Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM50466993 (CHEMBL4289691) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORbeta LBD (71 to 459 residues) expressed in Escherichia coli BL21(DE3) after 1... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM50466987 (CHEMBL4292343) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 15 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORbeta LBD (71 to 459 residues) expressed in Escherichia coli BL21(DE3) after 1... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM50466992 (CHEMBL4289114) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 26 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORbeta LBD (71 to 459 residues) expressed in Escherichia coli BL21(DE3) after 1... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM50467002 (CHEMBL4284016) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 34 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORbeta LBD (71 to 459 residues) expressed in Escherichia coli BL21(DE3) after 1... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM50466991 (CHEMBL4276720) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORbeta LBD (71 to 459 residues) expressed in Escherichia coli BL21(DE3) after 1... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM50466998 (CHEMBL4291888) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 76 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORbeta LBD (71 to 459 residues) expressed in Escherichia coli BL21(DE3) after 1... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM50466997 (CHEMBL4284644) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 87 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORbeta LBD (71 to 459 residues) expressed in Escherichia coli BL21(DE3) after 1... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM50467011 (CHEMBL4293341) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 90 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORbeta LBD (71 to 459 residues) expressed in Escherichia coli BL21(DE3) after 1... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM50467006 (CHEMBL4286904) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 90 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORbeta LBD (71 to 459 residues) expressed in Escherichia coli BL21(DE3) after 1... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM50467004 (CHEMBL4288028) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 94 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORbeta LBD (71 to 459 residues) expressed in Escherichia coli BL21(DE3) after 1... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM50466990 (CHEMBL4281271) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 130 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORbeta LBD (71 to 459 residues) expressed in Escherichia coli BL21(DE3) after 1... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM50467007 (CHEMBL4284441) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 180 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORbeta LBD (71 to 459 residues) expressed in Escherichia coli BL21(DE3) after 1... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM50467003 (CHEMBL4290788) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 180 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORbeta LBD (71 to 459 residues) expressed in Escherichia coli BL21(DE3) after 1... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM50466986 (CHEMBL4276733) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORbeta LBD (71 to 459 residues) expressed in Escherichia coli BL21(DE3) after 1... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM50466989 (CHEMBL4288937) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 220 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORbeta LBD (71 to 459 residues) expressed in Escherichia coli BL21(DE3) after 1... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM50467010 (CHEMBL4285419) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 230 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORbeta LBD (71 to 459 residues) expressed in Escherichia coli BL21(DE3) after 1... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM50467008 (CHEMBL4281036) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 230 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORbeta LBD (71 to 459 residues) expressed in Escherichia coli BL21(DE3) after 1... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM50466996 (CHEMBL4292696) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 240 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORbeta LBD (71 to 459 residues) expressed in Escherichia coli BL21(DE3) after 1... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50467006 (CHEMBL4286904) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 330 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORgamma LBD (265 to 518 residues) expressed in Escherichia coli BL21(DE3) after... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM50467009 (CHEMBL4284673) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 330 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORbeta LBD (71 to 459 residues) expressed in Escherichia coli BL21(DE3) after 1... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM50467005 (CHEMBL4277389) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 360 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORbeta LBD (71 to 459 residues) expressed in Escherichia coli BL21(DE3) after 1... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM50467001 (CHEMBL4285780) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 380 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORbeta LBD (71 to 459 residues) expressed in Escherichia coli BL21(DE3) after 1... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50466987 (CHEMBL4292343) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 460 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORgamma LBD (265 to 518 residues) expressed in Escherichia coli BL21(DE3) after... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM50466985 (CHEMBL4293998) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 470 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORbeta LBD (71 to 459 residues) expressed in Escherichia coli BL21(DE3) after 1... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM50466994 (CHEMBL4283486) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 570 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORbeta LBD (71 to 459 residues) expressed in Escherichia coli BL21(DE3) after 1... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM50460723 (CHEMBL4229273) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 610 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORbeta LBD (71 to 459 residues) expressed in Escherichia coli BL21(DE3) after 1... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50467007 (CHEMBL4284441) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 780 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORgamma LBD (265 to 518 residues) expressed in Escherichia coli BL21(DE3) after... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50466989 (CHEMBL4288937) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 790 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORgamma LBD (265 to 518 residues) expressed in Escherichia coli BL21(DE3) after... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM50466995 (CHEMBL4285720) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 800 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORbeta LBD (71 to 459 residues) expressed in Escherichia coli BL21(DE3) after 1... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM50466988 (CHEMBL4292527) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 980 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORbeta LBD (71 to 459 residues) expressed in Escherichia coli BL21(DE3) after 1... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50466986 (CHEMBL4276733) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORgamma LBD (265 to 518 residues) expressed in Escherichia coli BL21(DE3) after... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM50466999 (CHEMBL4294059) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORbeta LBD (71 to 459 residues) expressed in Escherichia coli BL21(DE3) after 1... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM50466998 (CHEMBL4291888) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Inverse agonist activity at GAL4-DNA binding domain-fused human RORbeta ligand binding domain expressed in HEK293T cells incubated for 20 hrs by luci... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM50467000 (CHEMBL4287249) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORbeta LBD (71 to 459 residues) expressed in Escherichia coli BL21(DE3) after 1... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50467003 (CHEMBL4290788) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORgamma LBD (265 to 518 residues) expressed in Escherichia coli BL21(DE3) after... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50466990 (CHEMBL4281271) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORgamma LBD (265 to 518 residues) expressed in Escherichia coli BL21(DE3) after... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50466993 (CHEMBL4289691) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORgamma LBD (265 to 518 residues) expressed in Escherichia coli BL21(DE3) after... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM50466993 (CHEMBL4289691) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Inverse agonist activity at GAL4-DNA binding domain-fused human RORbeta ligand binding domain expressed in HEK293T cells incubated for 20 hrs by luci... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM50466990 (CHEMBL4281271) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Inverse agonist activity at GAL4-DNA binding domain-fused human RORbeta ligand binding domain expressed in HEK293T cells incubated for 20 hrs by luci... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50467011 (CHEMBL4293341) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORgamma LBD (265 to 518 residues) expressed in Escherichia coli BL21(DE3) after... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50466998 (CHEMBL4291888) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORgamma LBD (265 to 518 residues) expressed in Escherichia coli BL21(DE3) after... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50467009 (CHEMBL4284673) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORgamma LBD (265 to 518 residues) expressed in Escherichia coli BL21(DE3) after... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50466992 (CHEMBL4289114) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORgamma LBD (265 to 518 residues) expressed in Escherichia coli BL21(DE3) after... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50467002 (CHEMBL4284016) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORgamma LBD (265 to 518 residues) expressed in Escherichia coli BL21(DE3) after... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50467008 (CHEMBL4281036) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.07E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORgamma LBD (265 to 518 residues) expressed in Escherichia coli BL21(DE3) after... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50466997 (CHEMBL4284644) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORgamma LBD (265 to 518 residues) expressed in Escherichia coli BL21(DE3) after... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50467010 (CHEMBL4285419) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORgamma LBD (265 to 518 residues) expressed in Escherichia coli BL21(DE3) after... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50460723 (CHEMBL4229273) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >4.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORgamma LBD (265 to 518 residues) expressed in Escherichia coli BL21(DE3) after... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50466991 (CHEMBL4276720) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >4.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORgamma LBD (265 to 518 residues) expressed in Escherichia coli BL21(DE3) after... | Bioorg Med Chem Lett 28: 3210-3215 (2018) Article DOI: 10.1016/j.bmcl.2018.08.017 BindingDB Entry DOI: 10.7270/Q2KW5JPB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen-related receptor gamma (Homo sapiens (Human)) | BDBM50455402 (CHEMBL4204689) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 700 | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Agonist activity at human N-terminal alphaHis-SUMO-tagged ERRgamma-LBD (229 to 458 residues) expressed in Escherichia coli BL21 gold (DE3) cells asse... | Bioorg Med Chem Lett 28: 1313-1319 (2018) Article DOI: 10.1016/j.bmcl.2018.03.019 BindingDB Entry DOI: 10.7270/Q2RF5XKM | |||||||||||
More data for this Ligand-Target Pair |
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