Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Arginase (Leishmania amazonensis) | BDBM50510706 (CHEMBL4515068) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 1.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Tecnologia em Farmacos Curated by ChEMBL | Assay Description Non-competitive inhibition of Leishmania amazonensis arginase using L-arginine as substrate incubated for 15 mins | Bioorg Med Chem 27: 3061-3069 (2019) Article DOI: 10.1016/j.bmc.2019.05.026 BindingDB Entry DOI: 10.7270/Q2SX6HJQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Arginase (Leishmania amazonensis) | BDBM50510709 (CHEMBL4571367) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Tecnologia em Farmacos Curated by ChEMBL | Assay Description Inhibition of recombinant Leishmania amazonensis arginase expressed in Escherichia coli using L-arginine as substrate | Bioorg Med Chem 27: 3061-3069 (2019) Article DOI: 10.1016/j.bmc.2019.05.026 BindingDB Entry DOI: 10.7270/Q2SX6HJQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Arginase (Leishmania amazonensis) | BDBM50510706 (CHEMBL4515068) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.65E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Tecnologia em Farmacos Curated by ChEMBL | Assay Description Non-competitive inhibition of Leishmania amazonensis arginase using L-arginine as substrate incubated for 15 mins | Bioorg Med Chem 27: 3061-3069 (2019) Article DOI: 10.1016/j.bmc.2019.05.026 BindingDB Entry DOI: 10.7270/Q2SX6HJQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Arginase (Leishmania amazonensis) | BDBM50510706 (CHEMBL4515068) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.65E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Tecnologia em Farmacos Curated by ChEMBL | Assay Description Inhibition of recombinant Leishmania amazonensis arginase expressed in Escherichia coli using L-arginine as substrate | Bioorg Med Chem 27: 3061-3069 (2019) Article DOI: 10.1016/j.bmc.2019.05.026 BindingDB Entry DOI: 10.7270/Q2SX6HJQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Arginase (Leishmania amazonensis) | BDBM50510711 (CHEMBL4467463) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Tecnologia em Farmacos Curated by ChEMBL | Assay Description Inhibition of recombinant Leishmania amazonensis arginase expressed in Escherichia coli using L-arginine as substrate | Bioorg Med Chem 27: 3061-3069 (2019) Article DOI: 10.1016/j.bmc.2019.05.026 BindingDB Entry DOI: 10.7270/Q2SX6HJQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Arginase (Leishmania amazonensis) | BDBM50510707 (CHEMBL4541649) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Tecnologia em Farmacos Curated by ChEMBL | Assay Description Inhibition of recombinant Leishmania amazonensis arginase expressed in Escherichia coli using L-arginine as substrate | Bioorg Med Chem 27: 3061-3069 (2019) Article DOI: 10.1016/j.bmc.2019.05.026 BindingDB Entry DOI: 10.7270/Q2SX6HJQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Arginase (Leishmania amazonensis) | BDBM50510708 (CHEMBL4456185) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Tecnologia em Farmacos Curated by ChEMBL | Assay Description Inhibition of recombinant Leishmania amazonensis arginase expressed in Escherichia coli using L-arginine as substrate | Bioorg Med Chem 27: 3061-3069 (2019) Article DOI: 10.1016/j.bmc.2019.05.026 BindingDB Entry DOI: 10.7270/Q2SX6HJQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Arginase (Leishmania amazonensis) | BDBM50510712 (CHEMBL4570250) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Tecnologia em Farmacos Curated by ChEMBL | Assay Description Inhibition of recombinant Leishmania amazonensis arginase expressed in Escherichia coli using L-arginine as substrate | Bioorg Med Chem 27: 3061-3069 (2019) Article DOI: 10.1016/j.bmc.2019.05.026 BindingDB Entry DOI: 10.7270/Q2SX6HJQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Arginase (Leishmania amazonensis) | BDBM50510710 (CHEMBL4438412) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto de Tecnologia em Farmacos Curated by ChEMBL | Assay Description Inhibition of recombinant Leishmania amazonensis arginase expressed in Escherichia coli using L-arginine as substrate | Bioorg Med Chem 27: 3061-3069 (2019) Article DOI: 10.1016/j.bmc.2019.05.026 BindingDB Entry DOI: 10.7270/Q2SX6HJQ | |||||||||||
More data for this Ligand-Target Pair |