Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Growth factor receptor-bound protein 2 (Homo sapiens (Human)) | BDBM50241558![]() (8-O-methylsclerotiorinamine | CHEMBL487793) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents | PubMed | n/a | n/a | 5.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Korea Research Institute of Bioscience & Biotechnology Curated by ChEMBL | Assay Description Inhibition of GST tagged Grb2 SH2 domain (unknown origin) binding to Shc-derived [3H]phosphopeptide | J Nat Prod 63: 1303-5 (2000) BindingDB Entry DOI: 10.7270/Q21R6Q7M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
RYamide receptor (Drosophila melanogaster) | BDBM50192749![]() (CHEMBL3944838) | UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 6.10E+3 | n/a | n/a | n/a | n/a |
Gwangju Institute of Science and Technology Curated by ChEMBL | Assay Description Agonist activity at Drosophila melanogaster RYamide receptor expressed in wild type CHO-K1 cells assessed as increase in calcium level after 20 secs ... | Bioorg Med Chem Lett 26: 5116-5118 (2016) Article DOI: 10.1016/j.bmcl.2016.08.039 BindingDB Entry DOI: 10.7270/Q2DF6T58 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
RYamide receptor (Drosophila melanogaster) | BDBM50192748![]() (CHEMBL3974271) | UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 6.80E+3 | n/a | n/a | n/a | n/a |
Gwangju Institute of Science and Technology Curated by ChEMBL | Assay Description Agonist activity at Drosophila melanogaster RYamide receptor expressed in wild type CHO-K1 cells assessed as increase in calcium level after 20 secs ... | Bioorg Med Chem Lett 26: 5116-5118 (2016) Article DOI: 10.1016/j.bmcl.2016.08.039 BindingDB Entry DOI: 10.7270/Q2DF6T58 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
RYamide receptor (Drosophila melanogaster) | BDBM50192742![]() (CHEMBL3982272) | UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.09E+4 | n/a | n/a | n/a | n/a |
Gwangju Institute of Science and Technology Curated by ChEMBL | Assay Description Agonist activity at Drosophila melanogaster RYamide receptor expressed in wild type CHO-K1 cells assessed as increase in calcium level after 20 secs ... | Bioorg Med Chem Lett 26: 5116-5118 (2016) Article DOI: 10.1016/j.bmcl.2016.08.039 BindingDB Entry DOI: 10.7270/Q2DF6T58 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
RYamide receptor (Drosophila melanogaster) | BDBM50192747![]() (CHEMBL3935892) | UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 5.90E+3 | n/a | n/a | n/a | n/a |
Gwangju Institute of Science and Technology Curated by ChEMBL | Assay Description Agonist activity at Drosophila melanogaster RYamide receptor expressed in wild type CHO-K1 cells assessed as increase in calcium level after 20 secs ... | Bioorg Med Chem Lett 26: 5116-5118 (2016) Article DOI: 10.1016/j.bmcl.2016.08.039 BindingDB Entry DOI: 10.7270/Q2DF6T58 | |||||||||||
More data for this Ligand-Target Pair |