Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Aspartate--tRNA ligase (Escherichia coli) | BDBM50339907![]() (((S)-2-amino-3-carboxypropanoyl)(((2R,3S,4R,5R)-5-...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Similars | Article PubMed | 0.0520 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
KU Leuven Curated by ChEMBL | Assay Description Inhibition of Escherichia coli BL21(DE3) Aspartyl-tRNA synthetase assessed as reduction in tRNA aminoacylation preincubated for 10 mins with Escheric... | Eur J Med Chem 148: 384-396 (2018) Article DOI: 10.1016/j.ejmech.2018.02.013 BindingDB Entry DOI: 10.7270/Q2057JJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Leucine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50458119![]() (Leusa) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase MCE PC cid PC sid PDB UniChem | PDB Article PubMed | 0.139 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
KU Leuven Curated by ChEMBL | Assay Description Inhibition of Escherichia coli BL21(DE3) Leucyl-tRNA synthetase assessed as reduction in tRNA aminoacylation preincubated for 10 mins with Escherichi... | Eur J Med Chem 148: 384-396 (2018) Article DOI: 10.1016/j.ejmech.2018.02.013 BindingDB Entry DOI: 10.7270/Q2057JJS | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
Serine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50339906![]() (((2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-dihyd...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL MCE MMDB PC cid PC sid PDB UniChem Similars | PDB Article PubMed | 0.180 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
KU Leuven Curated by ChEMBL | Assay Description Inhibition of Escherichia coli BL21(DE3) Seryl-tRNA synthetase assessed as reduction in tRNA aminoacylation preincubated for 10 mins with Escherichia... | Eur J Med Chem 148: 384-396 (2018) Article DOI: 10.1016/j.ejmech.2018.02.013 BindingDB Entry DOI: 10.7270/Q2057JJS | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
Leucine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50458122![]() (CHEMBL4204314) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem | Article PubMed | 0.654 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
KU Leuven Curated by ChEMBL | Assay Description Inhibition of Escherichia coli BL21(DE3) Leucyl-tRNA synthetase assessed as reduction in tRNA aminoacylation preincubated for 10 mins with Escherichi... | Eur J Med Chem 148: 384-396 (2018) Article DOI: 10.1016/j.ejmech.2018.02.013 BindingDB Entry DOI: 10.7270/Q2057JJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoleucine--tRNA ligase (Escherichia coli) | BDBM50524451![]() (CHEMBL4553017) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 1.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
KU Leuven Curated by ChEMBL | Assay Description Inhibition of recombinant Escherichia coli BL21(DE3) isoleucyl-tRNA synthetase expressed in Escherichia coli Rosetta 2 (DE3) assessed as reduction in... | Eur J Med Chem 174: 252-264 (2019) Article DOI: 10.1016/j.ejmech.2019.04.045 BindingDB Entry DOI: 10.7270/Q26M3B73 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoleucine--tRNA ligase (Escherichia coli) | BDBM50222902![]() (CHEMBL1163069) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | 1.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
KU Leuven Curated by ChEMBL | Assay Description Inhibition of Escherichia coli BL21(DE3) Isoleucyl-tRNA synthetase assessed as reduction in tRNA aminoacylation preincubated for 10 mins with Escheri... | Eur J Med Chem 148: 384-396 (2018) Article DOI: 10.1016/j.ejmech.2018.02.013 BindingDB Entry DOI: 10.7270/Q2057JJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Leucine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50569962![]() (CHEMBL4864835) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem | Article PubMed | 2.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of recombinant Escherichia coli LeuRS assessed as inhibition of 14C-radiolabelled leucine transfer to tRNA leucine preincubated for 10 min... | Citation and Details Article DOI: 10.1016/j.ejmech.2020.113021 BindingDB Entry DOI: 10.7270/Q2MC93SZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tyrosine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50458121![]() (CHEMBL1163085) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem | PDB Article PubMed | 2.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
KU Leuven Curated by ChEMBL | Assay Description Inhibition of Escherichia coli BL21(DE3) Tyrosyl-tRNA synthetase assessed as reduction in tRNA aminoacylation preincubated for 10 mins with Escherich... | Eur J Med Chem 148: 384-396 (2018) Article DOI: 10.1016/j.ejmech.2018.02.013 BindingDB Entry DOI: 10.7270/Q2057JJS | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
Leucine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50569952![]() (CHEMBL4869028) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem | Article PubMed | 5.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of recombinant Escherichia coli LeuRS assessed as inhibition of 14C-radiolabelled leucine transfer to tRNA leucine preincubated for 10 min... | Citation and Details Article DOI: 10.1016/j.ejmech.2020.113021 BindingDB Entry DOI: 10.7270/Q2MC93SZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Leucine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50524359![]() (CHEMBL4465674) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem | Article PubMed | 9.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
KU Leuven Curated by ChEMBL | Assay Description Inhibition of purified Escherichia coli BL21 (DE3) leuRS incubated for 10 mins in presence of 14C-labeled leucine by radiolabel transfer assay | Eur J Med Chem 173: 154-166 (2019) Article DOI: 10.1016/j.ejmech.2019.04.003 BindingDB Entry DOI: 10.7270/Q27M0CCG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoleucine--tRNA ligase (Escherichia coli) | BDBM50524360![]() (CHEMBL3265242) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 17 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
KU Leuven Curated by ChEMBL | Assay Description Inhibition of purified Escherichia coli BL21 (DE3) ileRS incubated for 10 mins in presence of 14C-labeled isoleucine by radiolabel transfer assay | Eur J Med Chem 173: 154-166 (2019) Article DOI: 10.1016/j.ejmech.2019.04.003 BindingDB Entry DOI: 10.7270/Q27M0CCG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Leucine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50569957![]() (CHEMBL4864965) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem | Article PubMed | 18 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of recombinant Escherichia coli LeuRS assessed as inhibition of 14C-radiolabelled leucine transfer to tRNA leucine preincubated for 10 min... | Citation and Details Article DOI: 10.1016/j.ejmech.2020.113021 BindingDB Entry DOI: 10.7270/Q2MC93SZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Leucine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50524355![]() (CHEMBL4467328) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem | Article PubMed | 21 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
KU Leuven Curated by ChEMBL | Assay Description Inhibition of purified Escherichia coli BL21 (DE3) leuRS incubated for 10 mins in presence of 14C-labeled leucine by radiolabel transfer assay | Eur J Med Chem 173: 154-166 (2019) Article DOI: 10.1016/j.ejmech.2019.04.003 BindingDB Entry DOI: 10.7270/Q27M0CCG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aspartate--tRNA ligase (Escherichia coli) | BDBM50458117![]() (CHEMBL4203761) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 25 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
KU Leuven Curated by ChEMBL | Assay Description Inhibition of Escherichia coli BL21(DE3) Aspartyl-tRNA synthetase assessed as reduction in tRNA aminoacylation preincubated for 10 mins with Escheric... | Eur J Med Chem 148: 384-396 (2018) Article DOI: 10.1016/j.ejmech.2018.02.013 BindingDB Entry DOI: 10.7270/Q2057JJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tyrosine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50458118![]() (CHEMBL4208126) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
KU Leuven Curated by ChEMBL | Assay Description Inhibition of Escherichia coli BL21(DE3) Tyrosyl-tRNA synthetase assessed as reduction in tRNA aminoacylation preincubated for 10 mins with Escherich... | Eur J Med Chem 148: 384-396 (2018) Article DOI: 10.1016/j.ejmech.2018.02.013 BindingDB Entry DOI: 10.7270/Q2057JJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Leucine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50524361![]() (CHEMBL4451258) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem | Article PubMed | 30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
KU Leuven Curated by ChEMBL | Assay Description Inhibition of purified Escherichia coli BL21 (DE3) leuRS incubated for 10 mins in presence of 14C-labeled leucine by radiolabel transfer assay | Eur J Med Chem 173: 154-166 (2019) Article DOI: 10.1016/j.ejmech.2019.04.003 BindingDB Entry DOI: 10.7270/Q27M0CCG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Leucine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50569963![]() (CHEMBL4855635) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem | Article PubMed | 31 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of recombinant Escherichia coli LeuRS assessed as inhibition of 14C-radiolabelled leucine transfer to tRNA leucine preincubated for 10 min... | Citation and Details Article DOI: 10.1016/j.ejmech.2020.113021 BindingDB Entry DOI: 10.7270/Q2MC93SZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Leucine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50569960![]() (CHEMBL4852287) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem | Article PubMed | 31 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of recombinant Escherichia coli LeuRS assessed as inhibition of 14C-radiolabelled leucine transfer to tRNA leucine preincubated for 10 min... | Citation and Details Article DOI: 10.1016/j.ejmech.2020.113021 BindingDB Entry DOI: 10.7270/Q2MC93SZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Leucine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50569958![]() (CHEMBL4864716) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem | Article PubMed | 32 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of recombinant Escherichia coli LeuRS assessed as inhibition of 14C-radiolabelled leucine transfer to tRNA leucine preincubated for 10 min... | Citation and Details Article DOI: 10.1016/j.ejmech.2020.113021 BindingDB Entry DOI: 10.7270/Q2MC93SZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tyrosine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50524357![]() (CHEMBL4558119) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem | PDB Article PubMed | 43 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
KU Leuven Curated by ChEMBL | Assay Description Inhibition of purified Escherichia coli BL21 (DE3) tyrRS incubated for 10 mins in presence of 14C-labeled tyrosine by radiolabel transfer assay | Eur J Med Chem 173: 154-166 (2019) Article DOI: 10.1016/j.ejmech.2019.04.003 BindingDB Entry DOI: 10.7270/Q27M0CCG | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
Leucine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50569954![]() (CHEMBL4867227) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem | Article PubMed | 52 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of recombinant Escherichia coli LeuRS assessed as inhibition of 14C-radiolabelled leucine transfer to tRNA leucine preincubated for 10 min... | Citation and Details Article DOI: 10.1016/j.ejmech.2020.113021 BindingDB Entry DOI: 10.7270/Q2MC93SZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoleucine--tRNA ligase (Escherichia coli) | BDBM50524354![]() (CHEMBL3265243) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 55 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
KU Leuven Curated by ChEMBL | Assay Description Inhibition of purified Escherichia coli BL21 (DE3) ileRS incubated for 10 mins in presence of 14C-labeled isoleucine by radiolabel transfer assay | Eur J Med Chem 173: 154-166 (2019) Article DOI: 10.1016/j.ejmech.2019.04.003 BindingDB Entry DOI: 10.7270/Q27M0CCG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoleucine--tRNA ligase (Escherichia coli) | BDBM50544145![]() (CHEMBL4636583) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 88 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
KU Leuven Curated by ChEMBL | Assay Description Inhibition of Escherichia coli BL21(DE3) ileRS overexpressed in Escherichia coli Rosetta2(DE3) assessed as reduction in tRNA aminoacylation preincuba... | Bioorg Med Chem 28: (2020) Article DOI: 10.1016/j.bmc.2020.115580 BindingDB Entry DOI: 10.7270/Q2XK8K4Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Leucine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50569955![]() (CHEMBL4876966) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem | Article PubMed | 108 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of recombinant Escherichia coli LeuRS assessed as inhibition of 14C-radiolabelled leucine transfer to tRNA leucine preincubated for 10 min... | Citation and Details Article DOI: 10.1016/j.ejmech.2020.113021 BindingDB Entry DOI: 10.7270/Q2MC93SZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoleucine--tRNA ligase (Escherichia coli) | BDBM50544146![]() (CHEMBL4648043) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 114 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
KU Leuven Curated by ChEMBL | Assay Description Inhibition of Escherichia coli BL21(DE3) ileRS overexpressed in Escherichia coli Rosetta2(DE3) assessed as reduction in tRNA aminoacylation preincuba... | Bioorg Med Chem 28: (2020) Article DOI: 10.1016/j.bmc.2020.115580 BindingDB Entry DOI: 10.7270/Q2XK8K4Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tyrosine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50524353![]() (CHEMBL4518549) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem | PDB Article PubMed | 149 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
KU Leuven Curated by ChEMBL | Assay Description Inhibition of purified Escherichia coli BL21 (DE3) tyrRS incubated for 10 mins in presence of 14C-labeled tyrosine by radiolabel transfer assay | Eur J Med Chem 173: 154-166 (2019) Article DOI: 10.1016/j.ejmech.2019.04.003 BindingDB Entry DOI: 10.7270/Q27M0CCG | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
Leucine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50569961![]() (CHEMBL4861722) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem | Article PubMed | 182 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of recombinant Escherichia coli LeuRS assessed as inhibition of 14C-radiolabelled leucine transfer to tRNA leucine preincubated for 10 min... | Citation and Details Article DOI: 10.1016/j.ejmech.2020.113021 BindingDB Entry DOI: 10.7270/Q2MC93SZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoleucine--tRNA ligase (Escherichia coli) | BDBM50458120![]() (CHEMBL4215986) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 213 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
KU Leuven Curated by ChEMBL | Assay Description Inhibition of Escherichia coli BL21(DE3) Isoleucyl-tRNA synthetase assessed as reduction in tRNA aminoacylation preincubated for 10 mins with Escheri... | Eur J Med Chem 148: 384-396 (2018) Article DOI: 10.1016/j.ejmech.2018.02.013 BindingDB Entry DOI: 10.7270/Q2057JJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Leucine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50569956![]() (CHEMBL4850408) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem | Article PubMed | 388 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of recombinant Escherichia coli LeuRS assessed as inhibition of 14C-radiolabelled leucine transfer to tRNA leucine preincubated for 10 min... | Citation and Details Article DOI: 10.1016/j.ejmech.2020.113021 BindingDB Entry DOI: 10.7270/Q2MC93SZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50458116![]() (CHEMBL4208640) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 523 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
KU Leuven Curated by ChEMBL | Assay Description Inhibition of Escherichia coli BL21(DE3) Seryl-tRNA synthetase assessed as reduction in tRNA aminoacylation preincubated for 10 mins with Escherichia... | Eur J Med Chem 148: 384-396 (2018) Article DOI: 10.1016/j.ejmech.2018.02.013 BindingDB Entry DOI: 10.7270/Q2057JJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoleucine--tRNA ligase (Escherichia coli) | BDBM50524358![]() (CHEMBL4475568) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 1.04E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
KU Leuven Curated by ChEMBL | Assay Description Inhibition of purified Escherichia coli BL21 (DE3) ileRS incubated for 10 mins in presence of 14C-labeled isoleucine by radiolabel transfer assay | Eur J Med Chem 173: 154-166 (2019) Article DOI: 10.1016/j.ejmech.2019.04.003 BindingDB Entry DOI: 10.7270/Q27M0CCG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Leucine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50569959![]() (CHEMBL4871282) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem | Article PubMed | 1.26E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of recombinant Escherichia coli LeuRS assessed as inhibition of 14C-radiolabelled leucine transfer to tRNA leucine preincubated for 10 min... | Citation and Details Article DOI: 10.1016/j.ejmech.2020.113021 BindingDB Entry DOI: 10.7270/Q2MC93SZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tyrosine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50524356![]() (CHEMBL4460886) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem | PDB Article PubMed | 1.48E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
KU Leuven Curated by ChEMBL | Assay Description Inhibition of purified Escherichia coli BL21 (DE3) tyrRS incubated for 10 mins in presence of 14C-labeled tyrosine by radiolabel transfer assay | Eur J Med Chem 173: 154-166 (2019) Article DOI: 10.1016/j.ejmech.2019.04.003 BindingDB Entry DOI: 10.7270/Q27M0CCG | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
Leucine--tRNA ligase (Escherichia coli (strain K12)) | BDBM50569953![]() (CHEMBL4871079) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem | Article PubMed | 2.97E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of recombinant Escherichia coli LeuRS assessed as inhibition of 14C-radiolabelled leucine transfer to tRNA leucine preincubated for 10 min... | Citation and Details Article DOI: 10.1016/j.ejmech.2020.113021 BindingDB Entry DOI: 10.7270/Q2MC93SZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoleucine--tRNA ligase (Escherichia coli) | BDBM50524451![]() (CHEMBL4553017) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.80 | n/a | n/a | n/a | n/a | n/a | n/a |
KU Leuven Curated by ChEMBL | Assay Description Inhibition of recombinant Escherichia coli BL21(DE3) isoleucyl-tRNA synthetase expressed in Escherichia coli Rosetta 2 (DE3) assessed as reduction in... | Eur J Med Chem 174: 252-264 (2019) Article DOI: 10.1016/j.ejmech.2019.04.045 BindingDB Entry DOI: 10.7270/Q26M3B73 | |||||||||||
More data for this Ligand-Target Pair |