Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Estrogen receptor (Homo sapiens (Human)) | BDBM50294178![]() (CHEMBL4160682) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 33 | n/a | n/a | n/a | n/a | n/a | n/a |
Central University of Punjab Curated by ChEMBL | Assay Description Displacement of fluoromone TM from recombinant human ERalpha after 2 hrs by fluorescence polarization analysis | Eur J Med Chem 146: 206-219 (2018) Article DOI: 10.1016/j.ejmech.2018.01.051 BindingDB Entry DOI: 10.7270/Q20C4Z9J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor (Homo sapiens (Human)) | BDBM50294174![]() (CHEMBL4170939) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 47 | n/a | n/a | n/a | n/a | n/a | n/a |
Central University of Punjab Curated by ChEMBL | Assay Description Displacement of fluoromone TM from recombinant human ERalpha after 2 hrs by fluorescence polarization analysis | Eur J Med Chem 146: 206-219 (2018) Article DOI: 10.1016/j.ejmech.2018.01.051 BindingDB Entry DOI: 10.7270/Q20C4Z9J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor (Homo sapiens (Human)) | BDBM50294181![]() (CHEMBL4169456) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 74 | n/a | n/a | n/a | n/a | n/a | n/a |
Central University of Punjab Curated by ChEMBL | Assay Description Displacement of fluoromone TM from recombinant human ERalpha after 2 hrs by fluorescence polarization analysis | Eur J Med Chem 146: 206-219 (2018) Article DOI: 10.1016/j.ejmech.2018.01.051 BindingDB Entry DOI: 10.7270/Q20C4Z9J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor (Homo sapiens (Human)) | BDBM50294182![]() (CHEMBL4161120) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 77 | n/a | n/a | n/a | n/a | n/a | n/a |
Central University of Punjab Curated by ChEMBL | Assay Description Displacement of fluoromone TM from recombinant human ERalpha after 2 hrs by fluorescence polarization analysis | Eur J Med Chem 146: 206-219 (2018) Article DOI: 10.1016/j.ejmech.2018.01.051 BindingDB Entry DOI: 10.7270/Q20C4Z9J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor (Homo sapiens (Human)) | BDBM50294175![]() (CHEMBL4167567) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 80 | n/a | n/a | n/a | n/a | n/a | n/a |
Central University of Punjab Curated by ChEMBL | Assay Description Displacement of fluoromone TM from recombinant human ERalpha after 2 hrs by fluorescence polarization analysis | Eur J Med Chem 146: 206-219 (2018) Article DOI: 10.1016/j.ejmech.2018.01.051 BindingDB Entry DOI: 10.7270/Q20C4Z9J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor (Homo sapiens (Human)) | BDBM50294185![]() (CHEMBL4168369) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 192 | n/a | n/a | n/a | n/a | n/a | n/a |
Central University of Punjab Curated by ChEMBL | Assay Description Displacement of fluoromone TM from recombinant human ERalpha after 2 hrs by fluorescence polarization analysis | Eur J Med Chem 146: 206-219 (2018) Article DOI: 10.1016/j.ejmech.2018.01.051 BindingDB Entry DOI: 10.7270/Q20C4Z9J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor (Homo sapiens (Human)) | BDBM50294176![]() (CHEMBL4164124) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 202 | n/a | n/a | n/a | n/a | n/a | n/a |
Central University of Punjab Curated by ChEMBL | Assay Description Displacement of fluoromone TM from recombinant human ERalpha after 2 hrs by fluorescence polarization analysis | Eur J Med Chem 146: 206-219 (2018) Article DOI: 10.1016/j.ejmech.2018.01.051 BindingDB Entry DOI: 10.7270/Q20C4Z9J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor (Homo sapiens (Human)) | BDBM50294179![]() (CHEMBL4168602) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 259 | n/a | n/a | n/a | n/a | n/a | n/a |
Central University of Punjab Curated by ChEMBL | Assay Description Displacement of fluoromone TM from recombinant human ERalpha after 2 hrs by fluorescence polarization analysis | Eur J Med Chem 146: 206-219 (2018) Article DOI: 10.1016/j.ejmech.2018.01.051 BindingDB Entry DOI: 10.7270/Q20C4Z9J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor (Homo sapiens (Human)) | BDBM50294180![]() (CHEMBL4164944) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 300 | n/a | n/a | n/a | n/a | n/a | n/a |
Central University of Punjab Curated by ChEMBL | Assay Description Displacement of fluoromone TM from recombinant human ERalpha after 2 hrs by fluorescence polarization analysis | Eur J Med Chem 146: 206-219 (2018) Article DOI: 10.1016/j.ejmech.2018.01.051 BindingDB Entry DOI: 10.7270/Q20C4Z9J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor (Homo sapiens (Human)) | BDBM50294177![]() (CHEMBL4170073) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 387 | n/a | n/a | n/a | n/a | n/a | n/a |
Central University of Punjab Curated by ChEMBL | Assay Description Displacement of fluoromone TM from recombinant human ERalpha after 2 hrs by fluorescence polarization analysis | Eur J Med Chem 146: 206-219 (2018) Article DOI: 10.1016/j.ejmech.2018.01.051 BindingDB Entry DOI: 10.7270/Q20C4Z9J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor (Homo sapiens (Human)) | BDBM50294183![]() (CHEMBL4171721) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 539 | n/a | n/a | n/a | n/a | n/a | n/a |
Central University of Punjab Curated by ChEMBL | Assay Description Displacement of fluoromone TM from recombinant human ERalpha after 2 hrs by fluorescence polarization analysis | Eur J Med Chem 146: 206-219 (2018) Article DOI: 10.1016/j.ejmech.2018.01.051 BindingDB Entry DOI: 10.7270/Q20C4Z9J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor (Homo sapiens (Human)) | BDBM50454051![]() (CHEMBL4207636) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.66E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Central University of Punjab Curated by ChEMBL | Assay Description Displacement of Fluormone-tagged ES2 from human recombinant ERalpha after 2 hrs by fluorescence polarization assay | Bioorg Med Chem 26: 266-277 (2018) Article DOI: 10.1016/j.bmc.2017.11.040 BindingDB Entry DOI: 10.7270/Q2K64MNF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor (Homo sapiens (Human)) | BDBM50454049![]() (CHEMBL4214332) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.84E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Central University of Punjab Curated by ChEMBL | Assay Description Displacement of Fluormone-tagged ES2 from human recombinant ERalpha after 2 hrs by fluorescence polarization assay | Bioorg Med Chem 26: 266-277 (2018) Article DOI: 10.1016/j.bmc.2017.11.040 BindingDB Entry DOI: 10.7270/Q2K64MNF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor (Homo sapiens (Human)) | BDBM50454048![]() (CHEMBL4213826) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.66E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Central University of Punjab Curated by ChEMBL | Assay Description Displacement of Fluormone-tagged ES2 from human recombinant ERalpha after 2 hrs by fluorescence polarization assay | Bioorg Med Chem 26: 266-277 (2018) Article DOI: 10.1016/j.bmc.2017.11.040 BindingDB Entry DOI: 10.7270/Q2K64MNF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor (Homo sapiens (Human)) | BDBM50099585![]() (1-(4-(2-(azepan-1-yl)ethoxy)benzyl)-2-(4-hydroxyph...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL DrugBank MCE PC cid PC sid PDB UniChem Patents Similars | PDB Article PubMed | n/a | n/a | 3.17E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Central University of Punjab Curated by ChEMBL | Assay Description Displacement of Fluormone-tagged ES2 from human recombinant ERalpha after 2 hrs by fluorescence polarization assay | Bioorg Med Chem 26: 266-277 (2018) Article DOI: 10.1016/j.bmc.2017.11.040 BindingDB Entry DOI: 10.7270/Q2K64MNF | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
Estrogen receptor (Homo sapiens (Human)) | BDBM50454053![]() (CHEMBL4203135) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.12E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Central University of Punjab Curated by ChEMBL | Assay Description Displacement of Fluormone-tagged ES2 from human recombinant ERalpha after 2 hrs by fluorescence polarization assay | Bioorg Med Chem 26: 266-277 (2018) Article DOI: 10.1016/j.bmc.2017.11.040 BindingDB Entry DOI: 10.7270/Q2K64MNF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor (Homo sapiens (Human)) | BDBM50454050![]() (CHEMBL4209434) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Central University of Punjab Curated by ChEMBL | Assay Description Displacement of Fluormone-tagged ES2 from human recombinant ERalpha after 2 hrs by fluorescence polarization assay | Bioorg Med Chem 26: 266-277 (2018) Article DOI: 10.1016/j.bmc.2017.11.040 BindingDB Entry DOI: 10.7270/Q2K64MNF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor (Homo sapiens (Human)) | BDBM50454057![]() (CHEMBL4218272) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.08E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Central University of Punjab Curated by ChEMBL | Assay Description Displacement of Fluormone-tagged ES2 from human recombinant ERalpha after 2 hrs by fluorescence polarization assay | Bioorg Med Chem 26: 266-277 (2018) Article DOI: 10.1016/j.bmc.2017.11.040 BindingDB Entry DOI: 10.7270/Q2K64MNF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor (Homo sapiens (Human)) | BDBM50454055![]() (CHEMBL4207948) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.11E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Central University of Punjab Curated by ChEMBL | Assay Description Displacement of Fluormone-tagged ES2 from human recombinant ERalpha after 2 hrs by fluorescence polarization assay | Bioorg Med Chem 26: 266-277 (2018) Article DOI: 10.1016/j.bmc.2017.11.040 BindingDB Entry DOI: 10.7270/Q2K64MNF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor (Homo sapiens (Human)) | BDBM50454056![]() (CHEMBL4215448) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.56E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Central University of Punjab Curated by ChEMBL | Assay Description Displacement of Fluormone-tagged ES2 from human recombinant ERalpha after 2 hrs by fluorescence polarization assay | Bioorg Med Chem 26: 266-277 (2018) Article DOI: 10.1016/j.bmc.2017.11.040 BindingDB Entry DOI: 10.7270/Q2K64MNF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor (Homo sapiens (Human)) | BDBM50454052![]() (CHEMBL4206393) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.82E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Central University of Punjab Curated by ChEMBL | Assay Description Displacement of Fluormone-tagged ES2 from human recombinant ERalpha after 2 hrs by fluorescence polarization assay | Bioorg Med Chem 26: 266-277 (2018) Article DOI: 10.1016/j.bmc.2017.11.040 BindingDB Entry DOI: 10.7270/Q2K64MNF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor (Homo sapiens (Human)) | BDBM50454054![]() (CHEMBL4218756) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.87E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Central University of Punjab Curated by ChEMBL | Assay Description Displacement of Fluormone-tagged ES2 from human recombinant ERalpha after 2 hrs by fluorescence polarization assay | Bioorg Med Chem 26: 266-277 (2018) Article DOI: 10.1016/j.bmc.2017.11.040 BindingDB Entry DOI: 10.7270/Q2K64MNF | |||||||||||
More data for this Ligand-Target Pair |