Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Beta-1 adrenergic receptor (Rattus norvegicus (Rat)) | BDBM50337291 (1-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroq...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Agonist activity at beta1 adrenoreceptor in rat left atria assessed as induction of ionotropic effect | Bioorg Med Chem Lett 21: 1545-8 (2011) Article DOI: 10.1016/j.bmcl.2010.12.096 BindingDB Entry DOI: 10.7270/Q2W09668 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-1 adrenergic receptor (Rattus norvegicus (Rat)) | BDBM50337301 (1-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroq...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Agonist activity at beta1 adrenoreceptor in rat left atria assessed as induction of ionotropic effect | Bioorg Med Chem Lett 21: 1545-8 (2011) Article DOI: 10.1016/j.bmcl.2010.12.096 BindingDB Entry DOI: 10.7270/Q2W09668 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-1 adrenergic receptor (Rattus norvegicus (Rat)) | BDBM50337293 (1-(4-fluorobenzyl)-3-(3-(2-(2-hydroxy-2-(8-hydroxy...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 6.30E+3 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Agonist activity at beta1 adrenoreceptor in rat left atria assessed as induction of ionotropic effect | Bioorg Med Chem Lett 21: 1545-8 (2011) Article DOI: 10.1016/j.bmcl.2010.12.096 BindingDB Entry DOI: 10.7270/Q2W09668 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-1 adrenergic receptor (Rattus norvegicus (Rat)) | BDBM50337294 (1-(2,6-dichlorobenzyl)-3-(3-(2-(2-hydroxy-2-(8-hyd...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.60E+3 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Agonist activity at beta1 adrenoreceptor in rat left atria assessed as induction of ionotropic effect | Bioorg Med Chem Lett 21: 1545-8 (2011) Article DOI: 10.1016/j.bmcl.2010.12.096 BindingDB Entry DOI: 10.7270/Q2W09668 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-1 adrenergic receptor (Rattus norvegicus (Rat)) | BDBM50337295 (1-benzhydryl-3-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 8.89E+3 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Agonist activity at beta1 adrenoreceptor in rat left atria assessed as induction of ionotropic effect | Bioorg Med Chem Lett 21: 1545-8 (2011) Article DOI: 10.1016/j.bmcl.2010.12.096 BindingDB Entry DOI: 10.7270/Q2W09668 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-1 adrenergic receptor (Rattus norvegicus (Rat)) | BDBM50337296 (1-(biphenyl-2-yl)-3-(3-(2-(2-hydroxy-2-(8-hydroxy-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 5.77E+3 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Agonist activity at beta1 adrenoreceptor in rat left atria assessed as induction of ionotropic effect | Bioorg Med Chem Lett 21: 1545-8 (2011) Article DOI: 10.1016/j.bmcl.2010.12.096 BindingDB Entry DOI: 10.7270/Q2W09668 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-1 adrenergic receptor (Rattus norvegicus (Rat)) | BDBM50337297 (1-Adamantan-1-ylmethyl-3-(3-{2-[2-hydroxy-2-(8-hyd...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 296 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Agonist activity at beta1 adrenoreceptor in rat left atria assessed as induction of ionotropic effect | Bioorg Med Chem Lett 21: 1545-8 (2011) Article DOI: 10.1016/j.bmcl.2010.12.096 BindingDB Entry DOI: 10.7270/Q2W09668 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-1 adrenergic receptor (Rattus norvegicus (Rat)) | BDBM50337298 (1-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroq...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.00E+4 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Agonist activity at beta1 adrenoreceptor in rat left atria assessed as induction of ionotropic effect | Bioorg Med Chem Lett 21: 1545-8 (2011) Article DOI: 10.1016/j.bmcl.2010.12.096 BindingDB Entry DOI: 10.7270/Q2W09668 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-1 adrenergic receptor (Rattus norvegicus (Rat)) | BDBM50318159 (8-Hydroxy-5-[(R)-1-hydroxy-2-(5,6-diethylindan-2-y...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.31E+3 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Agonist activity at beta1 adrenoreceptor in rat left atria assessed as induction of ionotropic effect | Bioorg Med Chem Lett 21: 1545-8 (2011) Article DOI: 10.1016/j.bmcl.2010.12.096 BindingDB Entry DOI: 10.7270/Q2W09668 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-2 adrenergic receptor (GUINEA PIG) | BDBM50337299 (1-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroq...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.0700 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Agonist activity at beta2 adrenoreceptor in guinea pig tracheal rings assessed as vasorelaxation | Bioorg Med Chem Lett 21: 1545-8 (2011) Article DOI: 10.1016/j.bmcl.2010.12.096 BindingDB Entry DOI: 10.7270/Q2W09668 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-2 adrenergic receptor (GUINEA PIG) | BDBM50337300 (1-benzyl-3-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.200 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Agonist activity at beta2 adrenoreceptor in guinea pig tracheal rings assessed as vasorelaxation | Bioorg Med Chem Lett 21: 1545-8 (2011) Article DOI: 10.1016/j.bmcl.2010.12.096 BindingDB Entry DOI: 10.7270/Q2W09668 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-2 adrenergic receptor (GUINEA PIG) | BDBM50337301 (1-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroq...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.0900 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Agonist activity at beta2 adrenoreceptor in guinea pig tracheal rings assessed as vasorelaxation | Bioorg Med Chem Lett 21: 1545-8 (2011) Article DOI: 10.1016/j.bmcl.2010.12.096 BindingDB Entry DOI: 10.7270/Q2W09668 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-2 adrenergic receptor (GUINEA PIG) | BDBM50337291 (1-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroq...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.0500 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Agonist activity at beta2 adrenoreceptor in guinea pig tracheal rings assessed as vasorelaxation | Bioorg Med Chem Lett 21: 1545-8 (2011) Article DOI: 10.1016/j.bmcl.2010.12.096 BindingDB Entry DOI: 10.7270/Q2W09668 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-2 adrenergic receptor (GUINEA PIG) | BDBM50337302 (3-((3-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihy...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.130 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Agonist activity at beta2 adrenoreceptor in guinea pig tracheal rings assessed as vasorelaxation | Bioorg Med Chem Lett 21: 1545-8 (2011) Article DOI: 10.1016/j.bmcl.2010.12.096 BindingDB Entry DOI: 10.7270/Q2W09668 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-2 adrenergic receptor (GUINEA PIG) | BDBM50337292 (1-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroq...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.200 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Agonist activity at beta2 adrenoreceptor in guinea pig tracheal rings assessed as vasorelaxation | Bioorg Med Chem Lett 21: 1545-8 (2011) Article DOI: 10.1016/j.bmcl.2010.12.096 BindingDB Entry DOI: 10.7270/Q2W09668 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-2 adrenergic receptor (GUINEA PIG) | BDBM50337293 (1-(4-fluorobenzyl)-3-(3-(2-(2-hydroxy-2-(8-hydroxy...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.200 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Agonist activity at beta2 adrenoreceptor in guinea pig tracheal rings assessed as vasorelaxation | Bioorg Med Chem Lett 21: 1545-8 (2011) Article DOI: 10.1016/j.bmcl.2010.12.096 BindingDB Entry DOI: 10.7270/Q2W09668 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-2 adrenergic receptor (GUINEA PIG) | BDBM50337294 (1-(2,6-dichlorobenzyl)-3-(3-(2-(2-hydroxy-2-(8-hyd...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.200 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Agonist activity at beta2 adrenoreceptor in guinea pig tracheal rings assessed as vasorelaxation | Bioorg Med Chem Lett 21: 1545-8 (2011) Article DOI: 10.1016/j.bmcl.2010.12.096 BindingDB Entry DOI: 10.7270/Q2W09668 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-2 adrenergic receptor (GUINEA PIG) | BDBM50337295 (1-benzhydryl-3-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.200 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Agonist activity at beta2 adrenoreceptor in guinea pig tracheal rings assessed as vasorelaxation | Bioorg Med Chem Lett 21: 1545-8 (2011) Article DOI: 10.1016/j.bmcl.2010.12.096 BindingDB Entry DOI: 10.7270/Q2W09668 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-2 adrenergic receptor (GUINEA PIG) | BDBM50337296 (1-(biphenyl-2-yl)-3-(3-(2-(2-hydroxy-2-(8-hydroxy-...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.700 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Agonist activity at beta2 adrenoreceptor in guinea pig tracheal rings assessed as vasorelaxation | Bioorg Med Chem Lett 21: 1545-8 (2011) Article DOI: 10.1016/j.bmcl.2010.12.096 BindingDB Entry DOI: 10.7270/Q2W09668 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-2 adrenergic receptor (GUINEA PIG) | BDBM50337297 (1-Adamantan-1-ylmethyl-3-(3-{2-[2-hydroxy-2-(8-hyd...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.20 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Agonist activity at beta2 adrenoreceptor in guinea pig tracheal rings assessed as vasorelaxation | Bioorg Med Chem Lett 21: 1545-8 (2011) Article DOI: 10.1016/j.bmcl.2010.12.096 BindingDB Entry DOI: 10.7270/Q2W09668 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-2 adrenergic receptor (GUINEA PIG) | BDBM50337298 (1-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroq...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Agonist activity at beta2 adrenoreceptor in guinea pig tracheal rings assessed as vasorelaxation | Bioorg Med Chem Lett 21: 1545-8 (2011) Article DOI: 10.1016/j.bmcl.2010.12.096 BindingDB Entry DOI: 10.7270/Q2W09668 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-2 adrenergic receptor (GUINEA PIG) | BDBM50337303 (1-(4-tert-butylbenzyl)-3-(3-(2-(2-hydroxy-2-(8-hyd...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.900 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Agonist activity at beta2 adrenoreceptor in guinea pig tracheal rings assessed as vasorelaxation | Bioorg Med Chem Lett 21: 1545-8 (2011) Article DOI: 10.1016/j.bmcl.2010.12.096 BindingDB Entry DOI: 10.7270/Q2W09668 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-2 adrenergic receptor (GUINEA PIG) | BDBM50318159 (8-Hydroxy-5-[(R)-1-hydroxy-2-(5,6-diethylindan-2-y...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 1 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Agonist activity at beta2 adrenoreceptor in guinea pig tracheal rings assessed as vasorelaxation | Bioorg Med Chem Lett 21: 1545-8 (2011) Article DOI: 10.1016/j.bmcl.2010.12.096 BindingDB Entry DOI: 10.7270/Q2W09668 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-1 adrenergic receptor (Rattus norvegicus (Rat)) | BDBM50337299 (1-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroq...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Agonist activity at beta1 adrenoreceptor in rat left atria assessed as induction of ionotropic effect | Bioorg Med Chem Lett 21: 1545-8 (2011) Article DOI: 10.1016/j.bmcl.2010.12.096 BindingDB Entry DOI: 10.7270/Q2W09668 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-1 adrenergic receptor (Rattus norvegicus (Rat)) | BDBM50337300 (1-benzyl-3-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 900 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Agonist activity at beta1 adrenoreceptor in rat left atria assessed as induction of ionotropic effect | Bioorg Med Chem Lett 21: 1545-8 (2011) Article DOI: 10.1016/j.bmcl.2010.12.096 BindingDB Entry DOI: 10.7270/Q2W09668 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-1 adrenergic receptor (Rattus norvegicus (Rat)) | BDBM50337292 (1-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroq...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 550 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Agonist activity at beta1 adrenoreceptor in rat left atria assessed as induction of ionotropic effect | Bioorg Med Chem Lett 21: 1545-8 (2011) Article DOI: 10.1016/j.bmcl.2010.12.096 BindingDB Entry DOI: 10.7270/Q2W09668 | |||||||||||
More data for this Ligand-Target Pair |