Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Proteasome subunit beta type-5 (Homo sapiens (Human)) | BDBM50088583 (CHEMBL3577367) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 360 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Prince Edward Island Curated by ChEMBL | Assay Description Inhibition of chymotrypsin-like activity of human erythrocyte-derived 20S proteasome using Suc-LLVY-AMC as substrate preincubated for 10 mins followe... | J Nat Prod 78: 822-6 (2015) Article DOI: 10.1021/np501060k BindingDB Entry DOI: 10.7270/Q2MG7R7X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteasome subunit beta type-5 (Homo sapiens (Human)) | BDBM50088584 (CHEMBL3577368) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 930 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Prince Edward Island Curated by ChEMBL | Assay Description Inhibition of chymotrypsin-like activity of human erythrocyte-derived 20S proteasome using Suc-LLVY-AMC as substrate preincubated for 10 mins followe... | J Nat Prod 78: 822-6 (2015) Article DOI: 10.1021/np501060k BindingDB Entry DOI: 10.7270/Q2MG7R7X | |||||||||||
More data for this Ligand-Target Pair |