Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50295263 ((S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-y...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Roma Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane by liquid scintillation counting | Bioorg Med Chem Lett 19: 4115-8 (2009) Article DOI: 10.1016/j.bmcl.2009.06.008 BindingDB Entry DOI: 10.7270/Q2ZS2WJX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50295264 ((S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-y...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 5.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Roma Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane by liquid scintillation counting | Bioorg Med Chem Lett 19: 4115-8 (2009) Article DOI: 10.1016/j.bmcl.2009.06.008 BindingDB Entry DOI: 10.7270/Q2ZS2WJX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50295262 ((S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-y...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 6.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Roma Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane by liquid scintillation counting | Bioorg Med Chem Lett 19: 4115-8 (2009) Article DOI: 10.1016/j.bmcl.2009.06.008 BindingDB Entry DOI: 10.7270/Q2ZS2WJX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50139013 ((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | 8.23 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
"Sapienza" Università di Roma Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 3 hrs by liquid scintillation counting | Eur J Med Chem 45: 4594-600 (2010) Article DOI: 10.1016/j.ejmech.2010.07.022 BindingDB Entry DOI: 10.7270/Q2KK9C0Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50320022 ((S)-1-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)-N...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 8.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Roma Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cells | J Med Chem 53: 4550-4 (2010) Article DOI: 10.1021/jm1001343 BindingDB Entry DOI: 10.7270/Q23F4PTK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50139013 ((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | 9.56 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Roma Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane by liquid scintillation counting | Bioorg Med Chem Lett 19: 4115-8 (2009) Article DOI: 10.1016/j.bmcl.2009.06.008 BindingDB Entry DOI: 10.7270/Q2ZS2WJX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50139013 ((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | 9.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Roma Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cells | J Med Chem 53: 4550-4 (2010) Article DOI: 10.1021/jm1001343 BindingDB Entry DOI: 10.7270/Q23F4PTK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50095155 ((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | 10.7 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Roma Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane by liquid scintillation counting | Bioorg Med Chem Lett 19: 4115-8 (2009) Article DOI: 10.1016/j.bmcl.2009.06.008 BindingDB Entry DOI: 10.7270/Q2ZS2WJX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50326889 ((S)-N-((S)-1-amino-1-oxo-3-phenylpropan-2-yl)-2-((...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 19 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
"Sapienza" Università di Roma Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 3 hrs by liquid scintillation counting | Eur J Med Chem 45: 4594-600 (2010) Article DOI: 10.1016/j.ejmech.2010.07.022 BindingDB Entry DOI: 10.7270/Q2KK9C0Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50326886 ((R)-1-((S)-2-(2-((R)-1-((S)-2-amino-3-(4-hydroxyph...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
"Sapienza" Università di Roma Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 3 hrs by liquid scintillation counting | Eur J Med Chem 45: 4594-600 (2010) Article DOI: 10.1016/j.ejmech.2010.07.022 BindingDB Entry DOI: 10.7270/Q2KK9C0Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50295261 (CHEMBL549770 | N-((S)-1-((S)-1-amino-1-oxo-3-pheny...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 34 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Roma Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane by liquid scintillation counting | Bioorg Med Chem Lett 19: 4115-8 (2009) Article DOI: 10.1016/j.bmcl.2009.06.008 BindingDB Entry DOI: 10.7270/Q2ZS2WJX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50295265 (CHEMBL540482 | N-((S)-1-((S)-1-amino-1-oxo-3-pheny...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 34 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Roma Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane by liquid scintillation counting | Bioorg Med Chem Lett 19: 4115-8 (2009) Article DOI: 10.1016/j.bmcl.2009.06.008 BindingDB Entry DOI: 10.7270/Q2ZS2WJX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50295265 (CHEMBL540482 | N-((S)-1-((S)-1-amino-1-oxo-3-pheny...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Roma Curated by ChEMBL | Assay Description Displacement of [3H]DPDE from delta opioid receptor in rat brain membrane by liquid scintillation counting | Bioorg Med Chem Lett 19: 4115-8 (2009) Article DOI: 10.1016/j.bmcl.2009.06.008 BindingDB Entry DOI: 10.7270/Q2ZS2WJX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50326885 ((S)-N-((S)-1-amino-1-oxo-3-phenylpropan-2-yl)-2-(2...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 58 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
"Sapienza" Università di Roma Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 3 hrs by liquid scintillation counting | Eur J Med Chem 45: 4594-600 (2010) Article DOI: 10.1016/j.ejmech.2010.07.022 BindingDB Entry DOI: 10.7270/Q2KK9C0Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50326888 ((S)-N-((S)-1-amino-1-oxo-3-phenylpropan-2-yl)-2-((...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 63 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
"Sapienza" Università di Roma Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 3 hrs by liquid scintillation counting | Eur J Med Chem 45: 4594-600 (2010) Article DOI: 10.1016/j.ejmech.2010.07.022 BindingDB Entry DOI: 10.7270/Q2KK9C0Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50326883 ((S)-N-((S)-1-amino-1-oxo-3-phenylpropan-2-yl)-2-((...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
"Sapienza" Università di Roma Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 3 hrs by liquid scintillation counting | Eur J Med Chem 45: 4594-600 (2010) Article DOI: 10.1016/j.ejmech.2010.07.022 BindingDB Entry DOI: 10.7270/Q2KK9C0Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50320023 ((S)-1-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)-N...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 130 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Roma Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cells | J Med Chem 53: 4550-4 (2010) Article DOI: 10.1021/jm1001343 BindingDB Entry DOI: 10.7270/Q23F4PTK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50166066 (CHEMBL362991 | H-Tyr-Pro-Phe-Pro-NH2 | MORPHICEPTI...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | 135 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
"Sapienza" Università di Roma Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 3 hrs by liquid scintillation counting | Eur J Med Chem 45: 4594-600 (2010) Article DOI: 10.1016/j.ejmech.2010.07.022 BindingDB Entry DOI: 10.7270/Q2KK9C0Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50320024 ((S)-N-(3-((S)-1-amino-1-oxo-3-phenylpropan-2-ylami...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 200 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Roma Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cells | J Med Chem 53: 4550-4 (2010) Article DOI: 10.1021/jm1001343 BindingDB Entry DOI: 10.7270/Q23F4PTK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50295260 (CHEMBL564939 | N-((S)-1-((S)-1-amino-1-oxo-3-pheny...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 210 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Roma Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane by liquid scintillation counting | Bioorg Med Chem Lett 19: 4115-8 (2009) Article DOI: 10.1016/j.bmcl.2009.06.008 BindingDB Entry DOI: 10.7270/Q2ZS2WJX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50326884 ((S)-N-((S)-1-amino-1-oxo-3-phenylpropan-2-yl)-2-(2...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 293 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
"Sapienza" Università di Roma Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 3 hrs by liquid scintillation counting | Eur J Med Chem 45: 4594-600 (2010) Article DOI: 10.1016/j.ejmech.2010.07.022 BindingDB Entry DOI: 10.7270/Q2KK9C0Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50386560 (CHEMBL2048250) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 310 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Chieti-Pescara G. d'Annunzio Curated by ChEMBL | Assay Description Displacement of [3H]-DAMGO from rat mu opioid receptor expressed in HN9.10 cells after 3 hrs by scintillation counting | J Med Chem 55: 3027-35 (2012) Article DOI: 10.1021/jm201402v BindingDB Entry DOI: 10.7270/Q2571D38 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50326890 ((S)-N-((S)-1-amino-1-oxo-3-phenylpropan-2-yl)-2-((...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 510 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
"Sapienza" Università di Roma Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 3 hrs by liquid scintillation counting | Eur J Med Chem 45: 4594-600 (2010) Article DOI: 10.1016/j.ejmech.2010.07.022 BindingDB Entry DOI: 10.7270/Q2KK9C0Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50386559 (CHEMBL2048248) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 660 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Chieti-Pescara G. d'Annunzio Curated by ChEMBL | Assay Description Displacement of [3H]-DAMGO from rat mu opioid receptor expressed in HN9.10 cells after 3 hrs by scintillation counting | J Med Chem 55: 3027-35 (2012) Article DOI: 10.1021/jm201402v BindingDB Entry DOI: 10.7270/Q2571D38 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50295261 (CHEMBL549770 | N-((S)-1-((S)-1-amino-1-oxo-3-pheny...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 710 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Roma Curated by ChEMBL | Assay Description Displacement of [3H]DPDE from delta opioid receptor in rat brain membrane by liquid scintillation counting | Bioorg Med Chem Lett 19: 4115-8 (2009) Article DOI: 10.1016/j.bmcl.2009.06.008 BindingDB Entry DOI: 10.7270/Q2ZS2WJX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Rattus norvegicus (rat)) | BDBM50326885 ((S)-N-((S)-1-amino-1-oxo-3-phenylpropan-2-yl)-2-(2...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 990 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
"Sapienza" Università di Roma Curated by ChEMBL | Assay Description Displacement of [3H]DPDPE from kappa opioid receptor in rat brain membrane after 3 hrs by liquid scintillation counting | Eur J Med Chem 45: 4594-600 (2010) Article DOI: 10.1016/j.ejmech.2010.07.022 BindingDB Entry DOI: 10.7270/Q2KK9C0Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50386561 (CHEMBL2048249) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Chieti-Pescara G. d'Annunzio Curated by ChEMBL | Assay Description Displacement of [3H]-DAMGO from rat mu opioid receptor expressed in HN9.10 cells after 3 hrs by scintillation counting | J Med Chem 55: 3027-35 (2012) Article DOI: 10.1021/jm201402v BindingDB Entry DOI: 10.7270/Q2571D38 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Rattus norvegicus (rat)) | BDBM50326889 ((S)-N-((S)-1-amino-1-oxo-3-phenylpropan-2-yl)-2-((...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
"Sapienza" Università di Roma Curated by ChEMBL | Assay Description Displacement of [3H]DPDPE from kappa opioid receptor in rat brain membrane after 3 hrs by liquid scintillation counting | Eur J Med Chem 45: 4594-600 (2010) Article DOI: 10.1016/j.ejmech.2010.07.022 BindingDB Entry DOI: 10.7270/Q2KK9C0Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50295263 ((S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-y...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Roma Curated by ChEMBL | Assay Description Displacement of [3H]DPDE from delta opioid receptor in rat brain membrane by liquid scintillation counting | Bioorg Med Chem Lett 19: 4115-8 (2009) Article DOI: 10.1016/j.bmcl.2009.06.008 BindingDB Entry DOI: 10.7270/Q2ZS2WJX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Rattus norvegicus (rat)) | BDBM50326887 ((R)-1-((S)-2-(2-((S)-1-((S)-2-amino-3-(4-hydroxyph...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
"Sapienza" Università di Roma Curated by ChEMBL | Assay Description Displacement of [3H]DPDPE from kappa opioid receptor in rat brain membrane after 3 hrs by liquid scintillation counting | Eur J Med Chem 45: 4594-600 (2010) Article DOI: 10.1016/j.ejmech.2010.07.022 BindingDB Entry DOI: 10.7270/Q2KK9C0Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Rattus norvegicus (rat)) | BDBM50326883 ((S)-N-((S)-1-amino-1-oxo-3-phenylpropan-2-yl)-2-((...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
"Sapienza" Università di Roma Curated by ChEMBL | Assay Description Displacement of [3H]DPDPE from kappa opioid receptor in rat brain membrane after 3 hrs by liquid scintillation counting | Eur J Med Chem 45: 4594-600 (2010) Article DOI: 10.1016/j.ejmech.2010.07.022 BindingDB Entry DOI: 10.7270/Q2KK9C0Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50295264 ((S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-y...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 5.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Roma Curated by ChEMBL | Assay Description Displacement of [3H]DPDE from delta opioid receptor in rat brain membrane by liquid scintillation counting | Bioorg Med Chem Lett 19: 4115-8 (2009) Article DOI: 10.1016/j.bmcl.2009.06.008 BindingDB Entry DOI: 10.7270/Q2ZS2WJX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50326887 ((R)-1-((S)-2-(2-((S)-1-((S)-2-amino-3-(4-hydroxyph...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 6.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
"Sapienza" Università di Roma Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 3 hrs by liquid scintillation counting | Eur J Med Chem 45: 4594-600 (2010) Article DOI: 10.1016/j.ejmech.2010.07.022 BindingDB Entry DOI: 10.7270/Q2KK9C0Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Rattus norvegicus (rat)) | BDBM50326890 ((S)-N-((S)-1-amino-1-oxo-3-phenylpropan-2-yl)-2-((...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 6.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
"Sapienza" Università di Roma Curated by ChEMBL | Assay Description Displacement of [3H]DPDPE from kappa opioid receptor in rat brain membrane after 3 hrs by liquid scintillation counting | Eur J Med Chem 45: 4594-600 (2010) Article DOI: 10.1016/j.ejmech.2010.07.022 BindingDB Entry DOI: 10.7270/Q2KK9C0Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50295260 (CHEMBL564939 | N-((S)-1-((S)-1-amino-1-oxo-3-pheny...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 6.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Roma Curated by ChEMBL | Assay Description Displacement of [3H]DPDE from delta opioid receptor in rat brain membrane by liquid scintillation counting | Bioorg Med Chem Lett 19: 4115-8 (2009) Article DOI: 10.1016/j.bmcl.2009.06.008 BindingDB Entry DOI: 10.7270/Q2ZS2WJX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Rattus norvegicus (rat)) | BDBM50326888 ((S)-N-((S)-1-amino-1-oxo-3-phenylpropan-2-yl)-2-((...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 7.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
"Sapienza" Università di Roma Curated by ChEMBL | Assay Description Displacement of [3H]DPDPE from kappa opioid receptor in rat brain membrane after 3 hrs by liquid scintillation counting | Eur J Med Chem 45: 4594-600 (2010) Article DOI: 10.1016/j.ejmech.2010.07.022 BindingDB Entry DOI: 10.7270/Q2KK9C0Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Homo sapiens (Human)) | BDBM50320023 ((S)-1-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)-N...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 7.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Roma Curated by ChEMBL | Assay Description Displacement of [3H]DPDPE from human delta opioid receptor expressed in HEK293 cells | J Med Chem 53: 4550-4 (2010) Article DOI: 10.1021/jm1001343 BindingDB Entry DOI: 10.7270/Q23F4PTK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Homo sapiens (Human)) | BDBM50320022 ((S)-1-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)-N...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Roma Curated by ChEMBL | Assay Description Displacement of [3H]DPDPE from human delta opioid receptor expressed in HEK293 cells | J Med Chem 53: 4550-4 (2010) Article DOI: 10.1021/jm1001343 BindingDB Entry DOI: 10.7270/Q23F4PTK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Rattus norvegicus (rat)) | BDBM50326886 ((R)-1-((S)-2-(2-((R)-1-((S)-2-amino-3-(4-hydroxyph...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
"Sapienza" Università di Roma Curated by ChEMBL | Assay Description Displacement of [3H]DPDPE from kappa opioid receptor in rat brain membrane after 3 hrs by liquid scintillation counting | Eur J Med Chem 45: 4594-600 (2010) Article DOI: 10.1016/j.ejmech.2010.07.022 BindingDB Entry DOI: 10.7270/Q2KK9C0Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Rattus norvegicus (rat)) | BDBM50326884 ((S)-N-((S)-1-amino-1-oxo-3-phenylpropan-2-yl)-2-(2...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
"Sapienza" Università di Roma Curated by ChEMBL | Assay Description Displacement of [3H]DPDPE from kappa opioid receptor in rat brain membrane after 3 hrs by liquid scintillation counting | Eur J Med Chem 45: 4594-600 (2010) Article DOI: 10.1016/j.ejmech.2010.07.022 BindingDB Entry DOI: 10.7270/Q2KK9C0Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (GUINEA PIG) | BDBM50139013 ((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 15 | n/a | n/a | n/a | n/a | n/a | n/a |
"Sapienza" Università di Roma Curated by ChEMBL | Assay Description Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contraction | Eur J Med Chem 45: 4594-600 (2010) Article DOI: 10.1016/j.ejmech.2010.07.022 BindingDB Entry DOI: 10.7270/Q2KK9C0Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (GUINEA PIG) | BDBM50139013 ((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 15 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Roma Curated by ChEMBL | Assay Description Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contraction | J Med Chem 53: 4550-4 (2010) Article DOI: 10.1021/jm1001343 BindingDB Entry DOI: 10.7270/Q23F4PTK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (GUINEA PIG) | BDBM50326886 ((R)-1-((S)-2-(2-((R)-1-((S)-2-amino-3-(4-hydroxyph...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 17 | n/a | n/a | n/a | n/a | n/a | n/a |
"Sapienza" Università di Roma Curated by ChEMBL | Assay Description Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contraction | Eur J Med Chem 45: 4594-600 (2010) Article DOI: 10.1016/j.ejmech.2010.07.022 BindingDB Entry DOI: 10.7270/Q2KK9C0Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (GUINEA PIG) | BDBM50320022 ((S)-1-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)-N...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 25 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Roma Curated by ChEMBL | Assay Description Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contraction | J Med Chem 53: 4550-4 (2010) Article DOI: 10.1021/jm1001343 BindingDB Entry DOI: 10.7270/Q23F4PTK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (MOUSE) | BDBM50326886 ((R)-1-((S)-2-(2-((R)-1-((S)-2-amino-3-(4-hydroxyph...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 96 | n/a | n/a | n/a | n/a | n/a | n/a |
"Sapienza" Università di Roma Curated by ChEMBL | Assay Description Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contraction | Eur J Med Chem 45: 4594-600 (2010) Article DOI: 10.1016/j.ejmech.2010.07.022 BindingDB Entry DOI: 10.7270/Q2KK9C0Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (GUINEA PIG) | BDBM50320024 ((S)-N-(3-((S)-1-amino-1-oxo-3-phenylpropan-2-ylami...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 170 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Roma Curated by ChEMBL | Assay Description Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contraction | J Med Chem 53: 4550-4 (2010) Article DOI: 10.1021/jm1001343 BindingDB Entry DOI: 10.7270/Q23F4PTK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (GUINEA PIG) | BDBM50326888 ((S)-N-((S)-1-amino-1-oxo-3-phenylpropan-2-yl)-2-((...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 220 | n/a | n/a | n/a | n/a | n/a | n/a |
"Sapienza" Università di Roma Curated by ChEMBL | Assay Description Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contraction | Eur J Med Chem 45: 4594-600 (2010) Article DOI: 10.1016/j.ejmech.2010.07.022 BindingDB Entry DOI: 10.7270/Q2KK9C0Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (GUINEA PIG) | BDBM50326885 ((S)-N-((S)-1-amino-1-oxo-3-phenylpropan-2-yl)-2-(2...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 260 | n/a | n/a | n/a | n/a | n/a | n/a |
"Sapienza" Università di Roma Curated by ChEMBL | Assay Description Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contraction | Eur J Med Chem 45: 4594-600 (2010) Article DOI: 10.1016/j.ejmech.2010.07.022 BindingDB Entry DOI: 10.7270/Q2KK9C0Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (GUINEA PIG) | BDBM50326889 ((S)-N-((S)-1-amino-1-oxo-3-phenylpropan-2-yl)-2-((...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 260 | n/a | n/a | n/a | n/a | n/a | n/a |
"Sapienza" Università di Roma Curated by ChEMBL | Assay Description Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contraction | Eur J Med Chem 45: 4594-600 (2010) Article DOI: 10.1016/j.ejmech.2010.07.022 BindingDB Entry DOI: 10.7270/Q2KK9C0Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (GUINEA PIG) | BDBM50320023 ((S)-1-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)-N...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 330 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Roma Curated by ChEMBL | Assay Description Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contraction | J Med Chem 53: 4550-4 (2010) Article DOI: 10.1021/jm1001343 BindingDB Entry DOI: 10.7270/Q23F4PTK | |||||||||||
More data for this Ligand-Target Pair |
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