Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
5-hydroxytryptamine receptor 3A (RAT) | BDBM50007871 (CHEMBL8197 | ICS 205-930 | TROPISETRON) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL KEGG PC cid PC sid PDB UniChem Patents Similars | PDB Article PubMed | 2.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by PDSP Ki Database | Naunyn Schmiedebergs Arch Pharmacol 345: 264-9 (1992) Article DOI: 10.1007/bf00168685 BindingDB Entry DOI: 10.7270/Q2P55KZ1 | ||||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) |