Found 44 hits with Last Name = 'bach' and Initial = 'hl' Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kJ/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Epidermal growth factor receptor
(Homo sapiens (Human)) | BDBM50007064
(2-Hydroxy-4-[4-(2-nitro-vinyl)-phenoxysulfonyl]-be...)Show SMILES OC(=O)c1ccc(cc1O)[S+]([O-])(=O)Oc1ccc(\C=C\[N+]([O-])=O)cc1 Show InChI InChI=1S/C15H11NO8S/c17-14-9-12(5-6-13(14)15(18)19)25(22,23)24-11-3-1-10(2-4-11)7-8-16(20)21/h1-9H,(H2-,17,18,19,22,23)/b8-7+ | PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet 
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 54 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of the epidermal growth factor receptor expressed in A431 cell line |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Epidermal growth factor receptor
(Homo sapiens (Human)) | BDBM50007083
(3-Hydroxy-4-[4-(2-nitro-vinyl)-phenoxysulfonyl]-be...)Show SMILES OC(=O)c1ccc(c(O)c1)[S+]([O-])(=O)Oc1ccc(\C=C\[N+]([O-])=O)cc1 Show InChI InChI=1S/C15H11NO8S/c17-13-9-11(15(18)19)3-6-14(13)25(22,23)24-12-4-1-10(2-5-12)7-8-16(20)21/h1-9H,(H2-,17,18,19,22,23)/b8-7+ | PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 310 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of the epidermal growth factor receptor expressed in A431 cell line |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Epidermal growth factor receptor
(Homo sapiens (Human)) | BDBM50007072
(4-(2-nitrovinyl)phenyl 4-(methylcarbamoyl)benzenes...)Show SMILES CNC(=O)c1ccc(cc1)[S+]([O-])(=O)Oc1ccc(\C=C\[N+]([O-])=O)cc1 Show InChI InChI=1S/C16H14N2O6S/c1-17-16(19)13-4-8-15(9-5-13)25(22,23)24-14-6-2-12(3-7-14)10-11-18(20)21/h2-11H,1H3,(H-,17,19,22,23)/b11-10+ | PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 400 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of the epidermal growth factor receptor expressed in A431 cell line |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Epidermal growth factor receptor
(Homo sapiens (Human)) | BDBM50229412
(CHEMBL453502)Show SMILES COc1cc(\C=C\[N+]([O-])=O)ccc1OS(=O)(=O)c1ccc(cc1)C(=O)OC[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(N)ncnc12 |r| Show InChI InChI=1S/C26H24N6O11S/c1-40-18-10-14(8-9-32(36)37)2-7-17(18)43-44(38,39)16-5-3-15(4-6-16)26(35)41-11-19-21(33)22(34)25(42-19)31-13-30-20-23(27)28-12-29-24(20)31/h2-10,12-13,19,21-22,25,33-34H,11H2,1H3,(H2,27,28,29)/b9-8+/t19-,21-,22-,25-/m1/s1 | PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 500 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of the epidermal growth factor receptor expressed in A431 cell line |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Epidermal growth factor receptor
(Homo sapiens (Human)) | BDBM50229411
(CHEMBL505705)Show SMILES Nc1ncnc2n(cnc12)[C@@H]1O[C@H](COC(=O)c2ccc(cc2)S(=O)(=O)Oc2ccc(\C=C\[N+]([O-])=O)cc2)[C@@H](O)[C@H]1O |r| Show InChI InChI=1S/C25H22N6O10S/c26-22-19-23(28-12-27-22)30(13-29-19)24-21(33)20(32)18(40-24)11-39-25(34)15-3-7-17(8-4-15)42(37,38)41-16-5-1-14(2-6-16)9-10-31(35)36/h1-10,12-13,18,20-21,24,32-33H,11H2,(H2,26,27,28)/b10-9+/t18-,20-,21-,24-/m1/s1 | PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 600 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of the epidermal growth factor receptor expressed in A431 cell line |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Epidermal growth factor receptor
(Homo sapiens (Human)) | BDBM50007075
(4-(4-(2-nitrovinyl)phenoxysulfonyl)benzoic acid | ...)Show SMILES OC(=O)c1ccc(cc1)[S+]([O-])(=O)Oc1ccc(\C=C\[N+]([O-])=O)cc1 Show InChI InChI=1S/C15H11NO7S/c17-15(18)12-3-7-14(8-4-12)24(21,22)23-13-5-1-11(2-6-13)9-10-16(19)20/h1-10H,(H-,17,18,21,22)/b10-9+ | PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of the epidermal growth factor receptor expressed in A431 cell line |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Epidermal growth factor receptor
(Homo sapiens (Human)) | BDBM50007073
(4-tert-Butylcarbamoyl-benzenesulfonic acid 4-(2-ni...)Show SMILES CC(C)(C)NC(=O)c1ccc(cc1)S(=O)(=O)Oc1ccc(\C=C\[N+]([O-])=O)cc1 Show InChI InChI=1S/C19H20N2O6S/c1-19(2,3)20-18(22)15-6-10-17(11-7-15)28(25,26)27-16-8-4-14(5-9-16)12-13-21(23)24/h4-13H,1-3H3,(H,20,22)/b13-12+ | PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 1.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of the epidermal growth factor receptor expressed in A431 cell line |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Epidermal growth factor receptor
(Homo sapiens (Human)) | BDBM50007076
(4-(2-nitrovinyl)phenyl 4-(2-(tert-butoxycarbonylam...)Show SMILES CC(C)(C)OC(=O)NCCNC(=O)c1ccc(cc1)[S+]([O-])(=O)Oc1ccc(C=C[N+]([O-])=O)cc1 |w:27.27| Show InChI InChI=1S/C22H25N3O8S/c1-22(2,3)32-21(27)24-14-13-23-20(26)17-6-10-19(11-7-17)34(30,31)33-18-8-4-16(5-9-18)12-15-25(28)29/h4-12,15H,13-14H2,1-3H3,(H2-,23,24,26,27,30,31) | PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 1.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of the epidermal growth factor receptor expressed in A431 cell line |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Epidermal growth factor receptor
(Homo sapiens (Human)) | BDBM50007081
(4-[4-(2-Nitro-vinyl)-phenoxysulfonyl]-benzoic acid...)Show SMILES COC(=O)c1ccc(cc1)[S+]([O-])(=O)Oc1ccc(\C=C\[N+]([O-])=O)cc1 Show InChI InChI=1S/C16H13NO7S/c1-23-16(18)13-4-8-15(9-5-13)25(21,22)24-14-6-2-12(3-7-14)10-11-17(19)20/h2-11H,1H3/b11-10+ | PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of the epidermal growth factor receptor expressed in A431 cell line |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Epidermal growth factor receptor
(Homo sapiens (Human)) | BDBM50007070
(2-Hydroxy-4-[4-(2-nitro-vinyl)-phenoxysulfonyl]-be...)Show SMILES COC(=O)c1ccc(cc1O)[S+]([O-])(=O)Oc1ccc(\C=C\[N+]([O-])=O)cc1 Show InChI InChI=1S/C16H13NO8S/c1-24-16(19)14-7-6-13(10-15(14)18)26(22,23)25-12-4-2-11(3-5-12)8-9-17(20)21/h2-10H,1H3,(H-,18,19,22,23)/b9-8+ | PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 1.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of the epidermal growth factor receptor expressed in A431 cell line |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Epidermal growth factor receptor
(Homo sapiens (Human)) | BDBM50007087
(4-(2-methoxy-4-(2-nitroprop-1-enyl)phenoxysulfonyl...)Show SMILES COc1cc(\C=C(/C)[N+]([O-])=O)ccc1O[S+]([O-])(=O)c1ccc(cc1)C(O)=O Show InChI InChI=1S/C17H15NO8S/c1-11(18(21)22)9-12-3-8-15(16(10-12)25-2)26-27(23,24)14-6-4-13(5-7-14)17(19)20/h3-10H,1-2H3,(H-,19,20,23,24)/b11-9+ | PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 2.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of the epidermal growth factor receptor expressed in A431 cell line |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Epidermal growth factor receptor
(Homo sapiens (Human)) | BDBM50007077
(4-(2-methoxy-4-(2-nitrovinyl)phenoxysulfonyl)benzo...)Show SMILES COc1cc(\C=C\[N+]([O-])=O)ccc1O[S+]([O-])(=O)c1ccc(cc1)C(O)=O Show InChI InChI=1S/C16H13NO8S/c1-24-15-10-11(8-9-17(20)21)2-7-14(15)25-26(22,23)13-5-3-12(4-6-13)16(18)19/h2-10H,1H3,(H-,18,19,22,23)/b9-8+ | PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 2.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of the epidermal growth factor receptor expressed in A431 cell line |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Epidermal growth factor receptor
(Homo sapiens (Human)) | BDBM50007084
(2-methoxy-4-(2-nitroprop-1-enyl)phenyl 4-(methylca...)Show SMILES CNC(=O)c1ccc(cc1)[S+]([O-])(=O)Oc1ccc(\C=C(/C)[N+]([O-])=O)cc1OC Show InChI InChI=1S/C18H18N2O7S/c1-12(20(22)23)10-13-4-9-16(17(11-13)26-3)27-28(24,25)15-7-5-14(6-8-15)18(21)19-2/h4-11H,1-3H3,(H-,19,21,24,25)/b12-10+ | PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 4.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of the epidermal growth factor receptor expressed in A431 cell line |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Epidermal growth factor receptor
(Homo sapiens (Human)) | BDBM50007074
(4-(2-nitrovinyl)phenyl 4-(butylcarbamoyl)benzenesu...)Show SMILES CCCCNC(=O)c1ccc(cc1)[S+]([O-])(=O)Oc1ccc(\C=C\[N+]([O-])=O)cc1 Show InChI InChI=1S/C19H20N2O6S/c1-2-3-13-20-19(22)16-6-10-18(11-7-16)28(25,26)27-17-8-4-15(5-9-17)12-14-21(23)24/h4-12,14H,2-3,13H2,1H3,(H-,20,22,25,26)/b14-12+ | PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 4.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of the epidermal growth factor receptor expressed in A431 cell line |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase ABL1/ABL2
(Homo sapiens (Human)) | BDBM50007080
(4-(2-Amino-ethylcarbamoyl)-benzenesulfonic acid 4-...)Show SMILES NCCNC(=O)c1ccc(cc1)S(=O)(=O)Oc1ccc(\C=C\[N+]([O-])=O)cc1 Show InChI InChI=1S/C17H17N3O6S/c18-10-11-19-17(21)14-3-7-16(8-4-14)27(24,25)26-15-5-1-13(2-6-15)9-12-20(22)23/h1-9,12H,10-11,18H2,(H,19,21)/b12-9+ | PDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of recombinant v-Abl tyrosine kinase. |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Epidermal growth factor receptor
(Homo sapiens (Human)) | BDBM50007080
(4-(2-Amino-ethylcarbamoyl)-benzenesulfonic acid 4-...)Show SMILES NCCNC(=O)c1ccc(cc1)S(=O)(=O)Oc1ccc(\C=C\[N+]([O-])=O)cc1 Show InChI InChI=1S/C17H17N3O6S/c18-10-11-19-17(21)14-3-7-16(8-4-14)27(24,25)26-15-5-1-13(2-6-15)9-12-20(22)23/h1-9,12H,10-11,18H2,(H,19,21)/b12-9+ | PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 5.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of the epidermal growth factor receptor expressed in A431 cell line |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Epidermal growth factor receptor
(Homo sapiens (Human)) | BDBM50007067
(2-[1-(4-{4-[2-nitro-(E)-1-ethenyl]phenyloxysulfony...)Show SMILES C[C@@H](NC(=O)[C@@H](C)NC(=O)c1ccc(cc1)S(=O)(=O)Oc1ccc(\C=C\[N+]([O-])=O)cc1)C(O)=O Show InChI InChI=1S/C21H21N3O9S/c1-13(19(25)23-14(2)21(27)28)22-20(26)16-5-9-18(10-6-16)34(31,32)33-17-7-3-15(4-8-17)11-12-24(29)30/h3-14H,1-2H3,(H,22,26)(H,23,25)(H,27,28)/b12-11+/t13-,14-/m1/s1 | PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
KEGG
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 7.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of the epidermal growth factor receptor expressed in A431 cell line |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Epidermal growth factor receptor
(Homo sapiens (Human)) | BDBM50007082
((E)-2-methoxy-4-(2-nitrovinyl)phenol | 2-Methoxy-4...)Show InChI InChI=1S/C9H9NO4/c1-14-9-6-7(2-3-8(9)11)4-5-10(12)13/h2-6,11H,1H3/b5-4+ | PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| Purchase
CHEMBL
MCE
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 7.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of the epidermal growth factor receptor expressed in A431 cell line |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Epidermal growth factor receptor
(Homo sapiens (Human)) | BDBM50007069
(4-(2-Nitro-vinyl)-benzene-1,2-diol | 4-(2-nitrovin...)Show InChI InChI=1S/C8H7NO4/c10-7-2-1-6(5-8(7)11)3-4-9(12)13/h1-5,10-11H/b4-3+ | PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Patents
Similars
| PubMed
| n/a | n/a | 8.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of the epidermal growth factor receptor expressed in A431 cell line |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Epidermal growth factor receptor
(Homo sapiens (Human)) | BDBM50007078
(4-(2-Nitro-propenyl)-benzene-1,2-diol | 4-(2-nitro...)Show InChI InChI=1S/C9H9NO4/c1-6(10(13)14)4-7-2-3-8(11)9(12)5-7/h2-5,11-12H,1H3/b6-4+ | PDB
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| n/a | n/a | 9.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of the epidermal growth factor receptor expressed in A431 cell line |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Epidermal growth factor receptor
(Homo sapiens (Human)) | BDBM50007085
((E)-4-(2-nitrovinyl)phenol | 4-(2-Nitro-vinyl)-phe...)Show InChI InChI=1S/C8H7NO3/c10-8-3-1-7(2-4-8)5-6-9(11)12/h1-6,10H/b6-5+ | PDB
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| n/a | n/a | 1.01E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of the epidermal growth factor receptor expressed in A431 cell line |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase ABL1/ABL2
(Homo sapiens (Human)) | BDBM50007079
(1-{4-[1-[1-(2-aminoethylcarbamoyl)-(1R)-ethylcarba...)Show SMILES C[C@@H](NC(=O)[C@@H](C)NC(=O)c1ccc(cc1)S(=O)(=O)Oc1ccc(\C=C\[N+]([O-])=O)cc1)C(=O)NCCN Show InChI InChI=1S/C23H27N5O8S/c1-15(21(29)25-13-12-24)26-22(30)16(2)27-23(31)18-5-9-20(10-6-18)37(34,35)36-19-7-3-17(4-8-19)11-14-28(32)33/h3-11,14-16H,12-13,24H2,1-2H3,(H,25,29)(H,26,30)(H,27,31)/b14-11+/t15-,16-/m1/s1 | PDB
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| n/a | n/a | 1.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of recombinant v-Abl tyrosine kinase. |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Epidermal growth factor receptor
(Homo sapiens (Human)) | BDBM50007079
(1-{4-[1-[1-(2-aminoethylcarbamoyl)-(1R)-ethylcarba...)Show SMILES C[C@@H](NC(=O)[C@@H](C)NC(=O)c1ccc(cc1)S(=O)(=O)Oc1ccc(\C=C\[N+]([O-])=O)cc1)C(=O)NCCN Show InChI InChI=1S/C23H27N5O8S/c1-15(21(29)25-13-12-24)26-22(30)16(2)27-23(31)18-5-9-20(10-6-18)37(34,35)36-19-7-3-17(4-8-19)11-14-28(32)33/h3-11,14-16H,12-13,24H2,1-2H3,(H,25,29)(H,26,30)(H,27,31)/b14-11+/t15-,16-/m1/s1 | PDB
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| n/a | n/a | 1.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of the epidermal growth factor receptor expressed in A431 cell line |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase ABL1/ABL2
(Homo sapiens (Human)) | BDBM50007064
(2-Hydroxy-4-[4-(2-nitro-vinyl)-phenoxysulfonyl]-be...)Show SMILES OC(=O)c1ccc(cc1O)[S+]([O-])(=O)Oc1ccc(\C=C\[N+]([O-])=O)cc1 Show InChI InChI=1S/C15H11NO8S/c17-14-9-12(5-6-13(14)15(18)19)25(22,23)24-11-3-1-10(2-4-11)7-8-16(20)21/h1-9H,(H2-,17,18,19,22,23)/b8-7+ | PDB
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| n/a | n/a | 2.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of recombinant v-Abl tyrosine kinase. |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase ABL1/ABL2
(Homo sapiens (Human)) | BDBM50007067
(2-[1-(4-{4-[2-nitro-(E)-1-ethenyl]phenyloxysulfony...)Show SMILES C[C@@H](NC(=O)[C@@H](C)NC(=O)c1ccc(cc1)S(=O)(=O)Oc1ccc(\C=C\[N+]([O-])=O)cc1)C(O)=O Show InChI InChI=1S/C21H21N3O9S/c1-13(19(25)23-14(2)21(27)28)22-20(26)16-5-9-18(10-6-16)34(31,32)33-17-7-3-15(4-8-17)11-12-24(29)30/h3-14H,1-2H3,(H,22,26)(H,23,25)(H,27,28)/b12-11+/t13-,14-/m1/s1 | PDB
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| n/a | n/a | 3.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of recombinant v-Abl tyrosine kinase. |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase ABL1/ABL2
(Homo sapiens (Human)) | BDBM50007072
(4-(2-nitrovinyl)phenyl 4-(methylcarbamoyl)benzenes...)Show SMILES CNC(=O)c1ccc(cc1)[S+]([O-])(=O)Oc1ccc(\C=C\[N+]([O-])=O)cc1 Show InChI InChI=1S/C16H14N2O6S/c1-17-16(19)13-4-8-15(9-5-13)25(22,23)24-14-6-2-12(3-7-14)10-11-18(20)21/h2-11H,1H3,(H-,17,19,22,23)/b11-10+ | PDB
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| n/a | n/a | 3.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of recombinant v-Abl tyrosine kinase. |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase ABL1/ABL2
(Homo sapiens (Human)) | BDBM50007077
(4-(2-methoxy-4-(2-nitrovinyl)phenoxysulfonyl)benzo...)Show SMILES COc1cc(\C=C\[N+]([O-])=O)ccc1O[S+]([O-])(=O)c1ccc(cc1)C(O)=O Show InChI InChI=1S/C16H13NO8S/c1-24-15-10-11(8-9-17(20)21)2-7-14(15)25-26(22,23)13-5-3-12(4-6-13)16(18)19/h2-10H,1H3,(H-,18,19,22,23)/b9-8+ | PDB
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| n/a | n/a | 4.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of recombinant v-Abl tyrosine kinase. |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Epidermal growth factor receptor
(Homo sapiens (Human)) | BDBM50007071
(CHEMBL312451 | tert-butyl 2-[1-(4-{4-[2-nitro-(E)-...)Show SMILES C[C@@H](NC(=O)c1ccc(cc1)S(=O)(=O)Oc1ccc(\C=C\[N+]([O-])=O)cc1)C(=O)N[C@H](C)C(=O)OC(C)(C)C Show InChI InChI=1S/C25H29N3O9S/c1-16(22(29)27-17(2)24(31)36-25(3,4)5)26-23(30)19-8-12-21(13-9-19)38(34,35)37-20-10-6-18(7-11-20)14-15-28(32)33/h6-17H,1-5H3,(H,26,30)(H,27,29)/b15-14+/t16-,17-/m1/s1 | PDB
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| n/a | n/a | 4.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of the epidermal growth factor receptor expressed in A431 cell line |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Epidermal growth factor receptor
(Homo sapiens (Human)) | BDBM50007065
(1-(4-{1-[1-(2-carboxy tertbutyl aminoethylcarbamoy...)Show SMILES C[C@@H](NC(=O)[C@@H](C)NC(=O)c1ccc(cc1)S(=O)(=O)Oc1ccc(C=C[N+]([O-])=O)cc1)C(=O)NCCNC(=O)OC(C)(C)C |w:25.26| Show InChI InChI=1S/C28H35N5O10S/c1-18(24(34)29-15-16-30-27(37)42-28(3,4)5)31-25(35)19(2)32-26(36)21-8-12-23(13-9-21)44(40,41)43-22-10-6-20(7-11-22)14-17-33(38)39/h6-14,17-19H,15-16H2,1-5H3,(H,29,34)(H,30,37)(H,31,35)(H,32,36)/t18-,19-/m1/s1 | PDB
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| n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of the epidermal growth factor receptor expressed in A431 cell line |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase ABL1/ABL2
(Homo sapiens (Human)) | BDBM50007075
(4-(4-(2-nitrovinyl)phenoxysulfonyl)benzoic acid | ...)Show SMILES OC(=O)c1ccc(cc1)[S+]([O-])(=O)Oc1ccc(\C=C\[N+]([O-])=O)cc1 Show InChI InChI=1S/C15H11NO7S/c17-15(18)12-3-7-14(8-4-12)24(21,22)23-13-5-1-11(2-6-13)9-10-16(19)20/h1-10H,(H-,17,18,21,22)/b10-9+ | PDB
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| n/a | n/a | 1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of recombinant v-Abl tyrosine kinase. |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase ABL1/ABL2
(Homo sapiens (Human)) | BDBM50007069
(4-(2-Nitro-vinyl)-benzene-1,2-diol | 4-(2-nitrovin...)Show InChI InChI=1S/C8H7NO4/c10-7-2-1-6(5-8(7)11)3-4-9(12)13/h1-5,10-11H/b4-3+ | PDB
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| n/a | n/a | 1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of recombinant v-Abl tyrosine kinase. |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase ABL1/ABL2
(Homo sapiens (Human)) | BDBM50007071
(CHEMBL312451 | tert-butyl 2-[1-(4-{4-[2-nitro-(E)-...)Show SMILES C[C@@H](NC(=O)c1ccc(cc1)S(=O)(=O)Oc1ccc(\C=C\[N+]([O-])=O)cc1)C(=O)N[C@H](C)C(=O)OC(C)(C)C Show InChI InChI=1S/C25H29N3O9S/c1-16(22(29)27-17(2)24(31)36-25(3,4)5)26-23(30)19-8-12-21(13-9-19)38(34,35)37-20-10-6-18(7-11-20)14-15-28(32)33/h6-17H,1-5H3,(H,26,30)(H,27,29)/b15-14+/t16-,17-/m1/s1 | PDB
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| n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of recombinant v-Abl tyrosine kinase. |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase ABL1/ABL2
(Homo sapiens (Human)) | BDBM50229411
(CHEMBL505705)Show SMILES Nc1ncnc2n(cnc12)[C@@H]1O[C@H](COC(=O)c2ccc(cc2)S(=O)(=O)Oc2ccc(\C=C\[N+]([O-])=O)cc2)[C@@H](O)[C@H]1O |r| Show InChI InChI=1S/C25H22N6O10S/c26-22-19-23(28-12-27-22)30(13-29-19)24-21(33)20(32)18(40-24)11-39-25(34)15-3-7-17(8-4-15)42(37,38)41-16-5-1-14(2-6-16)9-10-31(35)36/h1-10,12-13,18,20-21,24,32-33H,11H2,(H2,26,27,28)/b10-9+/t18-,20-,21-,24-/m1/s1 | PDB
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| n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of recombinant v-Abl tyrosine kinase. |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase ABL1/ABL2
(Homo sapiens (Human)) | BDBM50229412
(CHEMBL453502)Show SMILES COc1cc(\C=C\[N+]([O-])=O)ccc1OS(=O)(=O)c1ccc(cc1)C(=O)OC[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(N)ncnc12 |r| Show InChI InChI=1S/C26H24N6O11S/c1-40-18-10-14(8-9-32(36)37)2-7-17(18)43-44(38,39)16-5-3-15(4-6-16)26(35)41-11-19-21(33)22(34)25(42-19)31-13-30-20-23(27)28-12-29-24(20)31/h2-10,12-13,19,21-22,25,33-34H,11H2,1H3,(H2,27,28,29)/b9-8+/t19-,21-,22-,25-/m1/s1 | PDB
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| n/a | n/a | 1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of recombinant v-Abl tyrosine kinase. |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase ABL1/ABL2
(Homo sapiens (Human)) | BDBM50007076
(4-(2-nitrovinyl)phenyl 4-(2-(tert-butoxycarbonylam...)Show SMILES CC(C)(C)OC(=O)NCCNC(=O)c1ccc(cc1)[S+]([O-])(=O)Oc1ccc(C=C[N+]([O-])=O)cc1 |w:27.27| Show InChI InChI=1S/C22H25N3O8S/c1-22(2,3)32-21(27)24-14-13-23-20(26)17-6-10-19(11-7-17)34(30,31)33-18-8-4-16(5-9-18)12-15-25(28)29/h4-12,15H,13-14H2,1-3H3,(H2-,23,24,26,27,30,31) | PDB
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| n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of recombinant v-Abl tyrosine kinase. |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase ABL1/ABL2
(Homo sapiens (Human)) | BDBM50007070
(2-Hydroxy-4-[4-(2-nitro-vinyl)-phenoxysulfonyl]-be...)Show SMILES COC(=O)c1ccc(cc1O)[S+]([O-])(=O)Oc1ccc(\C=C\[N+]([O-])=O)cc1 Show InChI InChI=1S/C16H13NO8S/c1-24-16(19)14-7-6-13(10-15(14)18)26(22,23)25-12-4-2-11(3-5-12)8-9-17(20)21/h2-10H,1H3,(H-,18,19,22,23)/b9-8+ | PDB
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| n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of recombinant v-Abl tyrosine kinase. |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase ABL1/ABL2
(Homo sapiens (Human)) | BDBM50007074
(4-(2-nitrovinyl)phenyl 4-(butylcarbamoyl)benzenesu...)Show SMILES CCCCNC(=O)c1ccc(cc1)[S+]([O-])(=O)Oc1ccc(\C=C\[N+]([O-])=O)cc1 Show InChI InChI=1S/C19H20N2O6S/c1-2-3-13-20-19(22)16-6-10-18(11-7-16)28(25,26)27-17-8-4-15(5-9-17)12-14-21(23)24/h4-12,14H,2-3,13H2,1H3,(H-,20,22,25,26)/b14-12+ | PDB
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| n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of recombinant v-Abl tyrosine kinase. |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Epidermal growth factor receptor
(Homo sapiens (Human)) | BDBM50007066
(4-Butylcarbamoyl-benzenesulfonic acid 4-formyl-phe...)Show SMILES CCCCNC(=O)c1ccc(cc1)S(=O)(=O)Oc1ccc(C=O)cc1 Show InChI InChI=1S/C18H19NO5S/c1-2-3-12-19-18(21)15-6-10-17(11-7-15)25(22,23)24-16-8-4-14(13-20)5-9-16/h4-11,13H,2-3,12H2,1H3,(H,19,21) | PDB
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| n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of the epidermal growth factor receptor expressed in A431 cell line |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase ABL1/ABL2
(Homo sapiens (Human)) | BDBM50007081
(4-[4-(2-Nitro-vinyl)-phenoxysulfonyl]-benzoic acid...)Show SMILES COC(=O)c1ccc(cc1)[S+]([O-])(=O)Oc1ccc(\C=C\[N+]([O-])=O)cc1 Show InChI InChI=1S/C16H13NO7S/c1-23-16(18)13-4-8-15(9-5-13)25(21,22)24-14-6-2-12(3-7-14)10-11-17(19)20/h2-11H,1H3/b11-10+ | PDB
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UniChem
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Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of recombinant v-Abl tyrosine kinase. |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase ABL1/ABL2
(Homo sapiens (Human)) | BDBM50007082
((E)-2-methoxy-4-(2-nitrovinyl)phenol | 2-Methoxy-4...)Show InChI InChI=1S/C9H9NO4/c1-14-9-6-7(2-3-8(9)11)4-5-10(12)13/h2-6,11H,1H3/b5-4+ | PDB
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Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of recombinant v-Abl tyrosine kinase. |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase ABL1/ABL2
(Homo sapiens (Human)) | BDBM50007085
((E)-4-(2-nitrovinyl)phenol | 4-(2-Nitro-vinyl)-phe...)Show InChI InChI=1S/C8H7NO3/c10-8-3-1-7(2-4-8)5-6-9(11)12/h1-6,10H/b6-5+ | PDB
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| n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of recombinant v-Abl tyrosine kinase. |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase ABL1/ABL2
(Homo sapiens (Human)) | BDBM50007083
(3-Hydroxy-4-[4-(2-nitro-vinyl)-phenoxysulfonyl]-be...)Show SMILES OC(=O)c1ccc(c(O)c1)[S+]([O-])(=O)Oc1ccc(\C=C\[N+]([O-])=O)cc1 Show InChI InChI=1S/C15H11NO8S/c17-13-9-11(15(18)19)3-6-14(13)25(22,23)24-12-4-1-10(2-5-12)7-8-16(20)21/h1-9H,(H2-,17,18,19,22,23)/b8-7+ | PDB
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| n/a | n/a | 1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of recombinant v-Abl tyrosine kinase. |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase ABL1/ABL2
(Homo sapiens (Human)) | BDBM50007073
(4-tert-Butylcarbamoyl-benzenesulfonic acid 4-(2-ni...)Show SMILES CC(C)(C)NC(=O)c1ccc(cc1)S(=O)(=O)Oc1ccc(\C=C\[N+]([O-])=O)cc1 Show InChI InChI=1S/C19H20N2O6S/c1-19(2,3)20-18(22)15-6-10-17(11-7-15)28(25,26)27-16-8-4-14(5-9-16)12-13-21(23)24/h4-13H,1-3H3,(H,20,22)/b13-12+ | PDB
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Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of recombinant v-Abl tyrosine kinase. |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase ABL1/ABL2
(Homo sapiens (Human)) | BDBM50007078
(4-(2-Nitro-propenyl)-benzene-1,2-diol | 4-(2-nitro...)Show InChI InChI=1S/C9H9NO4/c1-6(10(13)14)4-7-2-3-8(11)9(12)5-7/h2-5,11-12H,1H3/b6-4+ | PDB
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| n/a | n/a | 1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Ciba-Geigy Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of recombinant v-Abl tyrosine kinase. |
J Med Chem 34: 2328-37 (1991)
BindingDB Entry DOI: 10.7270/Q24F1RB9 |
More data for this
Ligand-Target Pair | |
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