Compile Data Set for Download or QSAR

Found 1057 hits with Last Name = 'querolle' and Initial = 'oa'   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM523659 (US11136311, Compound 149) Show SMILES CN(C)C(=O)c1sc(Nc2nccc(n2)-c2cc3c(NC[C@]3(C)CO)c(c2)C#N)nc1C |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	0.700	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2J106BW
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM527664 (US11186589, Compound 30) Show SMILES CN1CCc2cc(Nc3nccc(n3)-c3cc4c(NC[C@]4(C)CO)c(c3)C#N)ccc2C1 |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	0.800	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2X06B7J
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM523658 (US11136311, Compound 148) Show SMILES Cc1nc(Nc2nccc(n2)-c2cc3c(NC[C@]3(C)CO)c(c2)C#N)sc1C |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	0.800	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2J106BW
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM523642 (US11136311, Compound 132) Show SMILES Cc1nn(CC(F)F)cc1Nc1nccc(n1)-c1cc2c(NC[C@]2(C)CO)c(c1)C#N |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	1	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2J106BW
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM527687 (US11186589, Compound 3b) Show SMILES CN1CCn2ncc(Nc3nccc(n3)-c3cc4c(NC[C@]4(C)CO)c(c3)C#N)c2C1=O |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	1	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2X06B7J
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM527662 (US11186589, Compound 28) Show SMILES Cc1nc2CCOCc2cc1Nc1nccc(n1)-c1cc2c(NC[C@]2(C)CO)c(c1)C#N |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	1.10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2X06B7J
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM523713 (US11136311, Compound 204) Show SMILES CC(C)c1nn(CC(F)F)cc1Nc1nccc(n1)-c1cc2c(NC[C@]2(C)CO)c(c1)C#N |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	1.10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2J106BW
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM523587 (US11136311, Compound 76) Show SMILES Cc1c(Nc2nccc(n2)-c2cc3c(NC[C@]3(C)CO)c(c2)C#N)cnn1CC1CCOCC1 |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	1.20	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2J106BW
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM523656 (US11136311, Compound 146) Show SMILES Cc1nscc1Nc1nccc(n1)-c1cc2c(NC[C@]2(C)CO)c(c1)C#N |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	1.30	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2J106BW
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM527642 (US11186589, Compound 13) Show SMILES CN(C)CC(=O)N1CCc2c1cc(Cl)cc2Nc1nccc(n1)-c1cc2c(NC[C@]2(C)CO)c(c1)C#N |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	1.30	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2X06B7J
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM523653 (US11136311, Compound 143) Show SMILES Cn1ccc(Nc2ncc(F)c(n2)-c2cc3c(NCC3(C)CO)c(c2)C#N)n1 Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	1.30	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2J106BW
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM527666 (US11186589, Compound 31) Show SMILES CN1CCc2ccc(Nc3nccc(n3)-c3cc4c(NC[C@]4(C)CO)c(c3)C#N)cc2C1 |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	1.40	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2X06B7J
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM527628 (US11186589, Compound 3) Show SMILES CN1CCc2ccc(Nc3nccc(n3)-c3cc4c(NCC4(C)CO)c(c3)C#N)cc2CC1 Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	1.40	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2X06B7J
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM523655 (US11136311, Compound 145) Show SMILES Cc1csc(Nc2nccc(n2)-c2cc3c(NC[C@]3(C)CO)c(c2)C#N)n1 |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	1.5	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2J106BW
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM523569 (US11136311, Compound 58) Show SMILES COC(C)(C)CCn1nc(Nc2nccc(n2)-c2cc3c(NC[C@]3(C)CO)c(c2)C#N)cc1C |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	1.5	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2J106BW
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM527696 (US11186589, Compound 12b) Show SMILES C[C@]1(CO)CNc2c1cc(cc2C#N)-c1ccnc(Nc2cnn3CCOCc23)n1 |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	1.5	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2X06B7J
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM527648 (US11186589, Compound 16) Show SMILES CN(C)CC(=O)N1CCc2c1c(Cl)cc(Nc1nccc(n1)-c1cc3c(NC[C@]3(C)CO)c(c1)C#N)c2C |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	1.60	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2X06B7J
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM523607 (US11136311, Compound 96) Show SMILES Cc1cc(Nc2nccc(n2)-c2cc3c(NC[C@]3(C)CO)c(c2)C#N)n(CCC2CC2)n1 |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	1.60	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2J106BW
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM523606 (US11136311, Compound 95) Show SMILES Cc1cc(Nc2nccc(n2)-c2cc3c(NC[C@]3(C)CO)c(c2)C#N)nn1CCC1CC1 |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	1.60	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2J106BW
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM523578 (US11136311, Compound 67) Show SMILES Cn1nc(cc1Nc1nccc(n1)-c1cc2c(NC[C@]2(C)CO)c(c1)C#N)C1CCOCC1 |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	1.60	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2J106BW
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM523633 (US11136311, Compound 123) Show SMILES CN1CCC(CC1)n1ncc(Nc2nccc(n2)-c2cc3c(NC[C@]3(C)CO)c(c2)C#N)c1C |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	1.60	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2J106BW
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM527670 (US11186589, Compound 48) Show SMILES Cn1c2CCOCc2cc(Nc2nccc(n2)-c2cc3c(NC[C@]3(C)CO)c(c2)C#N)c1=O |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	1.60	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2X06B7J
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM523691 (US11136311, Compound 182) Show SMILES Cc1cc(Nc2nccc(n2)-c2cc3c(NC[C@]3(C)CO)c(c2)C#N)nn1CCN1CCOCC1 |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	1.70	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2J106BW
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM527667 (US11186589, Compound 32 | US11186589, Compound 32b) Show SMILES CC1OCCn2nc(Nc3nccc(n3)-c3cc4c(NCC4(C)C)c(c3)C#N)cc12 Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	1.70	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2X06B7J
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM527659 (US11186589, Compound 25) Show SMILES COc1nc2CCOCc2cc1Nc1nccc(n1)-c1cc2c(NC[C@]2(C)CO)c(c1)C#N |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	1.70	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2X06B7J
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM527675 (US11186589, Compound 53) Show SMILES COc1nc2CN(C)CCc2cc1Nc1nccc(n1)-c1cc2c(NC[C@]2(C)CO)c(c1)C#N |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	1.80	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2X06B7J
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM527630 (US11186589, Compound 5 | US11186589, Compound 8) Show SMILES CC1(CO)CNc2c1cc(cc2C#N)-c1ccnc(Nc2ccc3COC(CO)Cc3c2)n1 Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	1.90	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2X06B7J
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM523584 (US11136311, Compound 73) Show SMILES Cc1cc(Nc2nccc(n2)-c2cc3c(NC[C@]3(C)CO)c(c2)C#N)n(CC=C)n1 |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	1.90	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2J106BW
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM523575 (US11136311, Compound 64) Show SMILES Cn1cc(Nc2nccc(n2)-c2cc3c(NC[C@]3(C)CO)c(c2)C#N)c(n1)C(F)(F)F |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	1.90	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2J106BW
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM523654 (US11136311, Compound 144) Show SMILES Cn1ccc(Nc2ncc(F)c(n2)-c2cc3c(NC[C@]3(C)CO)c(c2)C#N)n1 |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	2	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2J106BW
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM523661 (US11136311, Compound 151) Show SMILES CC(C)Cn1nc(CO)cc1Nc1nccc(n1)-c1cc2c(NC[C@]2(C)CO)c(c1)C#N |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	2	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2J106BW
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM523548 (US11136311, Compound 37) Show SMILES CN1CCC(CC1)n1ccc(Nc2nccc(n2)-c2cc3c(NC[C@]3(C)CO)c(c2)C#N)n1 |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	2	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2J106BW
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM523571 (US11136311, Compound 60) Show SMILES Cc1cc(Nc2nccc(n2)-c2cc3c(NC[C@]3(C)CO)c(c2)C#N)nn1CC1CCOCC1 |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	2	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2J106BW
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM523717 (US11136311, Compound 208) Show SMILES C[C@]1(CO)CNc2c1cc(cc2C#N)-c1ccnc(Nc2cnn(CCN3CCOCC3)c2Cl)n1 |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	2	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2J106BW
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM523608 (US11136311, Compound 97) Show SMILES CC(C)Cc1nn(C)cc1Nc1nccc(n1)-c1cc2c(NC[C@]2(C)CO)c(c1)C#N |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	2	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2J106BW
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM523609 (US11136311, Compound 98) Show SMILES CC(C)Cc1c(Nc2nccc(n2)-c2cc3c(NC[C@]3(C)CO)c(c2)C#N)cnn1C |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	2	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2J106BW
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM523637 (US11136311, Compound 127) Show SMILES CC(C)CCc1c(Nc2nccc(n2)-c2cc3c(NC[C@]3(C)CO)c(c2)C#N)cnn1CCO |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	2	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2J106BW
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM527626 (US11186589, Compound 1 | US11186589, Compound 1b |...) Show SMILES CC1CCn2ncc(Nc3nccc(n3)-c3cc4c(NC[C@]4(C)CO)c(c3)C#N)c2O1 |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	2	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2X06B7J
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM527697 (US11186589, Compound 13b) Show SMILES CN1CCn2nc(Nc3nccc(n3)-c3cc4c(NC[C@]4(C)CO)c(c3)C#N)cc2C1=O |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	2	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2X06B7J
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM527698 (US11186589, Compound 14b) Show SMILES C[C@]1(CO)CNc2c1cc(cc2C#N)-c1ccnc(Nc2cnn3CCCOc23)n1 |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	2	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2X06B7J
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM527630 (US11186589, Compound 5 | US11186589, Compound 8) Show SMILES CC1(CO)CNc2c1cc(cc2C#N)-c1ccnc(Nc2ccc3COC(CO)Cc3c2)n1 Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	2	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2X06B7J
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM527637 (US11186589, Compound 9 | US11186589, Compound 9c) Show SMILES CC(=O)N1CCc2c1c(Cl)cc(Nc1nccc(n1)-c1cc3c(NCC3(C)CO)c(c1)C#N)c2C Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	2	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2X06B7J
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM523552 (US11136311, Compound 41) Show SMILES Cn1nc(Cl)cc1Nc1nccc(n1)-c1cc2c(NC[C@]2(C)CO)c(c1)C#N |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	2.10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2J106BW
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM523611 (US11136311, Compound 100) Show SMILES CC(C)CCc1nn(C)cc1Nc1nccc(n1)-c1cc2c(NC[C@]2(C)CO)c(c1)C#N |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	2.10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2J106BW
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM523706 (US11136311, Compound 197) Show SMILES CNC(=O)c1cc(Nc2nccc(n2)-c2cc3c(NC[C@]3(C)CO)c(c2)C#N)nn1CC(F)F |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	2.10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2J106BW
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM523551 (US11136311, Compound 40) Show SMILES C[C@]1(CO)CNc2c1cc(cc2C#N)-c1ccnc(Nc2ccn(CC3CC3)n2)n1 |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	2.20	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2J106BW
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM523714 (US11136311, Compound 205) Show SMILES C[C@]1(CO)CNc2c1cc(cc2C#N)-c1ccnc(Nc2cn(CC(F)F)nc2C2CC2)n1 |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	2.20	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2J106BW
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM523530 (US11136311, Compound 19) Show SMILES Cn1ccc(Nc2nccc(n2)-c2cc3c(NC[C@]3(C)CO)c(c2)C#N)n1 |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	2.20	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2J106BW
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM523613 (US11136311, Compound 102) Show SMILES CC(C)CCc1c(Nc2nccc(n2)-c2cc3c(NC[C@]3(C)CO)c(c2)C#N)cnn1CCC(C)C |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	2.20	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2J106BW
					More data for this Ligand-Target Pair
Mitogen-activated protein kinase kinase kinase 14 (Homo sapiens (Human))	BDBM523680 (US11136311, Compound 170) Show SMILES Cc1c(Nc2nccc(n2)-c2cc3c(NC[C@]3(C)CO)c(c2)C#N)cnn1CCN1CCOCC1 |r| Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	2.20	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreen® (αscreen) format (Perkin Elmer). All compounds tested were dissolv...				Citation and Details BindingDB Entry DOI: 10.7270/Q2J106BW
					More data for this Ligand-Target Pair

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