Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Ubiquitin-like modifier-activating enzyme 1 (Homo sapiens (Human)) | BDBM50387035 (CHEMBL2046768) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Kumamoto University Curated by ChEMBL | Assay Description Inhibition of FLAG-tagged ubiquitin-activating enzyme E1 assessed as inhibition of GST-ubiquitin/FLAG-E1 intermediate formation by Western blot analy... | Bioorg Med Chem 20: 4437-42 (2012) Article DOI: 10.1016/j.bmc.2012.05.044 BindingDB Entry DOI: 10.7270/Q2WH2R2M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ubiquitin-like modifier-activating enzyme 1 (Homo sapiens (Human)) | BDBM50322422 (CHEMBL1173445 | Largazole) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 2.90E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kumamoto University Curated by ChEMBL | Assay Description Inhibition of recombinant fluorescein-tagged E1 assessed as inhibition of ubiquitin-E1 adduct formation incubated for 15 mins prior to ATP addition m... | Bioorg Med Chem 20: 4437-42 (2012) Article DOI: 10.1016/j.bmc.2012.05.044 BindingDB Entry DOI: 10.7270/Q2WH2R2M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ubiquitin-like modifier-activating enzyme 1 (Homo sapiens (Human)) | BDBM50387034 (CHEMBL2046769) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kumamoto University Curated by ChEMBL | Assay Description Inhibition of FLAG-tagged ubiquitin-activating enzyme E1 assessed as inhibition of GST-ubiquitin/FLAG-E1 intermediate formation by Western blot analy... | Bioorg Med Chem 20: 4437-42 (2012) Article DOI: 10.1016/j.bmc.2012.05.044 BindingDB Entry DOI: 10.7270/Q2WH2R2M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ubiquitin-like modifier-activating enzyme 1 (Homo sapiens (Human)) | BDBM50387036 (CHEMBL2046774) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kumamoto University Curated by ChEMBL | Assay Description Inhibition of ubiquitin-activating enzyme E1 | Bioorg Med Chem 20: 4437-42 (2012) Article DOI: 10.1016/j.bmc.2012.05.044 BindingDB Entry DOI: 10.7270/Q2WH2R2M | |||||||||||
More data for this Ligand-Target Pair |