Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
DNA topoisomerase 2-alpha (Homo sapiens (Human)) | BDBM50369152 (CHEMBL1627911) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.41E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Purdue University Curated by ChEMBL | Assay Description Inhibitory activity against topoisomerase II determined in catenation inhibition assay | J Med Chem 39: 3367-74 (1996) Article DOI: 10.1021/jm9602930 BindingDB Entry DOI: 10.7270/Q2736RKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 2-alpha (Homo sapiens (Human)) | BDBM50369153 (CHEMBL1628076) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >2.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Purdue University Curated by ChEMBL | Assay Description Inhibitory activity against topoisomerase II determined in catenation inhibition assay | J Med Chem 39: 3367-74 (1996) Article DOI: 10.1021/jm9602930 BindingDB Entry DOI: 10.7270/Q2736RKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 2-alpha (Homo sapiens (Human)) | BDBM50369151 (CHEMBL1627914) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >2.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Purdue University Curated by ChEMBL | Assay Description Inhibitory activity against topoisomerase II determined in catenation inhibition assay | J Med Chem 39: 3367-74 (1996) Article DOI: 10.1021/jm9602930 BindingDB Entry DOI: 10.7270/Q2736RKT | |||||||||||
More data for this Ligand-Target Pair |