Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Cytochrome P450 11B2, mitochondrial (Homo sapiens (Human)) | BDBM50323351 (6-[(S)-1-(4-Chloro-phenyl)-ethyl]-4-isobutyl-6,7-d...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.40 | n/a | n/a | n/a | n/a | n/a | n/a |
AbbVie Bioresearch Center Curated by ChEMBL | Assay Description Inhibition of human CYP11B2 | Bioorg Med Chem Lett 23: 5471-83 (2013) Article DOI: 10.1016/j.bmcl.2013.08.003 BindingDB Entry DOI: 10.7270/Q2R49S6F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 11B2, mitochondrial (Homo sapiens (Human)) | BDBM50323353 (1-{6-[(S)-1-(4-Chloro-phenyl)-ethyl]-5,5-dioxo-4,5...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a |
AbbVie Bioresearch Center Curated by ChEMBL | Assay Description Inhibition of human CYP11B2 | Bioorg Med Chem Lett 23: 5471-83 (2013) Article DOI: 10.1016/j.bmcl.2013.08.003 BindingDB Entry DOI: 10.7270/Q2R49S6F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475561 (1-[6-Chloro-5-(4-chloro-phenylmethanesulfonyl)-1H-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 15.8 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description The PHD2181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypept... | US Patent US10851083 (2020) BindingDB Entry DOI: 10.7270/Q25B05K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475561 (1-[6-Chloro-5-(4-chloro-phenylmethanesulfonyl)-1H-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 15.8 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The PHD2 181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypep... | Citation and Details BindingDB Entry DOI: 10.7270/Q2V69PHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475567 (1-[6-Chloro-5-(4-trifluoromethyl-phenylmethanesulf...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description The PHD2181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypept... | US Patent US10851083 (2020) BindingDB Entry DOI: 10.7270/Q25B05K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475569 (1-[6-Chloro-5-(2'-cyano-biphenyl-4-ylmethanesulfon...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description The PHD2181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypept... | US Patent US10851083 (2020) BindingDB Entry DOI: 10.7270/Q25B05K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475479 (1-[6-Chloro-5-(4-methoxy-phenylmethanesulfonyl)-1H...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description The PHD2181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypept... | US Patent US10851083 (2020) BindingDB Entry DOI: 10.7270/Q25B05K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475563 (1-(6-Chloro-5-cyclohexylmethanesulfonyl-1H- | US10...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The PHD2 181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypep... | Citation and Details BindingDB Entry DOI: 10.7270/Q2V69PHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475557 (1-[6-Chloro-5-(4-methyl-benzylsulfanyl)-1H- | US10...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description The PHD2181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypept... | US Patent US10851083 (2020) BindingDB Entry DOI: 10.7270/Q25B05K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475567 (1-[6-Chloro-5-(4-trifluoromethyl-phenylmethanesulf...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The PHD2 181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypep... | Citation and Details BindingDB Entry DOI: 10.7270/Q2V69PHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475569 (1-[6-Chloro-5-(2'-cyano-biphenyl-4-ylmethanesulfon...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The PHD2 181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypep... | Citation and Details BindingDB Entry DOI: 10.7270/Q2V69PHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475563 (1-(6-Chloro-5-cyclohexylmethanesulfonyl-1H- | US10...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description The PHD2181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypept... | US Patent US10851083 (2020) BindingDB Entry DOI: 10.7270/Q25B05K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475479 (1-[6-Chloro-5-(4-methoxy-phenylmethanesulfonyl)-1H...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The PHD2 181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypep... | Citation and Details BindingDB Entry DOI: 10.7270/Q2V69PHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475557 (1-[6-Chloro-5-(4-methyl-benzylsulfanyl)-1H- | US10...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The PHD2 181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypep... | Citation and Details BindingDB Entry DOI: 10.7270/Q2V69PHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475485 (1-(6-Methanesulfonyl-5-trifluoromethyl-1H- | US108...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 25.1 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The PHD2 181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypep... | Citation and Details BindingDB Entry DOI: 10.7270/Q2V69PHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475543 (1-(5-Ethylsulfonyl-6-trifluoromethoxy-1H-benzoimid...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 25.1 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description The PHD2181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypept... | US Patent US10851083 (2020) BindingDB Entry DOI: 10.7270/Q25B05K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475549 (1-(5-Benzenesulfonyl-6-trifluoromethyl-1H- | US108...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 25.1 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description The PHD2181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypept... | US Patent US10851083 (2020) BindingDB Entry DOI: 10.7270/Q25B05K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475550 (1-[5-(4-Methoxy-benzenesulfonyl)-6-trifluoromethyl...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 25.1 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description The PHD2181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypept... | US Patent US10851083 (2020) BindingDB Entry DOI: 10.7270/Q25B05K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475562 (1-[6-Chloro-5-(3-chloro-phenylmethanesulfonyl)-1H-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 25.1 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description The PHD2181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypept... | US Patent US10851083 (2020) BindingDB Entry DOI: 10.7270/Q25B05K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475564 (1-[6-Chloro-5-(3,4-dichloro-phenylmethanesulfonyl)...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 25.1 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description The PHD2181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypept... | US Patent US10851083 (2020) BindingDB Entry DOI: 10.7270/Q25B05K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475568 (1-[5-(2,4-Bis-trifluoromethyl-phenylmethanesulfony...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 25.1 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description The PHD2181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypept... | US Patent US10851083 (2020) BindingDB Entry DOI: 10.7270/Q25B05K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475542 (1-(5-Ethylsulfonyl-6-trifluoromethyl-1H-benzoimida...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 25.1 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The PHD2 181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypep... | Citation and Details BindingDB Entry DOI: 10.7270/Q2V69PHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475543 (1-(5-Ethylsulfonyl-6-trifluoromethoxy-1H-benzoimid...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 25.1 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The PHD2 181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypep... | Citation and Details BindingDB Entry DOI: 10.7270/Q2V69PHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475549 (1-(5-Benzenesulfonyl-6-trifluoromethyl-1H- | US108...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 25.1 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The PHD2 181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypep... | Citation and Details BindingDB Entry DOI: 10.7270/Q2V69PHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475550 (1-[5-(4-Methoxy-benzenesulfonyl)-6-trifluoromethyl...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 25.1 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The PHD2 181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypep... | Citation and Details BindingDB Entry DOI: 10.7270/Q2V69PHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475562 (1-[6-Chloro-5-(3-chloro-phenylmethanesulfonyl)-1H-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 25.1 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The PHD2 181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypep... | Citation and Details BindingDB Entry DOI: 10.7270/Q2V69PHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475564 (1-[6-Chloro-5-(3,4-dichloro-phenylmethanesulfonyl)...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 25.1 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The PHD2 181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypep... | Citation and Details BindingDB Entry DOI: 10.7270/Q2V69PHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475568 (1-[5-(2,4-Bis-trifluoromethyl-phenylmethanesulfony...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 25.1 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The PHD2 181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypep... | Citation and Details BindingDB Entry DOI: 10.7270/Q2V69PHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475401 (1-{5-[3-(2-Chloro-benzyloxy)-phenyl]-1H-benzoimida...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 25.1 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The PHD2 181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypep... | Citation and Details BindingDB Entry DOI: 10.7270/Q2V69PHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475401 (1-{5-[3-(2-Chloro-benzyloxy)-phenyl]-1H-benzoimida...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 25.1 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description The PHD2181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypept... | US Patent US10851083 (2020) BindingDB Entry DOI: 10.7270/Q25B05K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475485 (1-(6-Methanesulfonyl-5-trifluoromethyl-1H- | US108...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 25.1 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description The PHD2181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypept... | US Patent US10851083 (2020) BindingDB Entry DOI: 10.7270/Q25B05K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475542 (1-(5-Ethylsulfonyl-6-trifluoromethyl-1H-benzoimida...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 25.1 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description The PHD2181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypept... | US Patent US10851083 (2020) BindingDB Entry DOI: 10.7270/Q25B05K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475471 (1-(5-Benzenesulfonyl-6-chloro-1H-benzoimidazol-2-y...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 26.9 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description The PHD2181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypept... | US Patent US10851083 (2020) BindingDB Entry DOI: 10.7270/Q25B05K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475471 (1-(5-Benzenesulfonyl-6-chloro-1H-benzoimidazol-2-y...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 26.9 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The PHD2 181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypep... | Citation and Details BindingDB Entry DOI: 10.7270/Q2V69PHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475443 (1-[5-(4-Chloro-phenoxy)-6-trifluoromethyl-1H- | US...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 31.6 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The PHD2 181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypep... | Citation and Details BindingDB Entry DOI: 10.7270/Q2V69PHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475494 (1-[6-(Propane-1-sulfonyl)-5-trifluoromethoxy-1H- |...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 31.6 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description The PHD2181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypept... | US Patent US10851083 (2020) BindingDB Entry DOI: 10.7270/Q25B05K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475480 (1-[6-Chloro-5-(4-fluoro-phenylmethanesulfonyl)-1H-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 31.6 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The PHD2 181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypep... | Citation and Details BindingDB Entry DOI: 10.7270/Q2V69PHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475481 (1-[6-Chloro-5-(2-chloro-phenylmethanesulfonyl)-1H-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 31.6 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The PHD2 181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypep... | Citation and Details BindingDB Entry DOI: 10.7270/Q2V69PHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475488 (1-(6-Methanesulfonyl-5-trifluoromethoxy-1H- | US10...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 31.6 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The PHD2 181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypep... | Citation and Details BindingDB Entry DOI: 10.7270/Q2V69PHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475490 (1-[5-Chloro-6-(propane-1-sulfonyl)-1H-benzoimidazo...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 31.6 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The PHD2 181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypep... | Citation and Details BindingDB Entry DOI: 10.7270/Q2V69PHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475492 (1-[6-(Propane-1-sulfonyl)-5-trifluoromethyl-1H- | ...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 31.6 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The PHD2 181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypep... | Citation and Details BindingDB Entry DOI: 10.7270/Q2V69PHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475494 (1-[6-(Propane-1-sulfonyl)-5-trifluoromethoxy-1H- |...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 31.6 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The PHD2 181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypep... | Citation and Details BindingDB Entry DOI: 10.7270/Q2V69PHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475548 (1-[5-(4-Methoxy-phenylsulfanyl)-6-trifluoromethyl-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 31.6 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description The PHD2181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypept... | US Patent US10851083 (2020) BindingDB Entry DOI: 10.7270/Q25B05K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475560 (1-[6-Chloro-5-(2'-cyano-biphenyl-4-ylmethylsulfany...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 31.6 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description The PHD2181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypept... | US Patent US10851083 (2020) BindingDB Entry DOI: 10.7270/Q25B05K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475565 (1-[6-Chloro-5-(2,6-dichloro-phenylmethanesulfonyl)...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 31.6 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description The PHD2181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypept... | US Patent US10851083 (2020) BindingDB Entry DOI: 10.7270/Q25B05K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475548 (1-[5-(4-Methoxy-phenylsulfanyl)-6-trifluoromethyl-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 31.6 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The PHD2 181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypep... | Citation and Details BindingDB Entry DOI: 10.7270/Q2V69PHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475560 (1-[6-Chloro-5-(2'-cyano-biphenyl-4-ylmethylsulfany...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 31.6 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The PHD2 181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypep... | Citation and Details BindingDB Entry DOI: 10.7270/Q2V69PHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475565 (1-[6-Chloro-5-(2,6-dichloro-phenylmethanesulfonyl)...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 31.6 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The PHD2 181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypep... | Citation and Details BindingDB Entry DOI: 10.7270/Q2V69PHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475400 (1-{5-[3-(3-Chloro-benzyloxy)-phenyl]-1H-benzoimida...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 31.6 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The PHD2 181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypep... | Citation and Details BindingDB Entry DOI: 10.7270/Q2V69PHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Egl nine homolog 1 [181-417] (Homo sapiens (Human)) | BDBM475428 (1-(6-Chloro-5-nitro-1H-benzoimidazol-2-yl)-1H-pyra...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 31.6 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The PHD2 181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypep... | Citation and Details BindingDB Entry DOI: 10.7270/Q2V69PHV | |||||||||||
More data for this Ligand-Target Pair |
Displayed 1 to 50 (of 523 total ) | Next | Last >> |