ccc(NC(=O)NC2CCN(C3CCN(CC3)c3ncccn3)C2=O)cc1
PDB

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n/an/an/an/a 385n/an/an/an/a


TBA

Assay Description
Agonist activity at FPRL1 (unknown origin) expressed in CHO-K1 cells assessed as stimulation of beta-arrestin recruitment incubated for 150 mins by b...


Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113805
BindingDB Entry DOI: 10.7270/Q2QF8XRP
More data for this
Ligand-Target Pair
N-formyl peptide receptor 2


(Homo sapiens (Human))
BDBM50582815
PNG
(CHEMBL5078594)
Show SMILES Cc1nn(C)cc1N1CCC(NC(=O)Nc2ccc(Br)cc2)C1=O
PDB

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n/an/an/an/a 740n/an/an/an/a


TBA

Assay Description
Agonist activity at FPRL1 (unknown origin) expressed in CHO-K1 cells assessed as stimulation of beta-arrestin recruitment incubated for 150 mins by b...


Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113805
BindingDB Entry DOI: 10.7270/Q2QF8XRP
More data for this
Ligand-Target Pair
N-formyl peptide receptor 2


(Homo sapiens (Human))
BDBM50582824
PNG
(CHEMBL5088171)
Show SMILES Brc1ccc(NC(=O)NC2CCN(C2=O)c2cnn(c2)-c2ccncc2)cc1
PDB

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n/an/an/an/a 3.76E+3n/an/an/an/a


TBA

Assay Description
Agonist activity at FPRL1 (unknown origin) expressed in CHO-K1 cells assessed as stimulation of beta-arrestin recruitment incubated for 150 mins by b...


Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113805
BindingDB Entry DOI: 10.7270/Q2QF8XRP
More data for this
Ligand-Target Pair
N-formyl peptide receptor 2


(Homo sapiens (Human))
BDBM50582817
PNG
(CHEMBL5076914)
Show SMILES Brc1ccc(NC(=O)NC2CCN(C2=O)c2ccccc2)cc1
PDB

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n/an/an/an/a 300n/an/an/an/a


TBA

Assay Description
Agonist activity at FPRL1 (unknown origin) expressed in CHO-K1 cells assessed as stimulation of beta-arrestin recruitment incubated for 150 mins by b...


Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113805
BindingDB Entry DOI: 10.7270/Q2QF8XRP
More data for this
Ligand-Target Pair
N-formyl peptide receptor 2


(Homo sapiens (Human))
BDBM50582818
PNG
(CHEMBL5085666)
Show SMILES Fc1ccc(cc1)N1CCC(NC(=O)Nc2ccc(Br)cc2)C1=O
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n/an/an/an/a 510n/an/an/an/a


TBA

Assay Description
Agonist activity at FPRL1 (unknown origin) expressed in CHO-K1 cells assessed as stimulation of beta-arrestin recruitment incubated for 150 mins by b...


Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113805
BindingDB Entry DOI: 10.7270/Q2QF8XRP
More data for this
Ligand-Target Pair
N-formyl peptide receptor 2


(Homo sapiens (Human))
BDBM50582819
PNG
(CHEMBL5087710)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N1CCC(NC(=O)Nc2ccc(Br)cc2)C1=O
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n/an/an/an/a 6.30E+3n/an/an/an/a


TBA

Assay Description
Agonist activity at FPRL1 (unknown origin) expressed in CHO-K1 cells assessed as stimulation of beta-arrestin recruitment incubated for 150 mins by b...


Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113805
BindingDB Entry DOI: 10.7270/Q2QF8XRP
More data for this
Ligand-Target Pair
N-formyl peptide receptor 2


(Homo sapiens (Human))
BDBM50582820
PNG
(CHEMBL5090603)
Show SMILES CC(C)(C)OC(=O)N1CCC(CN2CCC(NC(=O)Nc3ccc(Br)cc3)C2=O)CC1
PDB

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n/an/an/an/a 2.16E+3n/an/an/an/a


TBA

Assay Description
Agonist activity at FPRL1 (unknown origin) expressed in CHO-K1 cells assessed as stimulation of beta-arrestin recruitment incubated for 150 mins by b...


Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113805
BindingDB Entry DOI: 10.7270/Q2QF8XRP
More data for this
Ligand-Target Pair
N-formyl peptide receptor 2


(Homo sapiens (Human))
BDBM50582821
PNG
(CHEMBL5084374)
Show SMILES Brc1ccc(NC(=O)NC2CCN(CC3CCNCC3)C2=O)cc1
PDB

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n/an/an/an/a 3.29E+3n/an/an/an/a


TBA

Assay Description
Agonist activity at FPRL1 (unknown origin) expressed in CHO-K1 cells assessed as stimulation of beta-arrestin recruitment incubated for 150 mins by b...


Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113805
BindingDB Entry DOI: 10.7270/Q2QF8XRP
More data for this
Ligand-Target Pair
N-formyl peptide receptor 2


(Homo sapiens (Human))
BDBM50582822
PNG
(CHEMBL5075000)
Show SMILES Brc1ccc(NC(=O)NC2CCN(C3CCNCC3)C2=O)cc1
PDB

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n/an/an/an/a 1.03E+3n/an/an/an/a


TBA

Assay Description
Agonist activity at FPRL1 (unknown origin) expressed in CHO-K1 cells assessed as stimulation of beta-arrestin recruitment incubated for 150 mins by b...


Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113805
BindingDB Entry DOI: 10.7270/Q2QF8XRP
More data for this
Ligand-Target Pair
fMet-Leu-Phe receptor


(Homo sapiens (Human))
BDBM50582817
PNG
(CHEMBL5076914)
Show SMILES Brc1ccc(NC(=O)NC2CCN(C2=O)c2ccccc2)cc1
PDB

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n/an/an/an/a 1.74E+3n/an/an/an/a


TBA

Assay Description
Agonist activity at human FPR1 expressed in HEK293-A cells assessed as ERK phosphorylation level incubated for 5 mins by ELISA assay


Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113805
BindingDB Entry DOI: 10.7270/Q2QF8XRP
More data for this
Ligand-Target Pair
N-formyl peptide receptor 2


(Homo sapiens (Human))
BDBM50582815
PNG
(CHEMBL5078594)
Show SMILES Cc1nn(C)cc1N1CCC(NC(=O)Nc2ccc(Br)cc2)C1=O
PDB

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n/an/an/an/a 4.88E+3n/an/an/an/a


TBA

Assay Description
Agonist activity at human FPR2 expressed in HEK293-A cells assessed as ERK phosphorylation level incubated for 5 mins by ELISA assay


Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113805
BindingDB Entry DOI: 10.7270/Q2QF8XRP
More data for this
Ligand-Target Pair
N-formyl peptide receptor 2


(Homo sapiens (Human))
BDBM50582809
PNG
(CHEMBL5070452)
Show SMILES Brc1ccc(NC(=O)NC2CCN(C3CCN(Cc4ccccc4)CC3)C2=O)cc1
PDB

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n/an/an/an/a 350n/an/an/an/a


TBA

Assay Description
Agonist activity at FPRL1 (unknown origin) expressed in CHO-K1 cells assessed as increase in calcium mobilization incubated for 2.5 hrs by cellular b...


Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113805
BindingDB Entry DOI: 10.7270/Q2QF8XRP
More data for this
Ligand-Target Pair