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Compile Data Set for Download or QSAR

Found 32 hits with Last Name = 'lloyd' and Initial = 'jh'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Translocator protein


(Homo sapiens (Human))
BDBM50556264
PNG
(CHEMBL4789235)
Show SMILES CCN(Cc1ccccc1)C(=O)Cc1c(nn2c(C)cc(C)nc12)-c1ccc(OC)cc1
KEGG

UniProtKB/SwissProt

DrugBank
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GoogleScholar
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PC sid
UniChem
Article
PubMed
6.20n/an/an/an/an/an/an/an/a


TBA

Assay Description
Displacement of [3H]-PK11195 from wild type TSPO (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 90 m...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112725
BindingDB Entry DOI: 10.7270/Q2VM4GZF
More data for this
Ligand-Target Pair
Translocator protein


(Homo sapiens (Human))
BDBM50556263
PNG
(CHEMBL4742003)
Show SMILES COc1ccc(cc1)-c1nn2c(C)cc(C)nc2c1CC(=O)N(C)Cc1ccccc1
KEGG

UniProtKB/SwissProt

DrugBank
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GoogleScholar
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UniChem
Article
PubMed
9.30n/an/an/an/an/an/an/an/a


TBA

Assay Description
Displacement of [3H]-PK11195 from wild type TSPO (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 90 m...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112725
BindingDB Entry DOI: 10.7270/Q2VM4GZF
More data for this
Ligand-Target Pair
Translocator protein


(Homo sapiens (Human))
BDBM50556271
PNG
(CHEMBL4742171)
Show SMILES CCN(Cc1ccccc1)C(=O)CN1c2ccccc2NC(=O)c2ccccc12
KEGG

UniProtKB/SwissProt

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UniChem
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16n/an/an/an/an/an/an/an/a


TBA

Assay Description
Displacement of [3H]-PK11195 from wild type TSPO (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 90 m...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112725
BindingDB Entry DOI: 10.7270/Q2VM4GZF
More data for this
Ligand-Target Pair
Translocator protein


(Homo sapiens (Human))
BDBM50327238
PNG
(2-[2-(4'-Methoxyphenyl)-5,7-dimethylpyrazolo[1,5-a...)
Show SMILES CCN(CC)C(=O)Cc1c(nn2c(C)cc(C)nc12)-c1ccc(OC)cc1
Show InChI InChI=1S/C21H26N4O2/c1-6-24(7-2)19(26)13-18-20(16-8-10-17(27-5)11-9-16)23-25-15(4)12-14(3)22-21(18)25/h8-12H,6-7,13H2,1-5H3
KEGG

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Article
PubMed
20n/an/an/an/an/an/an/an/a


TBA

Assay Description
Displacement of [3H]-PK11195 from wild type TSPO (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 90 m...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112725
BindingDB Entry DOI: 10.7270/Q2VM4GZF
More data for this
Ligand-Target Pair
Translocator protein


(Homo sapiens (Human))
BDBM50556263
PNG
(CHEMBL4742003)
Show SMILES COc1ccc(cc1)-c1nn2c(C)cc(C)nc2c1CC(=O)N(C)Cc1ccccc1
KEGG

UniProtKB/SwissProt

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UniChem
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27n/an/an/an/an/an/an/an/a


TBA

Assay Description
Displacement of [3H]-PK11195 from TSPO A147T mutant (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 9...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112725
BindingDB Entry DOI: 10.7270/Q2VM4GZF
More data for this
Ligand-Target Pair
Translocator protein


(Homo sapiens (Human))
BDBM50509034
PNG
(CHEMBL4173118)
Show SMILES CCN(CC)C(=O)Cn1c2ccccc2c2ccccc12
Show InChI InChI=1S/C18H20N2O/c1-3-19(4-2)18(21)13-20-16-11-7-5-9-14(16)15-10-6-8-12-17(15)20/h5-12H,3-4,13H2,1-2H3
KEGG

UniProtKB/SwissProt

DrugBank
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UniChem
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30n/an/an/an/an/an/an/an/a


TBA

Assay Description
Displacement of [3H]-PK11195 from wild type TSPO (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 90 m...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112725
BindingDB Entry DOI: 10.7270/Q2VM4GZF
More data for this
Ligand-Target Pair
Translocator protein


(Homo sapiens (Human))
BDBM50556267
PNG
(CHEMBL4745926)
Show SMILES CCN(Cc1ccccc1)C(=O)CN1Cc2cnn(C)c2Nc2ccccc12
KEGG

UniProtKB/SwissProt

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41n/an/an/an/an/an/an/an/a


TBA

Assay Description
Displacement of [3H]-PK11195 from wild type TSPO (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 90 m...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112725
BindingDB Entry DOI: 10.7270/Q2VM4GZF
More data for this
Ligand-Target Pair
Translocator protein


(Homo sapiens (Human))
BDBM50556266
PNG
(CHEMBL4758934)
Show SMILES CN(Cc1ccccc1)C(=O)CN1Cc2cnn(C)c2Nc2ccccc12
KEGG

UniProtKB/SwissProt

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41n/an/an/an/an/an/an/an/a


TBA

Assay Description
Displacement of [3H]-PK11195 from wild type TSPO (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 90 m...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112725
BindingDB Entry DOI: 10.7270/Q2VM4GZF
More data for this
Ligand-Target Pair
Translocator protein


(Homo sapiens (Human))
BDBM50509039
PNG
(CHEMBL4447335)
Show SMILES CN(Cc1ccccc1)C(=O)Cn1c2ccccc2c2ccccc12
Show InChI InChI=1S/C22H20N2O/c1-23(15-17-9-3-2-4-10-17)22(25)16-24-20-13-7-5-11-18(20)19-12-6-8-14-21(19)24/h2-14H,15-16H2,1H3
KEGG

UniProtKB/SwissProt

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UniChem
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53n/an/an/an/an/an/an/an/a


TBA

Assay Description
Displacement of [3H]-PK11195 from wild type TSPO (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 90 m...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112725
BindingDB Entry DOI: 10.7270/Q2VM4GZF
More data for this
Ligand-Target Pair
Translocator protein


(Homo sapiens (Human))
BDBM50556270
PNG
(CHEMBL4743573)
Show SMILES CN(Cc1ccccc1)C(=O)CN1c2ccccc2NC(=O)c2ccccc12
KEGG

UniProtKB/SwissProt

DrugBank
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UniChem
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PubMed
77n/an/an/an/an/an/an/an/a


TBA

Assay Description
Displacement of [3H]-PK11195 from wild type TSPO (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 90 m...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112725
BindingDB Entry DOI: 10.7270/Q2VM4GZF
More data for this
Ligand-Target Pair
Translocator protein


(Homo sapiens (Human))
BDBM50556264
PNG
(CHEMBL4789235)
Show SMILES CCN(Cc1ccccc1)C(=O)Cc1c(nn2c(C)cc(C)nc12)-c1ccc(OC)cc1
KEGG

UniProtKB/SwissProt

DrugBank
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GoogleScholar
AffyNet 
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PC sid
UniChem
Article
PubMed
81n/an/an/an/an/an/an/an/a


TBA

Assay Description
Displacement of [3H]-PK11195 from TSPO A147T mutant (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 9...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112725
BindingDB Entry DOI: 10.7270/Q2VM4GZF
More data for this
Ligand-Target Pair
Translocator protein


(Homo sapiens (Human))
BDBM50509028
PNG
(CHEMBL4161842)
Show SMILES CCN(Cc1ccccc1)C(=O)Cn1c2ccccc2c2ccccc12
Show InChI InChI=1S/C23H22N2O/c1-2-24(16-18-10-4-3-5-11-18)23(26)17-25-21-14-8-6-12-19(21)20-13-7-9-15-22(20)25/h3-15H,2,16-17H2,1H3
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
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UniChem
Article
PubMed
92n/an/an/an/an/an/an/an/a


TBA

Assay Description
Displacement of [3H]-PK11195 from wild type TSPO (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 90 m...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112725
BindingDB Entry DOI: 10.7270/Q2VM4GZF
More data for this
Ligand-Target Pair
Translocator protein


(Homo sapiens (Human))
BDBM50556271
PNG
(CHEMBL4742171)
Show SMILES CCN(Cc1ccccc1)C(=O)CN1c2ccccc2NC(=O)c2ccccc12
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
99n/an/an/an/an/an/an/an/a


TBA

Assay Description
Displacement of [3H]-PK11195 from TSPO A147T mutant (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 9...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112725
BindingDB Entry DOI: 10.7270/Q2VM4GZF
More data for this
Ligand-Target Pair
Translocator protein


(Homo sapiens (Human))
BDBM50327238
PNG
(2-[2-(4'-Methoxyphenyl)-5,7-dimethylpyrazolo[1,5-a...)
Show SMILES CCN(CC)C(=O)Cc1c(nn2c(C)cc(C)nc12)-c1ccc(OC)cc1
Show InChI InChI=1S/C21H26N4O2/c1-6-24(7-2)19(26)13-18-20(16-8-10-17(27-5)11-9-16)23-25-15(4)12-14(3)22-21(18)25/h8-12H,6-7,13H2,1-5H3
KEGG

UniProtKB/SwissProt

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CHEMBL
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Article
PubMed
99n/an/an/an/an/an/an/an/a


TBA

Assay Description
Displacement of [3H]-PK11195 from TSPO A147T mutant (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 9...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112725
BindingDB Entry DOI: 10.7270/Q2VM4GZF
More data for this
Ligand-Target Pair
Translocator protein


(Homo sapiens (Human))
BDBM50509039
PNG
(CHEMBL4447335)
Show SMILES CN(Cc1ccccc1)C(=O)Cn1c2ccccc2c2ccccc12
Show InChI InChI=1S/C22H20N2O/c1-23(15-17-9-3-2-4-10-17)22(25)16-24-20-13-7-5-11-18(20)19-12-6-8-14-21(19)24/h2-14H,15-16H2,1H3
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
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UniChem
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PubMed
132n/an/an/an/an/an/an/an/a


TBA

Assay Description
Displacement of [3H]-PK11195 from TSPO A147T mutant (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 9...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112725
BindingDB Entry DOI: 10.7270/Q2VM4GZF
More data for this
Ligand-Target Pair
Translocator protein


(Homo sapiens (Human))
BDBM50556270
PNG
(CHEMBL4743573)
Show SMILES CN(Cc1ccccc1)C(=O)CN1c2ccccc2NC(=O)c2ccccc12
KEGG

UniProtKB/SwissProt

DrugBank
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GoogleScholar
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UniChem
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PubMed
159n/an/an/an/an/an/an/an/a


TBA

Assay Description
Displacement of [3H]-PK11195 from TSPO A147T mutant (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 9...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112725
BindingDB Entry DOI: 10.7270/Q2VM4GZF
More data for this
Ligand-Target Pair
Translocator protein


(Homo sapiens (Human))
BDBM50509034
PNG
(CHEMBL4173118)
Show SMILES CCN(CC)C(=O)Cn1c2ccccc2c2ccccc12
Show InChI InChI=1S/C18H20N2O/c1-3-19(4-2)18(21)13-20-16-11-7-5-9-14(16)15-10-6-8-12-17(15)20/h5-12H,3-4,13H2,1-2H3
KEGG

UniProtKB/SwissProt

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UniChem
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177n/an/an/an/an/an/an/an/a


TBA

Assay Description
Displacement of [3H]-PK11195 from TSPO A147T mutant (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 9...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112725
BindingDB Entry DOI: 10.7270/Q2VM4GZF
More data for this
Ligand-Target Pair
Translocator protein


(Homo sapiens (Human))
BDBM50556266
PNG
(CHEMBL4758934)
Show SMILES CN(Cc1ccccc1)C(=O)CN1Cc2cnn(C)c2Nc2ccccc12
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
200n/an/an/an/an/an/an/an/a


TBA

Assay Description
Displacement of [3H]-PK11195 from TSPO A147T mutant (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 9...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112725
BindingDB Entry DOI: 10.7270/Q2VM4GZF
More data for this
Ligand-Target Pair
Translocator protein


(Homo sapiens (Human))
BDBM50556272
PNG
(CHEMBL4793373)
Show SMILES CCN(CC)C(=O)CN1c2ccccc2NC(=O)c2ccccc12
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
201n/an/an/an/an/an/an/an/a


TBA

Assay Description
Displacement of [3H]-PK11195 from wild type TSPO (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 90 m...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112725
BindingDB Entry DOI: 10.7270/Q2VM4GZF
More data for this
Ligand-Target Pair
Translocator protein


(Homo sapiens (Human))
BDBM50556267
PNG
(CHEMBL4745926)
Show SMILES CCN(Cc1ccccc1)C(=O)CN1Cc2cnn(C)c2Nc2ccccc12
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
227n/an/an/an/an/an/an/an/a


TBA

Assay Description
Displacement of [3H]-PK11195 from TSPO A147T mutant (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 9...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112725
BindingDB Entry DOI: 10.7270/Q2VM4GZF
More data for this
Ligand-Target Pair
Translocator protein


(Homo sapiens (Human))
BDBM50556265
PNG
(CHEMBL4753783)
Show SMILES COc1ccc(cc1)-c1nn2c(C)cc(C)nc2c1CC(=O)N(C)C
KEGG

UniProtKB/SwissProt

DrugBank
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GoogleScholar
AffyNet 
PC cid
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UniChem
Article
PubMed
338n/an/an/an/an/an/an/an/a


TBA

Assay Description
Displacement of [3H]-PK11195 from wild type TSPO (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 90 m...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112725
BindingDB Entry DOI: 10.7270/Q2VM4GZF
More data for this
Ligand-Target Pair
Translocator protein


(Homo sapiens (Human))
BDBM50509028
PNG
(CHEMBL4161842)
Show SMILES CCN(Cc1ccccc1)C(=O)Cn1c2ccccc2c2ccccc12
Show InChI InChI=1S/C23H22N2O/c1-2-24(16-18-10-4-3-5-11-18)23(26)17-25-21-14-8-6-12-19(21)20-13-7-9-15-22(20)25/h3-15H,2,16-17H2,1H3
KEGG

UniProtKB/SwissProt

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UniChem
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460n/an/an/an/an/an/an/an/a


TBA

Assay Description
Displacement of [3H]-PK11195 from TSPO A147T mutant (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 9...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112725
BindingDB Entry DOI: 10.7270/Q2VM4GZF
More data for this
Ligand-Target Pair
Translocator protein


(Homo sapiens (Human))
BDBM50556268
PNG
(CHEMBL4750743)
Show SMILES CCN(CC)C(=O)CN1Cc2cnn(C)c2Nc2ccccc12
KEGG

UniProtKB/SwissProt

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GoogleScholar
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PubMed
493n/an/an/an/an/an/an/an/a


TBA

Assay Description
Displacement of [3H]-PK11195 from wild type TSPO (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 90 m...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112725
BindingDB Entry DOI: 10.7270/Q2VM4GZF
More data for this
Ligand-Target Pair
Translocator protein


(Homo sapiens (Human))
BDBM50556265
PNG
(CHEMBL4753783)
Show SMILES COc1ccc(cc1)-c1nn2c(C)cc(C)nc2c1CC(=O)N(C)C
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
560n/an/an/an/an/an/an/an/a


TBA

Assay Description
Displacement of [3H]-PK11195 from TSPO A147T mutant (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 9...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112725
BindingDB Entry DOI: 10.7270/Q2VM4GZF
More data for this
Ligand-Target Pair
Translocator protein


(Homo sapiens (Human))
BDBM50556268
PNG
(CHEMBL4750743)
Show SMILES CCN(CC)C(=O)CN1Cc2cnn(C)c2Nc2ccccc12
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
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PC sid
UniChem
Article
PubMed
2.26E+3n/an/an/an/an/an/an/an/a


TBA

Assay Description
Displacement of [3H]-PK11195 from TSPO A147T mutant (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 9...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112725
BindingDB Entry DOI: 10.7270/Q2VM4GZF
More data for this
Ligand-Target Pair
Translocator protein


(Homo sapiens (Human))
BDBM50556272
PNG
(CHEMBL4793373)
Show SMILES CCN(CC)C(=O)CN1c2ccccc2NC(=O)c2ccccc12
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
2.36E+3n/an/an/an/an/an/an/an/a


TBA

Assay Description
Displacement of [3H]-PK11195 from TSPO A147T mutant (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 9...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112725
BindingDB Entry DOI: 10.7270/Q2VM4GZF
More data for this
Ligand-Target Pair
Translocator protein


(Homo sapiens (Human))
BDBM50509044
PNG
(CHEMBL4451744)
Show SMILES CN(C)C(=O)Cn1c2ccccc2c2ccccc12
Show InChI InChI=1S/C16H16N2O/c1-17(2)16(19)11-18-14-9-5-3-7-12(14)13-8-4-6-10-15(13)18/h3-10H,11H2,1-2H3
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
>1.00E+4n/an/an/an/an/an/an/an/a


TBA

Assay Description
Displacement of [3H]-PK11195 from TSPO A147T mutant (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 9...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112725
BindingDB Entry DOI: 10.7270/Q2VM4GZF
More data for this
Ligand-Target Pair
Translocator protein


(Homo sapiens (Human))
BDBM50556273
PNG
(CHEMBL4761316)
Show SMILES CN(C)C(=O)CN1c2ccccc2NC(=O)c2ccccc12
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
>1.00E+4n/an/an/an/an/an/an/an/a


TBA

Assay Description
Displacement of [3H]-PK11195 from wild type TSPO (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 90 m...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112725
BindingDB Entry DOI: 10.7270/Q2VM4GZF
More data for this
Ligand-Target Pair
Translocator protein


(Homo sapiens (Human))
BDBM50556273
PNG
(CHEMBL4761316)
Show SMILES CN(C)C(=O)CN1c2ccccc2NC(=O)c2ccccc12
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
>1.00E+4n/an/an/an/an/an/an/an/a


TBA

Assay Description
Displacement of [3H]-PK11195 from TSPO A147T mutant (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 9...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112725
BindingDB Entry DOI: 10.7270/Q2VM4GZF
More data for this
Ligand-Target Pair
Translocator protein


(Homo sapiens (Human))
BDBM50509044
PNG
(CHEMBL4451744)
Show SMILES CN(C)C(=O)Cn1c2ccccc2c2ccccc12
Show InChI InChI=1S/C16H16N2O/c1-17(2)16(19)11-18-14-9-5-3-7-12(14)13-8-4-6-10-15(13)18/h3-10H,11H2,1-2H3
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
>1.00E+4n/an/an/an/an/an/an/an/a


TBA

Assay Description
Displacement of [3H]-PK11195 from wild type TSPO (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 90 m...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112725
BindingDB Entry DOI: 10.7270/Q2VM4GZF
More data for this
Ligand-Target Pair
Translocator protein


(Homo sapiens (Human))
BDBM50556269
PNG
(CHEMBL4792527)
Show SMILES CN(C)C(=O)CN1Cc2cnn(C)c2Nc2ccccc12
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
>1.00E+4n/an/an/an/an/an/an/an/a


TBA

Assay Description
Displacement of [3H]-PK11195 from TSPO A147T mutant (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 9...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112725
BindingDB Entry DOI: 10.7270/Q2VM4GZF
More data for this
Ligand-Target Pair
Translocator protein


(Homo sapiens (Human))
BDBM50556269
PNG
(CHEMBL4792527)
Show SMILES CN(C)C(=O)CN1Cc2cnn(C)c2Nc2ccccc12
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
>1.00E+4n/an/an/an/an/an/an/an/a


TBA

Assay Description
Displacement of [3H]-PK11195 from wild type TSPO (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 90 m...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112725
BindingDB Entry DOI: 10.7270/Q2VM4GZF
More data for this
Ligand-Target Pair