Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Syntenin-1 (Homo sapiens) | BDBM50557298 (CHEMBL4750927) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c00382 BindingDB Entry DOI: 10.7270/Q2V98CRX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Syntenin-1 (Homo sapiens) | BDBM50557293 (CHEMBL4781637) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | 40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c00382 BindingDB Entry DOI: 10.7270/Q2V98CRX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Syntenin-1 (Homo sapiens) | BDBM50557299 (CHEMBL4799812) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 170 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) by SPR analysis | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c00382 BindingDB Entry DOI: 10.7270/Q2V98CRX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Syntenin-1 (Homo sapiens) | BDBM50557299 (CHEMBL4799812) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 190 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c00382 BindingDB Entry DOI: 10.7270/Q2V98CRX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Syntenin-1 (Homo sapiens) | BDBM50557297 (CHEMBL4747962) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 250 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c00382 BindingDB Entry DOI: 10.7270/Q2V98CRX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Syntenin-1 (Homo sapiens) | BDBM50557296 (CHEMBL4792861) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 250 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c00382 BindingDB Entry DOI: 10.7270/Q2V98CRX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Syntenin-1 (Homo sapiens) | BDBM50557295 (CHEMBL4758599) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | 250 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c00382 BindingDB Entry DOI: 10.7270/Q2V98CRX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Syntenin-1 (Homo sapiens) | BDBM50557294 (CHEMBL4749490) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 250 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c00382 BindingDB Entry DOI: 10.7270/Q2V98CRX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Syntenin-1 (Homo sapiens) | BDBM50557287 (CHEMBL4752622) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c00382 BindingDB Entry DOI: 10.7270/Q2V98CRX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Syntenin-1 (Homo sapiens) | BDBM50557286 (CHEMBL4798461) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c00382 BindingDB Entry DOI: 10.7270/Q2V98CRX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Syntenin-1 (Homo sapiens) | BDBM50557288 (CHEMBL4792781) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c00382 BindingDB Entry DOI: 10.7270/Q2V98CRX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Syntenin-1 (Homo sapiens) | BDBM50557289 (CHEMBL4740875) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 2.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c00382 BindingDB Entry DOI: 10.7270/Q2V98CRX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Syntenin-1 (Homo sapiens) | BDBM50557290 (CHEMBL4798840) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 4.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c00382 BindingDB Entry DOI: 10.7270/Q2V98CRX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Syntenin-1 (Homo sapiens) | BDBM50557291 (CHEMBL4785814) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c00382 BindingDB Entry DOI: 10.7270/Q2V98CRX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Syntenin-1 (Homo sapiens) | BDBM50557292 (CHEMBL4779632) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 1.10E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c00382 BindingDB Entry DOI: 10.7270/Q2V98CRX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Syntenin-1 (Homo sapiens) | BDBM50557285 (CHEMBL4788058) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c00382 BindingDB Entry DOI: 10.7270/Q2V98CRX | |||||||||||
More data for this Ligand-Target Pair |