Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50121716 ((3-methyl-4-(3-(pyridin-3-ylmethylamino)propoxy)be...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 0.390 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description In vitro inhibitory activity against candida albicans Nmt (CaNmt) using substrate peptide GLTISKLFR-R-NH2 (0.5 uM) and myristoyl-CoA (0.5 uM) | Bioorg Med Chem Lett 13: 87-91 (2003) BindingDB Entry DOI: 10.7270/Q25D8V2K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50220561 (CHEMBL173370) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 0.400 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description In vitro inhibitory activity against Candida albicans Nmt (CaNmt) using substrate peptide GLTISKLFR-R-NH2 (0.5 uM) and myristoyl-CoA (0.5 uM) | Bioorg Med Chem Lett 13: 87-91 (2003) BindingDB Entry DOI: 10.7270/Q25D8V2K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50220562 (CHEMBL171506) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | 0.580 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description In vitro inhibitory activity against Candida albicans Nmt (CaNmt) using substrate peptide GLTISKLFR-R-NH2 (0.5 uM) and myristoyl-CoA (0.5 uM) | Bioorg Med Chem Lett 13: 87-91 (2003) BindingDB Entry DOI: 10.7270/Q25D8V2K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50220565 (CHEMBL170524) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | 0.710 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description In vitro inhibitory activity against Candida albicans Nmt (CaNmt) using substrate peptide GLTISKLFR-R-NH2 (0.5 uM) and myristoyl-CoA (0.5 uM) | Bioorg Med Chem Lett 13: 87-91 (2003) BindingDB Entry DOI: 10.7270/Q25D8V2K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50220569 (CHEMBL422896) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | 1.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description In vitro inhibitory activity against Candida albicans Nmt (CaNmt) using substrate peptide GLTISKLFR-R-NH2 (0.5 uM) and myristoyl-CoA (0.5 uM) | Bioorg Med Chem Lett 13: 87-91 (2003) BindingDB Entry DOI: 10.7270/Q25D8V2K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50121720 ((1-METHYL-1H-IMIDAZOL-2-YL)-(3-METHYL-4-{3-[(PYRID...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL DrugBank MMDB PC cid PC sid PDB UniChem Similars | PubMed | n/a | n/a | 1.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description In vitro inhibitory activity against Candida albicans Nmt (CaNmt) using substrate peptide GLTISKLFR-R-NH2 (0.5 uM) and myristoyl-CoA (0.5 uM) | Bioorg Med Chem Lett 13: 87-91 (2003) BindingDB Entry DOI: 10.7270/Q25D8V2K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50220559 (CHEMBL422746) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description In vitro inhibitory activity against Candida albicans Nmt (CaNmt) using substrate peptide GLTISKLFR-R-NH2 (0.5 uM) and myristoyl-CoA (0.5 uM) | Bioorg Med Chem Lett 13: 87-91 (2003) BindingDB Entry DOI: 10.7270/Q25D8V2K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50220571 (CHEMBL355250) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | 3.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description In vitro inhibitory activity against Candida albicans Nmt (CaNmt) using substrate peptide GLTISKLFR-R-NH2 (0.5 uM) and myristoyl-CoA (0.5 uM) | Bioorg Med Chem Lett 13: 87-91 (2003) BindingDB Entry DOI: 10.7270/Q25D8V2K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50109882 (3-(3-methyl-2-((2,3,4-trifluorophenoxy)methyl)benz...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Patents Similars | PubMed | n/a | n/a | 3.70 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description Inhibitory activity against Candida albicans (Nmt) assessed as inhibitory concentration (nM); 3.7-9.4 nM | Bioorg Med Chem Lett 12: 607-10 (2002) BindingDB Entry DOI: 10.7270/Q2PC34K1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50219310 (CHEMBL155469) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 3.70 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description Inhibitory activity against Candida albicans N-Myristoyltransferase (Nmt) | Bioorg Med Chem Lett 12: 607-10 (2002) BindingDB Entry DOI: 10.7270/Q2PC34K1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50109879 (CHEMBL155301 | Non peptidic, 4 | {3-[2-(2,3-Difluo...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 3.70 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description Inhibitory activity against Candida albicans (Nmt) assessed as inhibitory concentration (nM) | Bioorg Med Chem Lett 12: 607-10 (2002) BindingDB Entry DOI: 10.7270/Q2PC34K1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50219305 (CHEMBL347895) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 3.70 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description Inhibitory activity against Candida albicans (Nmt) assessed as inhibitory concentration | Bioorg Med Chem Lett 12: 607-10 (2002) BindingDB Entry DOI: 10.7270/Q2PC34K1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50219312 (CHEMBL158172) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 3.70 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description Inhibitory activity against Candida albicans (Nmt) assessed as inhibitory concentration (nM) | Bioorg Med Chem Lett 12: 607-10 (2002) BindingDB Entry DOI: 10.7270/Q2PC34K1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50109879 (CHEMBL155301 | Non peptidic, 4 | {3-[2-(2,3-Difluo...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 3.70 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description Inhibitory activity against Candida albicans N-Myristoyltransferase (CaNmt) assessed as inhibitory concentration using substrate peptide and myristot... | Bioorg Med Chem Lett 12: 607-10 (2002) BindingDB Entry DOI: 10.7270/Q2PC34K1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50219303 (CHEMBL345893) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 3.70 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description Inhibitory activity against Candida albicans (Nmt) assessed as inhibitory concentration (nM) | Bioorg Med Chem Lett 12: 607-10 (2002) BindingDB Entry DOI: 10.7270/Q2PC34K1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50219312 (CHEMBL158172) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 5.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description Inhibitory activity against Candida albicans N-Myristoyltransferase (CaNmt) assessed as inhibitory concentration using substrate peptide and myristot... | Bioorg Med Chem Lett 12: 607-10 (2002) BindingDB Entry DOI: 10.7270/Q2PC34K1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50109882 (3-(3-methyl-2-((2,3,4-trifluorophenoxy)methyl)benz...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Patents Similars | PubMed | n/a | n/a | 5.60 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description Inhibitory activity against Candida albicans Nmt (CaNmt) | Bioorg Med Chem Lett 13: 87-91 (2003) BindingDB Entry DOI: 10.7270/Q25D8V2K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50109882 (3-(3-methyl-2-((2,3,4-trifluorophenoxy)methyl)benz...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Patents Similars | PubMed | n/a | n/a | 5.70 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description Inhibitory activity against Candida albicans N-Myristoyltransferase (CaNmt) assessed as inhibitory concentration using substrate peptide and myristot... | Bioorg Med Chem Lett 12: 607-10 (2002) BindingDB Entry DOI: 10.7270/Q2PC34K1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50219303 (CHEMBL345893) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 7.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description Inhibitory activity against Candida albicans N-Myristoyltransferase (CaNmt) assessed as inhibitory concentration using substrate peptide and myristot... | Bioorg Med Chem Lett 12: 607-10 (2002) BindingDB Entry DOI: 10.7270/Q2PC34K1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50219305 (CHEMBL347895) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 8.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description Inhibitory activity against Candida albicans N-Myristoyltransferase (CaNmt) assessed as inhibitory concentration using substrate peptide and myristot... | Bioorg Med Chem Lett 12: 607-10 (2002) BindingDB Entry DOI: 10.7270/Q2PC34K1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50219310 (CHEMBL155469) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 9.40 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description Inhibitory activity against Candida albicans N-Myristoyltransferase (CaNmt) assessed as inhibitory concentration using substrate peptide and myristot... | Bioorg Med Chem Lett 12: 607-10 (2002) BindingDB Entry DOI: 10.7270/Q2PC34K1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50219308 (CHEMBL351774) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 17 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description Inhibitory activity against Candida albicans N-Myristoyltransferase (CaNmt) assessed as inhibitory concentration using substrate peptide and myristot... | Bioorg Med Chem Lett 12: 607-10 (2002) BindingDB Entry DOI: 10.7270/Q2PC34K1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50219309 (CHEMBL158185) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 28 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description Inhibitory activity against Candida albicans N-Myristoyltransferase (CaNmt) assessed as inhibitory concentration using substrate peptide and myristot... | Bioorg Med Chem Lett 12: 607-10 (2002) BindingDB Entry DOI: 10.7270/Q2PC34K1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50220564 (CHEMBL353541) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 43 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description In vitro inhibitory activity against Candida albicans Nmt (CaNmt) using substrate peptide GLTISKLFR-R-NH2 (0.5 uM) and myristoyl-CoA (0.5 uM) | Bioorg Med Chem Lett 13: 87-91 (2003) BindingDB Entry DOI: 10.7270/Q25D8V2K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50220566 (CHEMBL172471) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 47 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description Inhibitory activity against Candida albicans Nmt (CaNmt) using substrate peptide GLTISKLFR-R-NH2 (0.5 uM) and myristoyl-CoA (0.5 uM) | Bioorg Med Chem Lett 13: 87-91 (2003) BindingDB Entry DOI: 10.7270/Q25D8V2K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50220563 (CHEMBL353249) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | 62 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description Inhibitory activity against Candida albicans Nmt (CaNmt) using substrate peptide GLTISKLFR-R-NH2 (0.5 uM) and myristoyl-CoA (0.5 uM) | Bioorg Med Chem Lett 13: 87-91 (2003) BindingDB Entry DOI: 10.7270/Q25D8V2K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50219311 (CHEMBL346363) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 72 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description Inhibitory activity against Candida albicans N-Myristoyltransferase (CaNmt) assessed as inhibitory concentration using substrate peptide and myristot... | Bioorg Med Chem Lett 12: 607-10 (2002) BindingDB Entry DOI: 10.7270/Q2PC34K1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50219304 (CHEMBL433886) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 73 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description Inhibitory activity against Candida albicans N-Myristoyltransferase (CaNmt) assessed as inhibitory concentration using substrate peptide and myristot... | Bioorg Med Chem Lett 12: 607-10 (2002) BindingDB Entry DOI: 10.7270/Q2PC34K1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50220560 (CHEMBL173962) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 91 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description In vitro inhibitory activity against Candida albicans Nmt (CaNmt) using substrate peptide GLTISKLFR-R-NH2 (0.5 uM) and myristoyl-CoA (0.5 uM) | Bioorg Med Chem Lett 13: 87-91 (2003) BindingDB Entry DOI: 10.7270/Q25D8V2K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50101969 (3-Methyl-4-{3-[(pyridin-3-ylmethyl)-amino]-propoxy...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description Inhibitory activity against Candida albicans N-Myristoyltransferase (CaNmt) assessed as inhibitory concentration using substrate peptide and myristot... | Bioorg Med Chem Lett 12: 607-10 (2002) BindingDB Entry DOI: 10.7270/Q2PC34K1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50219306 (CHEMBL154079) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 110 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description Inhibitory activity against Candida albicans N-Myristoyltransferase (CaNmt) assessed as inhibitory concentration using substrate peptide and myristot... | Bioorg Med Chem Lett 12: 607-10 (2002) BindingDB Entry DOI: 10.7270/Q2PC34K1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50220569 (CHEMBL422896) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | 480 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description In vitro inhibitory activity against Aspergillus fumigatus Nmt (AfNmt) using substrate peptide GLTISKLFR-R-NH2 (0.5 uM) and myristoyl-CoA (0.5 uM) | Bioorg Med Chem Lett 13: 87-91 (2003) BindingDB Entry DOI: 10.7270/Q25D8V2K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50109886 (3-(3-methyl-2-(phenylthiomethyl)benzofuran-4-yloxy...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | PubMed | n/a | n/a | 620 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description Inhibitory activity against Candida albicans N-Myristoyltransferase (CaNmt) assessed as inhibitory concentration using substrate peptide and myristot... | Bioorg Med Chem Lett 12: 607-10 (2002) BindingDB Entry DOI: 10.7270/Q2PC34K1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50219307 (CHEMBL345610) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description Inhibitory activity against Candida albicans N-Myristoyltransferase (CaNmt) assessed as inhibitory concentration using substrate peptide and myristot... | Bioorg Med Chem Lett 12: 607-10 (2002) BindingDB Entry DOI: 10.7270/Q2PC34K1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50220570 (CHEMBL172455) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description Inhibitory activity against Candida albicans Nmt (CaNmt) using substrate peptide GLTISKLFR-R-NH2 (0.5 uM) and myristoyl-CoA (0.5 uM) | Bioorg Med Chem Lett 13: 87-91 (2003) BindingDB Entry DOI: 10.7270/Q25D8V2K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50220568 (CHEMBL368134) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | 1.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description In vitro inhibitory activity against Candida albicans Nmt (CaNmt) using substrate peptide GLTISKLFR-R-NH2 (0.5 uM) and myristoyl-CoA (0.5 uM) | Bioorg Med Chem Lett 13: 87-91 (2003) BindingDB Entry DOI: 10.7270/Q25D8V2K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50220567 (CHEMBL355170) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | 1.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description Inhibitory activity against Candida albicans Nmt (CaNmt) using substrate peptide GLTISKLFR-R-NH2 (0.5 uM) and myristoyl-CoA (0.5 uM) | Bioorg Med Chem Lett 13: 87-91 (2003) BindingDB Entry DOI: 10.7270/Q25D8V2K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50219302 (CHEMBL155240) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description Inhibitory activity against Candida albicans N-Myristoyltransferase (CaNmt) assessed as inhibitory concentration using substrate peptide and myristot... | Bioorg Med Chem Lett 12: 607-10 (2002) BindingDB Entry DOI: 10.7270/Q2PC34K1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50121716 ((3-methyl-4-(3-(pyridin-3-ylmethylamino)propoxy)be...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 4.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description In vitro inhibitory activity against aspergillus fumigatus Nmt (AfNmt) using substrate peptide GLTISKLFR-R-NH2 (0.5 uM) and myristoyl-CoA (0.5 uM) | Bioorg Med Chem Lett 13: 87-91 (2003) BindingDB Entry DOI: 10.7270/Q25D8V2K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50220565 (CHEMBL170524) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | 4.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description In vitro inhibitory activity against Aspergillus fumigatus Nmt (AfNmt) using substrate peptide GLTISKLFR-R-NH2 (0.5 uM) and myristoyl-CoA (0.5 uM) | Bioorg Med Chem Lett 13: 87-91 (2003) BindingDB Entry DOI: 10.7270/Q25D8V2K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50220562 (CHEMBL171506) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | 5.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description In vitro inhibitory activity against Aspergillus fumigatus Nmt (AfNmt) using substrate peptide GLTISKLFR-R-NH2 (0.5 uM) and myristoyl-CoA (0.5 uM) | Bioorg Med Chem Lett 13: 87-91 (2003) BindingDB Entry DOI: 10.7270/Q25D8V2K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50220564 (CHEMBL353541) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description In vitro inhibitory activity against Aspergillus fumigatus Nmt (AfNmt) using substrate peptide GLTISKLFR-R-NH2 (0.5 uM) and myristoyl-CoA (0.5 uM) | Bioorg Med Chem Lett 13: 87-91 (2003) BindingDB Entry DOI: 10.7270/Q25D8V2K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50219307 (CHEMBL345610) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description Inhibitory activity against human N-Myristoyltransferase (HsNmt) assessed as inhibitory concentration using substrate peptide and myristotyl-CoA at 0... | Bioorg Med Chem Lett 12: 607-10 (2002) BindingDB Entry DOI: 10.7270/Q2PC34K1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50220561 (CHEMBL173370) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description In vitro inhibitory activity against Aspergillus fumigatus Nmt (AfNmt) using substrate peptide GLTISKLFR-R-NH2 (0.5 uM) and myristoyl-CoA (0.5 uM) | Bioorg Med Chem Lett 13: 87-91 (2003) BindingDB Entry DOI: 10.7270/Q25D8V2K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50220559 (CHEMBL422746) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description In vitro inhibitory activity against Aspergillus fumigatus Nmt (AfNmt) using substrate peptide GLTISKLFR-R-NH2 (0.5 uM) and myristoyl-CoA (0.5 uM) | Bioorg Med Chem Lett 13: 87-91 (2003) BindingDB Entry DOI: 10.7270/Q25D8V2K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50219308 (CHEMBL351774) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.90E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description Inhibitory activity against human N-Myristoyltransferase (HsNmt) assessed as inhibitory concentration using substrate peptide and myristotyl-CoA at 0... | Bioorg Med Chem Lett 12: 607-10 (2002) BindingDB Entry DOI: 10.7270/Q2PC34K1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50220560 (CHEMBL173962) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description In vitro inhibitory activity against human Nmt (HsNmt) using 0.5 uM peptide GNAASAR-R-NH2 and 0.5 uM myristoyl-CoA | Bioorg Med Chem Lett 13: 87-91 (2003) BindingDB Entry DOI: 10.7270/Q25D8V2K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50121720 ((1-METHYL-1H-IMIDAZOL-2-YL)-(3-METHYL-4-{3-[(PYRID...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL DrugBank MMDB PC cid PC sid PDB UniChem Similars | PubMed | n/a | n/a | 3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description In vitro inhibitory activity against Aspergillus fumigatus Nmt (AfNmt) using substrate peptide GLTISKLFR-R-NH2 (0.5 uM) and myristoyl-CoA (0.5 uM) | Bioorg Med Chem Lett 13: 87-91 (2003) BindingDB Entry DOI: 10.7270/Q25D8V2K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50220571 (CHEMBL355250) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | 4.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description In vitro inhibitory activity against Aspergillus fumigatus Nmt (AfNmt) using substrate peptide GLTISKLFR-R-NH2 (0.5 uM) and myristoyl-CoA (0.5 uM) | Bioorg Med Chem Lett 13: 87-91 (2003) BindingDB Entry DOI: 10.7270/Q25D8V2K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glycylpeptide N-tetradecanoyltransferase 1/2 (Homo sapiens (Human)) | BDBM50109879 (CHEMBL155301 | Non peptidic, 4 | {3-[2-(2,3-Difluo...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 6.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Nippon Roche Research Center Curated by ChEMBL | Assay Description Inhibitory activity against human N-Myristoyltransferase (HsNmt) assessed as inhibitory concentration using substrate peptide and myristotyl-CoA at 0... | Bioorg Med Chem Lett 12: 607-10 (2002) BindingDB Entry DOI: 10.7270/Q2PC34K1 | |||||||||||
More data for this Ligand-Target Pair |
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