Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Prothrombin (Bos taurus (Bovine)) | BDBM50442068 (CHEMBL2441057) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Bos taurus (Bovine)) | BDBM50442068 (CHEMBL2441057) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Bos taurus (Bovine)) | BDBM50442069 (CHEMBL2441037) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 31 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Bos taurus (Bovine)) | BDBM50442073 (CHEMBL2441035) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 53 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Bos taurus (Bovine)) | BDBM50442070 (CHEMBL2441054) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 63 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Bos taurus (Bovine)) | BDBM50442071 (CHEMBL2441055) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 64 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Bos taurus (Bovine)) | BDBM50442074 (CHEMBL2441036) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 83 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Bos taurus (Bovine)) | BDBM50442075 (CHEMBL2441047) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 124 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Coagulation factor X (Homo sapiens (Human)) | BDBM50442079 (CHEMBL2441033) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 133 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of human factor 10a using Z-D-Arg-Gly-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Bos taurus (Bovine)) | BDBM50442093 (CHEMBL2441053) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 156 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Bos taurus (Bovine)) | BDBM50442072 (CHEMBL2441058) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 211 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Bos taurus (Bovine)) | BDBM50442094 (CHEMBL2441052) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 260 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Coagulation factor X (Homo sapiens (Human)) | BDBM50442069 (CHEMBL2441037) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 606 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of human factor 10a using Z-D-Arg-Gly-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Coagulation factor X (Homo sapiens (Human)) | BDBM50442078 (CHEMBL2441030) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 774 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of human factor 10a using Z-D-Arg-Gly-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Coagulation factor X (Homo sapiens (Human)) | BDBM50442072 (CHEMBL2441058) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of human factor 10a using Z-D-Arg-Gly-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Bos taurus (Bovine)) | BDBM50442081 (CHEMBL2441039) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.15E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Bos taurus (Bovine)) | BDBM50442080 (CHEMBL2441040) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Bos taurus (Bovine)) | BDBM50442092 (CHEMBL2441051) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.03E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Bos taurus (Bovine)) | BDBM50442082 (CHEMBL2441038) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.03E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Coagulation factor X (Homo sapiens (Human)) | BDBM50442065 (CHEMBL2441032) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.14E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of human factor 10a using Z-D-Arg-Gly-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Bos taurus (Bovine)) | BDBM50442086 (CHEMBL2441044) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Coagulation factor X (Homo sapiens (Human)) | BDBM50442073 (CHEMBL2441035) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.72E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of human factor 10a using Z-D-Arg-Gly-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Bos taurus (Bovine)) | BDBM50442076 (CHEMBL2441029) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.72E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Coagulation factor X (Homo sapiens (Human)) | BDBM50442067 (CHEMBL2441027) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.83E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of human factor 10a using Z-D-Arg-Gly-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Bos taurus (Bovine)) | BDBM50442079 (CHEMBL2441033) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.46E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Bos taurus (Bovine)) | BDBM50442095 (CHEMBL2441056) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.64E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Coagulation factor X (Homo sapiens (Human)) | BDBM50442068 (CHEMBL2441057) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 5.64E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of human factor 10a using Z-D-Arg-Gly-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Bos taurus (Bovine)) | BDBM50442090 (CHEMBL2441049) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 5.85E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Coagulation factor X (Homo sapiens (Human)) | BDBM50442090 (CHEMBL2441049) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 6.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of human factor 10a using Z-D-Arg-Gly-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Coagulation factor X (Homo sapiens (Human)) | BDBM50442091 (CHEMBL2441050) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 6.31E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of human factor 10a using Z-D-Arg-Gly-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chymotrypsinogen A (Bos taurus (bovine)) | BDBM50442068 (CHEMBL2441057) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 6.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of bovine alpha-chymotrypsin using N-succinyl-Ala-Ala-Pro-Phe-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Bos taurus (Bovine)) | BDBM50442062 (CHEMBL2441025) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 6.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Coagulation factor X (Homo sapiens (Human)) | BDBM50442089 (CHEMBL2441048) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 6.73E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of human factor 10a using Z-D-Arg-Gly-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Coagulation factor X (Homo sapiens (Human)) | BDBM50442071 (CHEMBL2441055) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 6.83E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of human factor 10a using Z-D-Arg-Gly-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Coagulation factor X (Homo sapiens (Human)) | BDBM50442081 (CHEMBL2441039) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 7.23E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of human factor 10a using Z-D-Arg-Gly-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Coagulation factor X (Homo sapiens (Human)) | BDBM50442096 (CHEMBL2441060) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 7.46E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of human factor 10a using Z-D-Arg-Gly-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Coagulation factor X (Homo sapiens (Human)) | BDBM50442075 (CHEMBL2441047) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 7.73E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of human factor 10a using Z-D-Arg-Gly-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Bos taurus (Bovine)) | BDBM50442083 (CHEMBL2441041) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 8.19E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Coagulation factor X (Homo sapiens (Human)) | BDBM50442095 (CHEMBL2441056) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 8.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of human factor 10a using Z-D-Arg-Gly-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Bos taurus (Bovine)) | BDBM50442085 (CHEMBL2441043) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Coagulation factor X (Homo sapiens (Human)) | BDBM50442082 (CHEMBL2441038) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.11E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of human factor 10a using Z-D-Arg-Gly-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutrophil elastase (Homo sapiens (Human)) | BDBM50442068 (CHEMBL2441057) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.13E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of human neutrophil leukocyte elastase using N-(methoxysuccinyl)-Ala-Ala-Pro-Val-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Coagulation factor X (Homo sapiens (Human)) | BDBM50442083 (CHEMBL2441041) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.22E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of human factor 10a using Z-D-Arg-Gly-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Bos taurus (Bovine)) | BDBM50442087 (CHEMBL2441046) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.23E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Bos taurus (Bovine)) | BDBM50442064 (CHEMBL2441028) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.23E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Bos taurus (Bovine)) | BDBM50442064 (CHEMBL2441028) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.24E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Bos taurus (Bovine)) | BDBM50442084 (CHEMBL2441042) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.33E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Bos taurus (Bovine)) | BDBM50442100 (CHEMBL2441064) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.53E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Coagulation factor X (Homo sapiens (Human)) | BDBM50442088 (CHEMBL2441045) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.56E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of human factor 10a using Z-D-Arg-Gly-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prothrombin (Bos taurus (Bovine)) | BDBM50442088 (CHEMBL2441045) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.59E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bari "Aldo Moro" Curated by ChEMBL | Assay Description Inhibition of bovine thrombin using D-Phe-Pip-Arg-p-NA as substrate by chromogenic assay | J Med Chem 56: 8696-711 (2013) Article DOI: 10.1021/jm401169a BindingDB Entry DOI: 10.7270/Q2SN0BDT | |||||||||||
More data for this Ligand-Target Pair |
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