BindingDB PrimarySearch

Found 8 hits with Last Name = 'désaubry' and Initial = 'l'
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
cGMP-dependent 3',5'-cyclic phosphodiesterase (Homo sapiens (Human))	BDBM50034908 ((2R,3S)-3-((R)-6-Amino-purin-9-yl)-nonan-2-ol \| (2...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Similars	Article PubMed	2.80E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
UPR 421 du CNRS Curated by ChEMBL					Assay Description Inhibition of Phosphodiesterase 2				J Med Chem 40: 1768-70 (1997) Article DOI: 10.1021/jm960827x BindingDB Entry DOI: 10.7270/Q25T3M4T
UPR 421 du CNRS Curated by ChEMBL					More data for this Ligand-Target Pair
cGMP-specific 3',5'-cyclic phosphodiesterase (Homo sapiens (Human))	BDBM50058210 (CHEMBL445098 \| [9-(2-Fluoro-benzyl)-9H-purin-6-yl]...) Show SMILES CNc1ncnc2n(Cc3ccccc3F)cnc12 Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Similars	Article PubMed	6.50E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
UPR 421 du CNRS Curated by ChEMBL					Assay Description Inhibition of Phosphodiesterase 5				J Med Chem 40: 1768-70 (1997) Article DOI: 10.1021/jm960827x BindingDB Entry DOI: 10.7270/Q25T3M4T
UPR 421 du CNRS Curated by ChEMBL					More data for this Ligand-Target Pair
cGMP-dependent 3',5'-cyclic phosphodiesterase (Homo sapiens (Human))	BDBM50058210 (CHEMBL445098 \| [9-(2-Fluoro-benzyl)-9H-purin-6-yl]...) Show SMILES CNc1ncnc2n(Cc3ccccc3F)cnc12 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Similars	Article PubMed	1.22E+5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
UPR 421 du CNRS Curated by ChEMBL					Assay Description Inhibition of Phosphodiesterase 2				J Med Chem 40: 1768-70 (1997) Article DOI: 10.1021/jm960827x BindingDB Entry DOI: 10.7270/Q25T3M4T
UPR 421 du CNRS Curated by ChEMBL					More data for this Ligand-Target Pair
cGMP-specific 3',5'-cyclic phosphodiesterase (Homo sapiens (Human))	BDBM14361 ((R,S)-Rolipram \| 4-(3-cyclopentyloxy-4-methoxy-phe...) Show SMILES COc1ccc(cc1OC1CCCC1)C1CNC(=O)C1 Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars	Article PubMed	>2.00E+5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
UPR 421 du CNRS Curated by ChEMBL					Assay Description Inhibition of Phosphodiesterase 5				J Med Chem 40: 1768-70 (1997) Article DOI: 10.1021/jm960827x BindingDB Entry DOI: 10.7270/Q25T3M4T
UPR 421 du CNRS Curated by ChEMBL					More data for this Ligand-Target Pair
cGMP-specific 3',5'-cyclic phosphodiesterase (Homo sapiens (Human))	BDBM50034908 ((2R,3S)-3-((R)-6-Amino-purin-9-yl)-nonan-2-ol \| (2...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Similars	Article PubMed	>2.00E+5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
UPR 421 du CNRS Curated by ChEMBL					Assay Description Inhibition of Phosphodiesterase 5				J Med Chem 40: 1768-70 (1997) Article DOI: 10.1021/jm960827x BindingDB Entry DOI: 10.7270/Q25T3M4T
UPR 421 du CNRS Curated by ChEMBL					More data for this Ligand-Target Pair
cGMP-dependent 3',5'-cyclic phosphodiesterase (Homo sapiens (Human))	BDBM14361 ((R,S)-Rolipram \| 4-(3-cyclopentyloxy-4-methoxy-phe...) Show SMILES COc1ccc(cc1OC1CCCC1)C1CNC(=O)C1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars	Article PubMed	>2.00E+5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
UPR 421 du CNRS Curated by ChEMBL					Assay Description Inhibition of Phosphodiesterase 2				J Med Chem 40: 1768-70 (1997) Article DOI: 10.1021/jm960827x BindingDB Entry DOI: 10.7270/Q25T3M4T
UPR 421 du CNRS Curated by ChEMBL					More data for this Ligand-Target Pair
cGMP-specific 3',5'-cyclic phosphodiesterase (Homo sapiens (Human))	BDBM50058212 (9-(2-fluorobenzyl)-N-methyl-2-(trifluoromethyl)-9H...) Show SMILES CNc1nc(nc2n(Cc3ccccc3F)cnc12)C(F)(F)F Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	5.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
UPR 421 du CNRS Curated by ChEMBL					Assay Description Inhibition of phosphodiesterase 5				J Med Chem 40: 1768-70 (1997) Article DOI: 10.1021/jm960827x BindingDB Entry DOI: 10.7270/Q25T3M4T
UPR 421 du CNRS Curated by ChEMBL					More data for this Ligand-Target Pair
Adenosine receptor A1 (Homo sapiens (Human))	BDBM50058210 (CHEMBL445098 \| [9-(2-Fluoro-benzyl)-9H-purin-6-yl]...) Show SMILES CNc1ncnc2n(Cc3ccccc3F)cnc12 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
UPR 421 du CNRS Curated by ChEMBL					Assay Description Displacement of [3H]CHA from Adenosine A1 receptor				J Med Chem 40: 1768-70 (1997) Article DOI: 10.1021/jm960827x BindingDB Entry DOI: 10.7270/Q25T3M4T
UPR 421 du CNRS Curated by ChEMBL					More data for this Ligand-Target Pair